Beilstein Journal of Organic Chemistry

Article	Citations
Synthetic reactions driven by electron-donor–acceptor (EDA) complexes	116
19F NMR as a tool in chemical biology	62
Chemical approaches to discover the full potential of peptide nucleic acids in biomedical applications	47
Development of N-F fluorinating agents and their fluorinations: Historical perspective	45
A comprehensive review of flow chemistry techniques tailored to the flavours and fragrances industries	44
Valorisation of plastic waste via metal-catalysed depolymerisation	38
A recent overview on the synthesis of 1,4,5-trisubstituted 1,2,3-triazoles	33
The preparation and properties of 1,1-difluorocyclopropane derivatives	33
Microwave-assisted multicomponent reactions in heterocyclic chemistry and mechanistic aspects	33
Prins cyclization-mediated stereoselective synthesis of tetrahydropyrans and dihydropyrans: an inspection of twenty years	30
Cryogels: recent applications in 3D-bioprinting, injectable cryogels, drug delivery, and wound healing	28
Recent advances in organocatalytic asymmetric aza-Michael reactions of amines and amides	26
Recent advances in the tandem annulation of 1,3-enynes to functionalized pyridine and pyrrole derivatives	25
Photoredox catalysis in nickel-catalyzed C–H functionalization	25
Visible-light-mediated copper photocatalysis for organic syntheses	24
Progress and challenges in the synthesis of sequence controlled polysaccharides	23
N-tert-Butanesulfinyl imines in the asymmetric synthesis of nitrogen-containing heterocycles	23
Secondary metabolites of Bacillus subtilis impact the assembly of soil-derived semisynthetic bacterial communities	22
Beyond ribose and phosphate: Selected nucleic acid modifications for structure–function investigations and therapeutic applications	22
Amine–borane complex-initiated SF5Cl radical addition on alkenes and alkynes	22
Insight into functionalized-macrocycles-guided supramolecular photocatalysis	20
Enhanced target cell specificity and uptake of lipid nanoparticles using RNA aptamers and peptides	20
Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes	19
Using multiple self-sorting for switching functions in discrete multicomponent systems	19
Biochemistry of fluoroprolines: the prospect of making fluorine a bioelement	19

Recent advances in the asymmetric phosphoric acid-catalyzed synthesis of axially chiral compounds	19
On the application of 3d metals for C–H activation toward bioactive compounds: The key step for the synthesis of silver bullets	19
Photoredox catalysis harvesting multiple photon or electrochemical energies	18
Halides as versatile anions in asymmetric anion-binding organocatalysis	17
Incorporation of a metal-mediated base pair into an ATP aptamer – using silver(I) ions to modulate aptamer function	17
Molecular basis for protein–protein interactions	16
Towards new NIR dyes for free radical photopolymerization processes	16
Earth-abundant 3d transition metals on the rise in catalysis	16
Antiviral therapy in shrimp through plant virus VLP containing VP28 dsRNA against WSSV	16
CF3-substituted carbocations: underexploited intermediates with great potential in modern synthetic chemistry	15
BINOL as a chiral element in mechanically interlocked molecules	15
All-carbon [3 + 2] cycloaddition in natural product synthesis	15
Synthetic accesses to biguanide compounds	15
Synthesis and investigation of quadruplex-DNA-binding, 9-O-substituted berberine derivatives	14
Constrained thermoresponsive polymers – new insights into fundamentals and applications	14
Regioselective N-alkylation of the 1H-indazole scaffold; ring substituent and N-alkylating reagent effects on regioisomeric distribution	14
