Beilstein Journal of Organic Chemistry

Papers
(The TQCC of Beilstein Journal of Organic Chemistry is 6. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2022-08-01 to 2026-08-01.)
ArticleCitations
Photoredox-catalyzed arylation of isonitriles by diaryliodonium salts towards benzamides54
Recent advances in electrochemical copper catalysis for modern organic synthesis52
Redox-active molecules as organocatalysts for selective oxidative transformations – an unperceived organocatalysis field43
Biobased carbon dots as photoreductants – an investigation by using triarylsulfonium salts40
Chiral phosphoric acid-catalyzed asymmetric synthesis of helically chiral, planarly chiral and inherently chiral molecules36
Anion-dependent ion-pairing assemblies of triazatriangulenium cation that interferes with stacking structures35
Asymmetric synthesis of a stereopentade fragment toward latrunculins34
Cyclization of 1-aryl-4,4,4-trichlorobut-2-en-1-ones into 3-trichloromethylindan-1-ones in triflic acid32
Facile approach to N,O,S-heteropentacycles via condensation of sterically crowded 3 H -phenoxazin-3-one with ortho- 32
Entry to 2-aminoprolines via electrochemical decarboxylative amidation of N ‑acetylamino malonic acid monoesters28
Chemoenzymatic synthesis of the cardenolide rhodexin A and its aglycone sarmentogenin27
Improved synthesis and physicochemical characterization of the selective serotonin 2A receptor agonist 25CN-NBOH25
Synthesis of diaryl phosphates using phytic acid as a phosphorus source23
Bioinspired total syntheses of natural products: a personal adventure23
Efficacy of radical reactions of isocyanides with heteroatom radicals in organic synthesis23
A new analog of dihydroxybenzoic acid from Saccharopolyspora sp. KR21-000122
Computational model predicts protein binding sites of a luminescent ligand equipped with guanidiniocarbonyl-pyrrole groups22
Finding the most potent compounds using active learning on molecular pairs22
Modular synthesis of 2-furyl carbinols from 3-benzyldimethylsilylfurfural platforms relying on oxygen-assisted C–Si bond functionalization22
A novel recyclable organocatalyst for the gram-scale enantioselective synthesis of ( S )-baclofen21
Enzymes in biosynthesis21
Synthesis of novel 1,2,4-oxadiazole-isoxazoline hybrids and their in silico potential with adenosine receptors20
Two-fold addition reaction of silylene to C 60 : structural and electronic properties of a bis-adduct20
Deciphering the mechanism of γ-cyclodextrin’s hydrophobic cavity hydration: an integrated experimental and theoretical study20
Efficient synthesis of fluorinated triphenylenes with enhanced arene–perfluoroarene interactions in columnar mesophases19
Hydrogen-bond activation enables aziridination of unactivated olefins with simple iminoiodinanes19
Rhodium-catalysed connective synthesis of diverse reactive probes bearing S(VI) electrophilic warheads19
Synthesis of N -acetyl diazocine derivatives via cross-coupling reaction19
Solar thermal fuels: azobenzene as a cyclic photon–heat transduction platform19
One-pot four-component sequential synthesis of S -alkyl dithiocarbamates using lipase as a biocatalyst19
Synthesis of tricyclic fused pyrrolidine nitroxides from 2-alkynylpyrrolidine-1-oxyls19
Synthesis of extended fluorinated tripeptides based on the tetrahydropyridazine scaffold18
Preparation of an advanced intermediate for the synthesis of leustroducsins and phoslactomycins by heterocycloaddition18
Domino reactions of chromones with activated carbonyl compounds18
Synthesis, α-mannosidase inhibition studies and molecular modeling of 1,4-imino-ᴅ-lyxitols and their C-5-altered N -arylalkyl derivatives18
Electrochemical and spectroscopic properties of twisted dibenzo[ g , p ]chrysene derivatives17
Sustainable tandem acylation/Diels–Alder reaction toward versatile tricyclic epoxyisoindole-7-carboxylic acids in renewable green solvents17
Green and sustainable approaches for the Friedel–Crafts reaction between aldehydes and indoles17
