OOIR: Observatory of International Research

Papers

(The TQCC of Molecular Pharmaceutics is 9. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-09-01 to 2025-09-01.)

Article	Citations
High Molecular Weight Poly(glutamic acid) to Improve BMP2-Induced Osteogenic Differentiation	167
A Model Study to Assess Fibrillation and Product Stability to Support Peptide Drug Design	117
Construction and Preclinical Evaluation of a ^124/125I-Labeled Specific Antibody Targeting PD-L2 in Lung Cancer	90
Coupled Discrete Phase and Eulerian Wall Film Models for Drug Deposition Efficacy Analysis in Human Respiratory Airways	86
Fluorophore-Conjugated Anti-ICOS Antibody Enables Precise Prediction of Therapeutic Response of the STING Agonist in Colorectal Cancer via NIRF Imaging	85
Analysis of Cimetidine Crystal Polymorphs by X-ray Absorption Near-Edge Spectroscopy	80
Mechanical Extrusion of the Plasma Membrane to Generate Ectosome-Mimetic Nanovesicles for Lung Targeting	79
Exploration of Verticillins in High-Grade Serous Ovarian Cancer and Evaluation of Multiple Formulations in Preclinical In Vitro and In Vivo Models	75
Pterostilbene-Loaded Soluplus/Poloxamer 188 Mixed Micelles for Protection against Acetaminophen-Induced Acute Liver Injury	74
Enhanced Therapeutic Efficacy Against Melanoma through Exosomal Delivery of Hesperidin	72
Quantitative Characterization of Clinically Relevant Drug-Metabolizing Enzymes and Transporters in Rat Liver and Intestinal Segments for Applications in PBPK Modeling	72
Invisible Bridges: Unveiling the Role and Prospects of Tunneling Nanotubes in Cancer Therapy	70
Transition Metal (Molybdenum)-Doped Drug-like Conformational Nanoarchitectonics with Altered Valence States (Mn²⁺/Mn⁴⁺ and Mo⁵⁺/Mo⁶⁺) for Augmented Cancer T	68
Understanding the Roles of Excipients in Moisture Management in Solid Dosage Forms	63
Difference in Endocytosis Pathways Used by Differentiated Versus Nondifferentiated Epithelial Caco-2 Cells to Internalize Nanosized Particles	62
Pharmacokinetics in Penguins Compared to Other Avian Species: A Review of Enrofloxacin and Voriconazole	62
Revolutionizing Neurological Therapies: The Multifaceted Potential of Zein-Based Nanoparticles for Brain-Targeted Drug Delivery	61
Issue Editorial Masthead	59
Issue Editorial Masthead	53
Advancing Amorphous Solid Dispersions Design: Insights into Dissolution Kinetics via Thermodynamic Descriptor and Machine Learning	52
Solid-State Evaluation of a Newly Emerged Polymorph for Early-Stage Pharmaceutical Development	51
Issue Publication Information	50
Pharmacokinetic Bioequivalence between Generic and Originator Orally Inhaled Drug Products: Validity of Administration of Doses above the Approved Single Maximum Dose	49
Structured Sponsorship: An Option for Improved Workplace Inclusion in the Pharmaceutical Sciences	49
Evaluation of a Tumor-Targeting Oligosaccharide Nanosystem in BNCT on an Orthotopic Hepatocellular Carcinoma Model	48