Synthesis of trifluoromethyl ketones by nucleophilic trifluoromethylation of esters under a fluoroform/KHMDS/triglyme system	14
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition	14
Sustainable manganese catalysis for late-stage C–H functionalization of bioactive structural motifs	14
Palladium-catalyzed solid-state borylation of aryl halides using mechanochemistry	13
Heteroleptic metallosupramolecular aggregates/complexation for supramolecular catalysis	13
A new glance at the chemosphere of macroalgal–bacterial interactions: In situ profiling of metabolites in symbiosis by mass spectrometry	13
Design, synthesis and photophysical properties of novel star-shaped truxene-based heterocycles utilizing ring-closing metathesis, Clauson–Kaas, Van Leusen and Ullmann-type reactions as key tools	13
Selected peptide-based fluorescent probes for biological applications	12
One-pot multicomponent green Hantzsch synthesis of 1,2-dihydropyridine derivatives with antiproliferative activity	12
Recent advances in the syntheses of anthracene derivatives	12
Cytochrome P450 monooxygenase-mediated tailoring of triterpenoids and steroids in plants	12
Continuous flow synthesis of azobenzenes via Baeyer–Mills reaction	12
Efficient production of clerodane and ent-kaurane diterpenes through truncated artificial pathways in Escherichia coli	12
Synthetic strategies for the preparation of γ-phostams: 1,2-azaphospholidine 2-oxides and 1,2-azaphospholine 2-oxides	12
Navigating and expanding the roadmap of natural product genome mining tools	11
Deoxyfluorination of acyl fluorides to trifluoromethyl compounds by FLUOLEAD®/Olah’s reagent under solvent-free conditions	11
In-depth characterization of self-healing polymers based on π–π nteractions	11
Unsaturated fatty acids and a prenylated tryptophan derivative from a rare actinomycete of the genus Couchioplanes	11
Construction of hexabenzocoronene-based chiral nanographenes	11
Recent advances in the application of isoindigo derivatives in materials chemistry	11
Inclusion complexes of the steroid hormones 17β-estradiol and progesterone with β- and γ-cyclodextrin hosts: syntheses, X-ray structures, thermal analyses and API solubility enhancements	11
Diels–Alder reaction of β-fluoro-β-nitrostyrenes with cyclic dienes	11
Nomimicins B–D, new tetronate-class polyketides from a marine-derived actinomycete of the genus Actinomadura	11
A sustainable strategy for the straightforward preparation of 2H-azirines and highly functionalized NH-aziridines from vinyl azides using a single solvent flow-batch approach	11
Germacrene B – a central intermediate in sesquiterpene biosynthesis	11
Metal-free nucleophilic trifluoromethylselenolation via an iodide-mediated umpolung reactivity of trifluoromethylselenotoluenesulfonate	11
Synthesis of (Z)-3-[amino(phenyl)methylidene]-1,3-dihydro-2H-indol-2-ones using an Eschenmoser coupling reaction	10
Structural basis for endoperoxide-forming oxygenases	10
Substituted nitrogen-bridged diazocines	10
Synthesis of functionalized imidazo[4,5-e]thiazolo[3,2-b]triazines by condensation of imidazo[4,5-e]triazinethiones with DMAD or DEAD and rearrangement to imidazo[4,5-e]thi	10
Menadione: a platform and a target to valuable compounds synthesis	10
Nocarimidazoles C and D, antimicrobial alkanoylimidazoles from a coral-derived actinomycete Kocuria sp.: application of 1JC,H coupling constants for the unequivocal	10
Transition-metal-catalyzed domino reactions of strained bicyclic alkenes	10
Inductive heating and flow chemistry – a perfect synergy of emerging enabling technologies	10

Tetraphenylethylene-embedded pillar[5]arene-based orthogonal self-assembly for efficient photocatalysis in water	10