Rongalite addition to dienones: diastereoselectivity in cyclic sulfone synthesis; stereochemical rationalization and prospects as a general conjugate nucleophile17
Tandem hydrothiocyanation/cyclization of CF 3 -iminopropargyl alcohols with NaSCN in the presence of AcOH16
Gold extraction at the molecular level using α- and β-cyclodextrins16
Synthesis of protected precursors of chitin oligosaccharides by electrochemical polyglycosylation of thioglycosides16
N -Boc-α-diazo glutarimide as efficient reagent for assembling N-heterocycle-glutarimide diads via Rh(II)-catalyzed N–H insertion reaction16
Ambident reactivity of enolizable 5-mercapto-1 H -tetrazoles in trapping reactions with in situ-generated thiocarbonyl S 16
A study of the DIBAL-promoted selective debenzylation of α-cyclodextrin protected with two different benzyl groups15
Site-specific labelling of native peptides and proteins: chemical and enzymatic strategies15
Bromination of endo- 7-norbornene derivatives revisited: failure of a computational NMR method in elucidating the configuration of an organic structure15
Multi-redox indenofluorene chromophores incorporating dithiafulvene donor and ene/enediyne acceptor units15
Catalytic aza-Nazarov cyclization reactions to access α-methylene-γ-lactam heterocycles15
Design, synthesis, and evaluation of chiral thiophosphorus acids as organocatalysts15
Novel truxene-based dipyrromethanes (DPMs): synthesis, spectroscopic characterization and photophysical properties15
Streptoquinolines A and B, new antibacterial meroterpenoids produced by Streptomyces sp. TMPU-A067914
Ring opening of photogenerated azetidinols as a strategy for the synthesis of aminodioxolanes14
Inclusion complexes of the steroid hormones 17β-estradiol and progesterone with β- and γ-cyclodextrin hosts: syntheses, X-ray structures, thermal analyses and API solubility enhancements14
Palladium-catalyzed three-component radical-polar crossover carboamination of 1,3-dienes or allenes with diazo esters and amines14
Synthesis of disulfides and 3-sulfenylchromones from sodium sulfinates catalyzed by TBAI14
Photoluminescence color-tuning with polymer-dispersed fluorescent films containing two fluorinated diphenylacetylene-type fluorophores14
1-Butyl-3-methylimidazolium tetrafluoroborate as suitable solvent for BF 3 : the case of alkyne hydration. Chemistry vs electrochemistry14
Synthesis and anti-cancer activity of naphthalimide–organylselanyl conjugates13
Copper-catalyzed N -arylation of amines with aryliodonium ylides in water13
Photocatalytic sequential C–H functionalization expediting acetoxymalonylation of imidazo heterocycles13
Formal synthesis of a selective estrogen receptor modulator with tetrahydrofluorenone structure using [3 + 2 + 1] cycloaddition of yne-vinylcyclopropanes and CO13
Reactivity of hypervalent iodine(III) reagents bearing a benzylamine with sulfenate salts13
Mild and efficient synthesis and base-promoted rearrangement of novel isoxazolo[4,5- b ]pyridines13
Synthesis of π-conjugated polycyclic compounds by late-stage extrusion of chalcogen fragments12
Copper-promoted C5-selective bromination of 8-aminoquinoline amides with alkyl bromides12
HFIP as a versatile solvent in resorcin[ n ]arene synthesis12
Total syntheses of highly oxidative Ryania diterpenoids facilitated by innovations in synthetic strategies12
Electrophotochemical metal-catalyzed synthesis of alkylnitriles from simple aliphatic carboxylic acids12
Methodology for awakening the potential secondary metabolic capacity in actinomycetes12
Harnessing tethered nitreniums for diastereoselective amino-sulfonoxylation of alkenes12
Unsymmetrical sulfoxides with sterically hindered catechol fragment: synthesis, structure, electrochemical properties, and antiradical activity12
Palladium-catalyzed enantioselective three-component synthesis of α-arylglycine derivatives from glyoxylic acid, sulfonamides and aryltrifluoroborates12
Ugi bisamides based on pyrrolyl-β-chlorovinylaldehyde and their unusual transformations12
Development and mechanistic studies of calcium–BINOL phosphate-catalyzed hydrocyanation of hydrazones12