Correction to “Effects of PEGylation on Imaging Contrast of ⁶⁸Ga-Labeled Bicyclic Peptide PET Probes Targeting Nectin-4”	47
Development of Broad-Spectrum Nanobodies for the Therapy and Diagnosis of SARS-CoV-2 and Its Multiple Variants	47
A Positron Emission Tomography Tracer Targeting the S2 Subunit of SARS-CoV-2 in Extrapulmonary Infections	45
Deconstructing Annealing Phenomena in Modified Release Lipid Multiparticulates	45
In Vitro Release from Polymeric Core/Shell Nanoparticles through the Lens of Multiscale Modeling	44
Mesoporous Matrices as a Promising New Generation of Carriers for Multipolymorphic Active Pharmaceutical Ingredient Aripiprazole	44
Fluorescent Self-Reporting Lipid Nanoparticles for Nitric Oxide/Gene Co-Delivery and Combination Therapy	43
Delivery and Expression of mRNA in the Secondary Lymphoid Organs Drive Immune Responses to Lipid Nanoparticle-mRNA Vaccines after Intramuscular Injection	41
⁶⁴Cu Radiolabeled PDGFRβ-Targeting Affibody for PET Imaging in Pancreatic Cancer	41
NIR-II Navigation with an EGFR-Targeted Probe Improves Imaging Resolution and Sensitivity of Detecting Micrometastases in Esophageal Squamous Cell Carcinoma Xenograft Models	40
Correlating Differences in the Surface Activity to Interface-Induced Particle Formation in Different Protein Modalities: IgG mAb Versus Fc-Fusion Protein	38
Highly Soluble Dacarbazine Multicomponent Crystals Less Prone to Photodegradation	38
Gold Nanoparticle-Decorated Drug Nanocrystals for Enhancing Anticancer Efficacy and Reversing Drug Resistance Through Chemo-/Photothermal Therapy	37
Co-amorphous Systems of Sinomenine with Platensimycin or Sulfasalazine: Physical Stability and Excipient-Adjusted Release Behavior	37
Stem Cell-Derived Extracellular Vesicles for Cancer Therapy and Tissue Engineering Applications	37
Exploring Bimetallic Nanoparticles in Alzheimer’s Therapy: A Novel Bio-Assisted Synthesis with Multitarget Potential	37
Lactoferrin-Modified Gambogic Acid Liposomes for Colorectal Cancer Treatment	36
Options of Therapeutics and Novel Delivery Systems of Drugs for the Treatment of Melanoma	35
Effects of Lyophilization, Vacuum Drying, and Microglassification on Two Model Proteins Assessed at the Residue Level Using Liquid Observed Vapor Exchange Nuclear Magnetic Resonance Spectroscopy (LOVE	35
Monoclonal Antibody Delivery Using 3D Printed Biobased Hollow μNe3dle Arrays for the Treatment of Osteoporosis	35
Influence of Nucleation on Relaxation, Molecular Cooperativity, and Physical Stability of Celecoxib Glass	35
Predicting Experimental B₂₂ Values and the Effects of Histidine Charge States for Monoclonal Antibodies Using Coarse-Grained Molecular Simulations	35
A Biopharmaceutical Perspective on Higher-Order Structure and Thermal Stability of mRNA Vaccines	34
The Dawn of a New Era: Tumor-Targeting Boron Agents for Neutron Capture Therapy	34
The Potency of Cowpea Mosaic Virus Particles for Cancer In Situ Vaccination Is Unaffected by the Specific Encapsidated Viral RNA	34
Knowledge Gaps in Generating Cell-Based Drug Delivery Systems and a Possible Meeting with Artificial Intelligence	33
pH-Responsive Liposomes Loaded with Targeting Procoagulant Proteins as Potential Embolic Agents for Solid Tumor-Targeted Therapy	33
Computational-Based Polyphenol Therapy for Nonsmall Cell Lung Cancer: Naringin Coamorphous Systems for Solubility and Bioavailability Enhancement	33
Defining the Intravital Renal Disposition of Fluorescence-Quenched Exenatide	32
Preparation of a Self-Assembled Rhein–Doxorubicin Nanogel Targeting Mitochondria and Investigation on Its Antihepatoma Activity	32
Bridging the Gap between Food Effects under Clinical Trial Conditions and Real Life: Modeling Delayed Gastric Emptying of Drug Substances and Gastric Content Volume Based on Meal Characteristics	32
Investigating Key Molecular Descriptors Affecting Particle Size: A Predictive Exemplary Approach for Self-Emulsifying System	32
New Model to Predict the Concentration-Dependent Viscosity of Monoclonal Antibody Solutions	31
Immuno-PET Imaging of TNF-α in Colitis Using ⁸⁹Zr-DFO-infliximab	31
Correction to Reshaping Tumor Blood Vessels to Enhance Drug Penetration with a Multistrategy Synergistic Nanosystem	31
[⁶⁴Cu]Cu(DDC)₂ NPs: A Novel PET Probe for Noninvasive Visualization of NPL4 Expression in Tumors In Vivo	31
Effect of Moisture Sorption and Lactose Type on Tablet Quality: A Hygroscopicity Study between Lactose Powder and Tablets	31
The Effect of Lipid Composition on the Liposomal Delivery of Camptothecin Developed by Active Click Loading	30
Mechanism-Based Pharmacokinetic Modeling of Absorption and Disposition of a Deferoxamine-Based Nanochelator in Rats	30
Cytidinyl/Cationic Lipid Encapsulating Insulin-Like Growth Factor 1 Receptor siRNA for Hepatocellular Carcinoma Therapy	30
Development of PLGA Nanoparticles with a Glycosylated Myelin Oligodendrocyte Glycoprotein Epitope (MOG_35–55) against Experimental Autoimmune Encephalomyelitis (EAE)	30
Assessment of In Vitro Models of the Human Buccal Mucosa for Vaccine and Adjuvant Development	30
Synthesis, Molecular Docking, and Biological Activity of New EGFR-Targeted Photosensitizers Based on Cationic Porphyrins Encapsulated into Pluronic F127 Micelles	30
iBCS: 1. Principles and Framework of an Inhalation-Based Biopharmaceutics Classification System	29
Clinical and Preclinical Methods of Heat-Stabilization of Human Vaccines	29
Phytochemical-Based Nanomedicine for Targeting Tumor Microenvironment and Inhibiting Cancer Chemoresistance: Recent Advances and Pharmacological Insights	29
Targeted Hyperbranched Nanoparticles for Delivery of Doxorubicin in Breast Cancer Brain Metastasis	28
Prediction of Multi-Pharmacokinetics Property in Multi-Species: Bayesian Neural Network Stacking Model with Uncertainty	28
Optimizing Drug Development: Harnessing the Sustainability of Pharmaceutical Cocrystals	28
Optimizing siRNA Therapeutics Targeting HIF-1α: Computational Design, Screening, and Molecular Dynamics Simulation Studies	28