Deoxygenative C2-heteroarylation of quinoline N-oxides: facile access to α-triazolylquinolines	10
DNA with zwitterionic and negatively charged phosphate modifications: Formation of DNA triplexes, duplexes and cell uptake studies	10
Natural products in the predatory defence of the filamentous fungal pathogen Aspergillus fumigatus	10
Synthesis and antimicrobial activity of 1H-1,2,3-triazole and carboxylate analogues of metronidazole	10
Controlled decomposition of SF6 by electrochemical reduction	10
Inline purification in continuous flow synthesis – opportunities and challenges	10
Chemical syntheses and salient features of azulene-containing homo- and copolymers	10
B–N/B–H Transborylation: borane-catalysed nitrile hydroboration	9
[2 + 1] Cycloaddition reactions of fullerene C60 based on diazo compounds	9
Synthesis, crystal structures and properties of carbazole-based [6]helicenes fused with an azine ring	9
Transition-metal-catalyzed C–H bond activation as a sustainable strategy for the synthesis of fluorinated molecules: an overview	9
Asymmetric organocatalyzed synthesis of coumarin derivatives	9
Targeting active site residues and structural anchoring positions in terpene synthases	9
Recent developments and trends in the iron- and cobalt-catalyzed Sonogashira reactions	9
Ionic multiresonant thermally activated delayed fluorescence emitters for light emitting electrochemical cells	9
Iron-catalyzed domino coupling reactions of π-systems	9
Cerium-photocatalyzed aerobic oxidation of benzylic alcohols to aldehydes and ketones	9
The PIFA-initiated oxidative cyclization of 2-(3-butenyl)quinazolin-4(3H)-ones – an efficient approach to 1-(hydroxymethyl)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-ones	9
The enzyme mechanism of patchoulol synthase	9
Radical cation Diels–Alder reactions of arylidene cycloalkanes	9
New efficient synthesis of polysubstituted 3,4-dihydroquinazolines and 4H-3,1-benzothiazines through a Passerini/Staudinger/aza-Wittig/addition/nucleophilic substitution sequence	9
A study of the photochemical behavior of terarylenes containing allomaltol and pyrazole fragments	9
Cholyl 1,3,4-oxadiazole hybrid compounds: design, synthesis and antimicrobial assessment	8
Annulation of a 1,3-dithiole ring to a sterically hindered o-quinone core. Novel ditopic redox-active ligands	8
Heterogeneous photocatalytic cyanomethylarylation of alkenes with acetonitrile: synthesis of diverse nitrogenous heterocyclic compounds	8
Recent advances in palladium-catalysed asymmetric 1,4–additions of arylboronic acids to conjugated enones and chromones	8
Fluorine effect in nucleophilic fluorination at C4 of 1,6-anhydro-2,3-dideoxy-2,3-difluoro-β-D-hexopyranose	8
Synthesis of highly substituted fluorenones via metal-free TBHP-promoted oxidative cyclization of 2-(aminomethyl)biphenyls. Application to the total synthesis of nobilone	8
Scope of tetrazolo[1,5-a]quinoxalines in CuAAC reactions for the synthesis of triazoloquinoxalines, imidazoloquinoxalines, and rhenium complexes thereof	8
Glycosylated coumarins, flavonoids, lignans and phenylpropanoids from Wikstroemia nutans and their biological activities	8
A systems-based framework to computationally describe putative transcription factors and signaling pathways regulating glycan biosynthesis	8
The synthesis of chiral β-naphthyl-β-sulfanyl ketones via enantioselective sulfa-Michael reaction in the presence of a bifunctional cinchona/sulfonamide organocatalyst	8
A new and efficient methodology for olefin epoxidation catalyzed by supported cobalt nanoparticles	8
Efficient synthesis of polyfunctionalized carbazoles and pyrrolo[3,4-c]carbazoles via domino Diels–Alder reaction	8