Photochemically assisted synthesis of phenacenes fluorinated at the terminal benzene rings and their electronic spectra12
Synthesis of 1,4-azaphosphinine nucleosides and evaluation as inhibitors of human cytidine deaminase and APOBEC3A11
Aryl iodane-induced cascade arylation–1,2-silyl shift–heterocyclization of propargylsilanes under copper catalysis11
Characterization of a new fusicoccane-type diterpene synthase and an associated P450 enzyme11
Copper catalysis: a constantly evolving field11
Enantioselective radical chemistry: a bright future ahead11
Correction: Diastereoselective synthesis of highly substituted cyclohexanones and tetrahydrochromene-4-ones via conjugate addition of curcumins to arylidenemalonates11
Knoevenagel condensation of 4,5- and 1,8-diazafluorenes11
Synthesis and biological profile of 2,3-dihydro[1,3]thiazolo[4,5-b]pyridines, a novel class of acyl-ACP thioesterase inhibitors11
A m -quaterphenyl probe for absolute configurational assignments of primary and secondary amines11
The application of desymmetric enantioselective reduction of cyclic 1,3-dicarbonyl compounds in the total synthesis of terpenoid and alkaloid natural products11
Arene activation via π-bond localization: concepts and opportunities10
Dissecting Mechanochemistry III10
An efficient metal-free and catalyst-free C–S/C–O bond-formation strategy: synthesis of pyrazole-conjugated thioamides and amides10
Rhodium-catalyzed homo-coupling reaction of aryl Grignard reagents and its application for the synthesis of an integrin inhibitor10
Facile synthesis of hydantoin/1,2,4-oxadiazoline spiro-compounds via 1,3-dipolar cycloaddition of nitrile oxides to 5-iminohydantoins10
Three-component N -alkenylation of azoles with alkynes and iodine(III) electrophile: synthesis of multisubstituted N 10
Kinetically stabilized 1,3-diarylisobenzofurans and the possibility of preparing large, persistent isoacenofurans with unusually small HOMO–LUMO gaps10
(Bio)isosteres of ortho - and meta -substituted benzenes10
Synthesis of the aggregation pheromone of Tribolium castaneum10
N -Salicyl-amino acid derivatives with antiparasitic activity from Pseudomonas sp. UIAU-6B10
Synthesis of cyclic β-1,6-oligosaccharides from glucosamine monomers by electrochemical polyglycosylation10
Access to cyclopropanes with geminal trifluoromethyl and difluoromethylphosphonate groups10
Advancements in hydrochlorination of alkenes10
Orthogonal photoswitching of heterobivalent azobenzene glycoclusters: the effect of glycoligand orientation in bacterial adhesion10
Applications of microscopy and small angle scattering techniques for the characterisation of supramolecular gels10
C3-Alkylation of furfural derivatives by continuous flow homogeneous catalysis10
Recent advances in the stereoselective synthesis of distal biaxially chiral molecules10
Electrogenerated base-promoted cyclopropanation using alkyl 2-chloroacetates10
Chitosan-supported CuI-catalyzed cascade reaction of 2-halobenzoic acids and amidines for the synthesis of quinazolinones10
Get a better glimpse on sequential photoreactions of trisnorbornadienes with 19 F NMR spectroscopy10
Total synthesis: an enabling science10
Computational studies of Brønsted acid-catalyzed transannular cycloadditions of cycloalkenone hydrazones10
Kinetic resolution of racemic planar-chiral vinylcymantrenes by molybdenum-catalyzed asymmetric metathesis dimerization10
New azodyrecins identified by a genome mining-directed reactivity-based screening10
Reactions of acryl thioamides with iminoiodinanes as a one-step synthesis of N -sulfonyl-2,3-dihydro-1,2-thiazoles10
Recent advances in amidyl radical-mediated photocatalytic direct intermolecular hydrogen atom transfer9
Metal catalyst-free N-allylation/alkylation of imidazole and benzimidazole with Morita–Baylis–Hillman (MBH) alcohols and acetates9
One-pot nucleophilic substitution–double click reactions of biazides leading to functionalized bis(1,2,3-triazole) derivatives9
Quantifying the ability of the CF 2 H group as a hydrogen bond donor9
Synthesis and structural elucidation of a novel bis-spirooxindole from isatin and ethylenediamine9