Redox-active molecules as organocatalysts for selective oxidative transformations – an unperceived organocatalysis field	8
Methodologies for the synthesis of quaternary carbon centers via hydroalkylation of unactivated olefins: twenty years of advances	8
Radical ligand transfer: a general strategy for radical functionalization	8
A Se···O bonding catalysis approach to the synthesis of calix[4]pyrroles	8
Synthesis of dibenzosuberenone-based novel polycyclic π-conjugated dihydropyridazines, pyridazines and pyrroles	8
Electron-rich triarylphosphines as nucleophilic catalysts for oxa-Michael reactions	8
Group 13 exchange and transborylation in catalysis	8
Co-crystallization of an organic solid and a tetraaryladamantane at room temperature	8
Semiautomated glycoproteomics data analysis workflow for maximized glycopeptide identification and reliable quantification	8
β-Lactamase inhibition profile of new amidine-substituted diazabicyclooctanes	8
Manganese/bipyridine-catalyzed non-directed C(sp3)–H bromination using NBS and TMSN3	8
Efficient synthesis of ethyl 2-(oxazolin-2-yl)alkanoates via ethoxycarbonylketene-induced electrophilic ring expansion of aziridines	8
3-Acetoxy-fatty acid isoprenyl esters from androconia of the ithomiine butterfly Ithomia salapia	8
Characterization of a new fusicoccane-type diterpene synthase and an associated P450 enzyme	7
Enantioenriched α-substituted glutamates/pyroglutamates via enantioselective cyclopropenimine-catalyzed Michael addition of amino ester imines	7
Benzothiazolium salts as reagents for the deoxygenative perfluoroalkylthiolation of alcohols	7
Exploring the role of halogen bonding in iodonium ylides: insights into unexpected reactivity and reaction control	7
UV resonance Raman spectroscopy of the supramolecular ligand guanidiniocarbonyl indole (GCI) with 244 nm laser excitation	7
Make or break: the thermodynamic equilibrium of polyphosphate kinase-catalysed reactions	7
Synthesis of imidazo[1,5-a]pyridines via cyclocondensation of 2-(aminomethyl)pyridines with electrophilically activated nitroalkanes	7
Cyclodextrins as building blocks for new materials	7
Synthesis and electrochemical properties of 3,4,5-tris(chlorophenyl)-1,2-diphosphaferrocenes	7
Synthesis of O6-alkylated preQ1 derivatives	7
Polymer and small molecule mechanochemistry: closer than ever	7
Regioselective synthesis of heterocyclic N-sulfonyl amidines from heteroaromatic thioamides and sulfonyl azides	7
Naphthalonitriles featuring efficient emission in solution and in the solid state	7
Combining the best of both worlds: radical-based divergent total synthesis	7
Rapid gas–liquid reaction in flow. Continuous synthesis and production of cyclohexene oxide	7
Metal-free glycosylation with glycosyl fluorides in liquid SO2	7
An efficient metal-free and catalyst-free C–S/C–O bond-formation strategy: synthesis of pyrazole-conjugated thioamides and amides	7
DABCO-promoted photocatalytic C–H functionalization of aldehydes	7
Quinoxaline derivatives as attractive electron-transporting materials	7
A straightforward conversion of 1,4-quinones into polycyclic pyrazoles via [3 + 2]-cycloaddition with fluorinated nitrile imines	7
Post-functionalization of drug-loaded nanoparticles prepared by polymerization-induced self-assembly (PISA) with mitochondria targeting ligands	7
A novel and robust heterogeneous Cu catalyst using modified lignosulfonate as support for the synthesis of nitrogen-containing heterocycles	7
DDQ in mechanochemical C–N coupling reactions	7
The effect of dark states on the intersystem crossing and thermally activated delayed fluorescence of naphthalimide-phenothiazine dyads	6
Cationic oligonucleotide derivatives and conjugates: A favorable approach for enhanced DNA and RNA targeting oligonucleotides	6
Correction: Amine–borane complex-initiated SF5Cl radical addition on alkenes and alkynes	6
Selective construction of dispiro[indoline-3,2'-quinoline-3',3''-indoline] and dispiro[indoline-3,2'-pyrrole-3',3''-indoline] via three-component reaction	6
Synthesis of new bile acid-fused tetrazoles using the Schmidt reaction	6
Electrocatalytic C(sp3)–H/C(sp)–H cross-coupling in continuous flow through TEMPO/copper relay catalysis	6
Metal-free visible-light-enabled vicinal trifluoromethyl dithiolation of unactivated alkenes	6
Regioselective synthesis of methyl 5-(N-Boc-cycloaminyl)-1,2-oxazole-4-carboxylates as new amino acid-like building blocks	6
Double-headed nucleosides: Synthesis and applications	6

A novel methodology for the efficient synthesis of 3-monohalooxindoles by acidolysis of 3-phosphate-substituted oxindoles with haloid acids	6
Synthesis of odorants in flow and their applications in perfumery	6
Chemical and chemoenzymatic routes to bridged homoarabinofuranosylpyrimidines: Bicyclic AZT analogues	6
Thermally activated delayed fluorescence (TADF) emitters: sensing and boosting spin-flipping by aggregation	6
Multi-faceted reactivity of N-fluorobenzenesulfonimide (NFSI) under mechanochemical conditions: fluorination, fluorodemethylation, sulfonylation, and amidation reactions	6
Simulating the enzymes of ganglioside biosynthesis with Glycologue	6
Chemoselective N-acylation of indoles using thioesters as acyl source	6
Designed whole-cell-catalysis-assisted synthesis of 9,11-secosterols	6
1,2,3-Triazoles as leaving groups in SNAr–Arbuzov reactions: synthesis of C6-phosphonated purine derivatives	6
Mechanochemical halogenation of unsymmetrically substituted azobenzenes	6
α,γ-Dioxygenated amides via tandem Brook rearrangement/radical oxygenation reactions and their application to syntheses of γ-lactams	6
Access to cyclopropanes with geminal trifluoromethyl and difluoromethylphosphonate groups	6
Electrochemical hydrogenation of enones using a proton-exchange membrane reactor: selectivity and utility	6
Recent progress in the synthesis of homotropane alkaloids adaline, euphococcinine and N-methyleuphococcinine	6
Synthesis of multiply fluorinated N-acetyl-D-glucosamine and D-galactosamine analogs via the corresponding deoxyfluorinated glucosazide and galactosazide phenyl thioglycosides	6
Synthesis of phenanthridines via a novel photochemically-mediated cyclization and application to the synthesis of triphaeridine	6
Synthesis of legonmycins A and B, C(7a)-hydroxylated bacterial pyrrolizidines	6
Tenacibactins K–M, cytotoxic siderophores from a coral-associated gliding bacterium of the genus Tenacibaculum	6
Unexpected rearrangements and a novel synthesis of 1,1-dichloro-1-alkenones from 1,1,1-trifluoroalkanones with aluminium trichloride	6
Insight into oral amphiphilic cyclodextrin nanoparticles for colorectal cancer: comprehensive mathematical model of drug release kinetic studies and antitumoral efficacy in 3D spheroid colon tumors	5
Facile preparation and conversion of 4,4,4-trifluorobut-2-yn-1-ones to aromatic and heteroaromatic compounds	5
Aromatic C–H bond functionalization through organocatalyzed asymmetric intermolecular aza-Friedel–Crafts reaction: a recent update	5
Anti-inflammatory aromadendrane- and cadinane-type sesquiterpenoids from the South China Sea sponge Acanthella cavernosa	5
Solvent-free synthesis of enantioenriched β-silyl nitroalkanes under organocatalytic conditions	5
Tri(n-butyl)phosphine-promoted domino reaction for the efficient construction of spiro[cyclohexane-1,3'-indolines] and spiro[indoline-3,2'-furan-3',3''-indolines]	5
Modern flow chemistry – prospect and advantage	5