Total synthesis of asperdinones B, C, D, E and terezine D9
Chemical structure metagenomics of microbial natural products: surveying nonribosomal peptides and beyond9
Studies on the syntheses of β-carboline alkaloids brevicarine and brevicolline9
Stereoselective mechanochemical synthesis of thiomalonate Michael adducts via iminium catalysis by chiral primary amines9
N -Glycosides of indigo, indirubin, and isoindigo: blue, red, and yellow sugars and their cancerostatic activity9
Conformational analysis of difluoromethylornithine: factors influencing its gas-phase and bioactive conformations9
Oxidative hydrolysis of aliphatic bromoalkenes: scope study and reactivity insights9
Total synthesis of the capsular polysaccharide repeating unit towards the development of a glycoconjugate vaccine against Klebsiella pneumoniae ST5129
Navigating and expanding the roadmap of natural product genome mining tools9
Enhanced reactivity of Li + @C 60 toward thermal [2 + 2] cycloaddition by encapsulated Li 9
Effect of substitution position of aryl groups on the thermal back reactivity of aza-diarylethene photoswitches and prediction by density functional theory8
Acetaldehyde in the Enders triple cascade reaction via acetaldehyde dimethyl acetal8
Chiral phosphoric acid-catalyzed transfer hydrogenation of 3,3-difluoro-3 H -indoles8
Intramolecular C–H arylation of pyridine derivatives with a palladium catalyst for the synthesis of multiply fused heteroaromatic compounds8
Biphenylene-containing polycyclic conjugated compounds8
Mechanochemical difluoromethylations of ketones8
A novel bis-triazole scaffold accessed via two tandem [3 + 2] cycloaddition events including an uncatalyzed, room temperature azide–alkyne click reaction8
Ligand effects, solvent cooperation, and large kinetic solvent deuterium isotope effects in gold(I)-catalyzed intramolecular alkene hydroamination8
Solid-phase total synthesis and structural confirmation of antimicrobial longicatenamide A8
Regioselective quinazoline C2 modifications through the azide–tetrazole tautomeric equilibrium8
Manganese-catalyzed C–C and C–N bond formation with alcohols via borrowing hydrogen or hydrogen auto-transfer8
Selective and scalable oxygenation of heteroatoms using the elements of nature: air, water, and light8
Three-component reactions of conjugated dienes, CH acids and formaldehyde under diffusion mixing conditions8
Recent advances in controllable/divergent synthesis8
Unique halogen–π association detected in single crystals of C–N atropisomeric N -(2-halophenyl)quinolin-2-one derivatives and the thione analogue8
Advances in nitrogen-containing helicenes: synthesis, chiroptical properties, and optoelectronic applications8
Cycloaddition reactions of heterocyclic azides with 2-cyanoacetamidines as a new route to C , N -diheteroa8
An Fe(II)-catalyzed synthesis of spiro[indoline-3,2'-pyrrolidine] derivatives8
A novel spirocyclic scaffold accessed via tandem Claisen rearrangement/intramolecular oxa-Michael addition8
The unique reactivity of 5,6-unsubstituted 1,4-dihydropyridine in the Huisgen 1,4-diploar cycloaddition and formal [2 + 2] cycloaddition8
Mechanistic investigations of polyaza[7]helicene in photoredox and energy transfer catalysis8
4,6-Diaryl-5,5-difluoro-1,3-dioxanes as chiral dopants for liquid crystal compositions8
Z -Selective semihydrogenation of alkynes via Ni/Lewis acid synergistic catalyzed system using DMF as hydrogen source and solvent8
Continuous-flow-enabled intensification in nitration processes: a review of technological developments and practical applications over the past decade8
Facile access to 3-sulfonylquinolines via Knoevenagel condensation/aza-Wittig reaction cascade involving ortho -azidobenzaldehydes and β-ketosulfonamides8
Mechanistic insights into hydroxy(tosyloxy)iodobenzene-mediated ditosyloxylation of chalcones: a DFT study8
Retraction: α,ß-Didehydrosuberoylanilide hydroxamic acid (DDSAHA) as precursor and possible analogue of the anticancer drug SAHA8
Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine8