On the mass spectrometric fragmentations of the bacterial sesterterpenes sestermobaraenes A–C	5
Functionalization of imidazole N-oxide: a recent discovery in organic transformations	5
Synthesis of C6-modified mannose 1-phosphates and evaluation of derived sugar nucleotides against GDP-mannose dehydrogenase	5
α-Ketol and α-iminol rearrangements in synthetic organic and biosynthetic reactions	5
Amino- and polyaminophthalazin-1(2H)-ones: synthesis, coordination properties, and biological activity	5
Helicene synthesis by Brønsted acid-catalyzed cycloaromatization in HFIP [(CF3)2CHOH]	5
Pyridine C(sp2)–H bond functionalization under transition-metal and rare earth metal catalysis	5
Cascade intramolecular Prins/Friedel–Crafts cyclization for the synthesis of 4-aryltetralin-2-ols and 5-aryltetrahydro-5H-benzo[7]annulen-7-ols	5
2,4-Bis(arylethynyl)-9-chloro-5,6,7,8-tetrahydroacridines: synthesis and photophysical properties	5
Multiswitchable photoacid–hydroxyflavylium–polyelectrolyte nano-assemblies	5
Organocatalytic asymmetric Michael/acyl transfer reaction between α-nitroketones and 4-arylidenepyrrolidine-2,3-diones	5
Hydrazides in the reaction with hydroxypyrrolines: less nucleophilicity – more diversity	5
Peptide stapling by late-stage Suzuki–Miyaura cross-coupling	5
Four bioactive new steroids from the soft coral Lobophytum pauciflorum collected in South China Sea	5
Transition-metal-free intramolecular Friedel–Crafts reaction by alkene activation: A method for the synthesis of some novel xanthene derivatives	5
Copper-catalyzed multicomponent reactions for the efficient synthesis of diverse spirotetrahydrocarbazoles	5
1,2-Naphthoquinone-4-sulfonic acid salts in organic synthesis	5
An isoxazole strategy for the synthesis of 4-oxo-1,4-dihydropyridine-3-carboxylates	5
Terpenoids from Glechoma hederacea var. longituba and their biological activities	5
Automated grindstone chemistry: a simple and facile way for PEG-assisted stoichiometry-controlled halogenation of phenols and anilines using N-halosuccinimides	5
Synthesis of bis-spirocyclic derivatives of 3-azabicyclo[3.1.0]hexane via cyclopropene cycloadditions to the stable azomethine ylide derived from Ruhemann's purple	5
Chemical constituents of Chaenomeles sinensis twigs and their biological activity	5
Site-selective reactions mediated by molecular containers	5
Base-free enantioselective SN2 alkylation of 2-oxindoles via bifunctional phase-transfer catalysis	5
Synthetic strategies toward 1,3-oxathiolane nucleoside analogues	5
Iodine-catalyzed electrophilic substitution of indoles: Synthesis of (un)symmetrical diindolylmethanes with a quaternary carbon center	5
N-Sulfinylpyrrolidine-containing ureas and thioureas as bifunctional organocatalysts	5
Chemistry of polyhalogenated nitrobutadienes, 17: Efficient synthesis of persubstituted chloroquinolinyl-1H-pyrazoles and evaluation of their antimalarial, anti-SARS-CoV-2, antibacterial, and c	5
Clauson–Kaas pyrrole synthesis using diverse catalysts: a transition from conventional to greener approach	5
A resorcin[4]arene hexameric capsule as a supramolecular catalyst in elimination and isomerization reactions	5
Synthesis of α-(perfluoroalkylsulfonyl)propiophenones: a new set of reagents for the light-mediated perfluoroalkylation of aromatics	5
Selective sulfonylation and isonitrilation of para-quinone methides employing TosMIC as a source of sulfonyl group or isonitrile group	5
Highly regio- and stereoselective phosphinylphosphination of terminal alkynes with tetraphenyldiphosphine monoxide under radical conditions	5
Application of the Meerwein reaction of 1,4-benzoquinone to a metal-free synthesis of benzofuropyridine analogues	5
A trustworthy mechanochemical route to isocyanides	5