Ortho -ester-substituted diaryliodonium salts enabled regioselective arylocyclization of naphthols toward 3,4-benzocoumarins7
Advances in the use of metal-free tetrapyrrolic macrocycles as catalysts7
Transition-metal-catalyzed C–H bond activation as a sustainable strategy for the synthesis of fluorinated molecules: an overview7
Digyalipopeptide A, an antiparasitic cyclic peptide from the Ghanaian Bacillus sp. strain DE2B7
4-(1-Methylamino)ethylidene-1,5-disubstituted pyrrolidine-2,3-diones: synthesis, anti-inflammatory effect and in silico approaches7
Electroreductive coupling of 2-acylbenzoates with α,β-unsaturated carbonyl compounds: density functional theory study on product selectivity7
Synthesis of benzo[ f ]quinazoline-1,3(2 H ,4 H )-diones7
Divergent role of PIDA and PIFA in the AlX 3 (X = Cl, Br) halogenation of 2-naphthol: a mechanistic study7
Tandem diazotization/cyclization approach for the synthesis of a fused 1,2,3-triazinone-furazan/furoxan heterocyclic system7
On drug discovery against infectious diseases and academic medicinal chemistry contributions7
Synthesis of substituted 8 H -benzo[ h ]pyrano[2,3- f ]quin7
Discovery and biosynthesis of bacterial drimane-type sesquiterpenoids from Streptomyces clavuligerus7
High-pressure activation for the solvent- and catalyst-free syntheses of heterocycles, pharmaceuticals and esters7
Beyond symmetric self-assembly and effective molarity: unlocking functional enzyme mimics with robust organic cages7
New cembrane-type diterpenoids with anti-inflammatory activity from the South China Sea soft coral Sinularia sp.7
Discrimination of β-cyclodextrin/hazelnut ( Corylus avellana L.) oil/flavonoid glycoside and flavonolignan ternary complexes by Fourier-transform infrare7
Synthesis of β-ketophosphonates through aerobic copper(II)-mediated phosphorylation of enol acetates7
Pentacyclic aromatic heterocycles from Pd-catalyzed annulation of 1,5-diaryl-1,2,3-triazoles7
Rapid construction of tricyclic tetrahydrocyclopenta[4,5]pyrrolo[2,3- b ]pyridine via isocyanide-based multicomponent reaction7
Discovery of sugarnitriles A and B, and structural reassignment of SF-2140, from a sugarcane endophytic actinomycete Amycolatopsis sp. JS-O277
Advances in Zr-mediated radical transformations and applications to total synthesis7
Synthesis and applications of alkenyl chlorides (vinyl chlorides): a review7
Synthesis of the tetracyclic skeleton of Aspidosperma alkaloids via PET-initiated cationic radical-derived interrupted [2 + 2]/ re7
Mechanochemical bottom-up synthesis of phosphorus-linked, heptazine-based carbon nitrides using sodium phosphide7
Synthesis and antimycotic activity of new derivatives of imidazo[1,2- a ]pyrimidines7
Sustainable electrochemical synthesis of aliphatic nitro- NNO -azoxy compounds employing ammonium dinitramide and their in vitro evaluation as potential 7
Long oligodeoxynucleotides: chemical synthesis, isolation via catching-by-polymerization, verification via sequencing, and gene expression demonstration7
Enantioselective desymmetrization strategy of prochiral 1,3-diols in natural product synthesis7
Synthesis of polycyclic aromatic quinones by continuous flow electrochemical oxidation: anodic methoxylation of polycyclic aromatic phenols (PAPs)7
Rotaxanes with integrated photoswitches: design principles, functional behavior, and emerging applications7
Harnessing unprotected deactivated amines and arylglyoxals in the Ugi reaction for the synthesis of fused complex nitrogen heterocycles7
Functions of enzyme domains in 2-methylisoborneol biosynthesis and enzymatic synthesis of non-natural analogs7
Cage-like microstructures via sequential Ugi reactions in aqueous emulsions7
Synthesis and reactivity of the di(9-anthryl)methyl radical7
Practical synthesis of isocoumarins via Rh(III)-catalyzed C–H activation/annulation cascade7
Asymmetric tandem conjugate addition and reaction with carbocations on acylimidazole Michael acceptors7
Azide–alkyne cycloaddition (click) reaction in biomass-derived solvent Cyrene TM under one-pot conditions6
Mining raw plant transcriptomic data for new cyclopeptide alkaloids6
Mechanisms for radical reactions initiating from N -hydroxyphthalimide esters6
Heteroannulations of cyanoacetamide-based MCR scaffolds utilizing formamide6
Halogenated azobenzene acrylates: from efficient solution photoswitching to stable solid-state photochromic materials6
Phenanthridine–pyrene conjugates as fluorescent probes for DNA/RNA and an inactive mutant of dipeptidyl peptidase enzyme6
Synthesis of new tetra- and pentacyclic, methylenedioxy- and ethylenedioxy-substituted derivatives of the dibenzo[ c , f 6
Design, synthesis, and biological evaluation of FXR/ASK1 dual-target modulators6
Identification and determination of the absolute configuration of amorph-4-en-10β-ol, a cadinol-type sesquiterpene from the scent glands of the African reed frog Hyperolius cinn6
GlAIcomics: a deep neural network classifier for spectroscopy-augmented mass spectrometric glycans data6
One-pot synthesis of 2-arylated and 2-alkylated benzoxazoles and benzimidazoles based on triphenylbismuth dichloride-promoted desulfurization of thioamides6
Semisynthetic derivatives of massarilactone D with cytotoxic and nematicidal activities6
Novel macrocycles: from synthesis to supramolecular function6
Cell-free protein synthesis with technical additives – expanding the parameter space of in vitro gene expression6
Molecular diversity of the reactions of MBH carbonates of isatins and various nucleophiles6
Thermodynamics and polarity-driven properties of fluorinated cyclopropanes6
Cascade transformation of 2-(diazoacetyl)-2 H -azirines to 2-aroyl-3-hydroxy-1 H -pyrroles via condensatio6
1,2-Difluoroethylene (HFO-1132): synthesis and chemistry6
Insight into oral amphiphilic cyclodextrin nanoparticles for colorectal cancer: comprehensive mathematical model of drug release kinetic studies and antitumoral efficacy in 3D spheroid colon tumors6
Synthesis of tetrahydrofuro[3,2- c ]pyridines via Pictet–Spengler reaction6
Configuration–packing synergy enabling integrated crystalline-state RTP and amorphous-state TADF6
Modern flow chemistry – prospect and advantage6
Red light excitation: illuminating photocatalysis in a new spectrum6
Fe-catalyzed efficient synthesis of 2,4- and 4-substituted quinolines via C(sp 2 )–C(sp 2 ) bond s6
Bismuth(III) triflate: an economical and environmentally friendly catalyst for the Nazarov reaction6
Charge carrier transport in perylene-based and pyrene-based columnar liquid crystals6
Symmetrical D–π–A–π–D indanone dyes: a new design for nonlinear optics and cyanide detection6
Synthesis of spiroindolenines through a one-pot multistep process mediated by visible light6
Confirmation of the stereochemistry of spiroviolene6
Effect of a photoswitchable rotaxane on membrane permeabilization across lipid compositions6
Revisiting the bromination of 3β-hydroxycholest-5-ene with CBr 4 /PPh 3 and the subsequent azidoly6
Rhodopyran, a carboxylated hexahydrocyclopenta[ b ]pyran from Rhodococcus6
A myo -inositol dehydrogenase involved in aminocyclitol biosynthesis of hygromycin A6
Synthesis of electrophile-tethered preQ 1 analogs for covalent attachment to preQ 1 RNA6
Mechanochemical solid state synthesis of copper(I)/NHC complexes with K 3 PO 46
Thermodynamic equilibrium between locally excited and charge transfer states in perylene–phenothiazine dyads6
Optimizing reaction conditions for the light-driven hydrogen evolution in a loop photoreactor6
Ex-situ generation of gaseous nitriles in two-chamber glassware for facile haloacetimidate synthesis6
Synthesis of N-doped chiral macrocycles by regioselective palladium-catalyzed arylation6
Controlled oligomerization of [1.1.1]propellane through radical polarity matching: selective synthesis of SF 5 - and CF 36
Synthesis of new representatives of A 3 B-type carboranylporphyrins based on meso -tetra(pentafluoroph6
Synthesis and biological evaluation of new brassinosteroid analogs with C-22 benzoate function6
Organophosphorus chemistry: from model to application6
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