Development of Edaravone Ionic Liquids and Their Application for the Treatment of Cerebral Ischemia/Reperfusion Injury	28
Development of a Specifically Labeled ⁸⁹Zr Antibody for the Noninvasive Imaging of Tumors Overexpressing B7-H3	28
Longitudinal MicroSPECT Imaging of Systemic Sclerosis Model Mice with [^99mTc]Tc-HYNFA via Folate Receptor Targeting	27
Functional Characterization of Six SLCO1B1 (OATP1B1) Variants Observed in Finnish Individuals with a Psychotic Disorder	27
Azide-Locked Prodrug Co-Assembly into Nanoparticles with Indocyanine Green for Chemophotothermal Therapy	27
Intradermal Injection of a Thermoresponsive Polymeric Dexamethasone Prodrug (ProGel-Dex) Ameliorate Dermatitis in an Imiquimod (IMQ)-Induced Psoriasis-like Mouse Model	27
Quantitative Analysis of Drug Supersaturation Region by Temperature-Variable Nuclear Magnetic Resonance Measurements, Part 2: Effects of Solubilizer	27
Correction to “Novel HER2-Targeted Peptide for NIR-II Imaging of Tumor”	27
Opto-Laser-Responsive Smart NanoGel with Mild Hyperthermia, Vascularization, and Anti-Inflammatory Potential for Boosting Hard-to-Heal Wounds in a Diabetic Mice Model	26
Biomimetic Nanoparticles Loaded with Ulinastatin for the Targeted Treatment of Acute Pancreatitis	26
Polymeric Iron Chelators Enhancing Pro-Oxidant Antitumor Efficacy of Vitamin C by Inhibiting the Extracellular Fenton Reaction	26
Therapeutic Immunomodulation of Tumor-Lymphatic Crosstalk via Intratumoral Immunotherapy	26
Correction to “H₂O₂ Self-Supplying and GSH-Depleting Nanocatalyst for Copper Metabolism-Based Synergistic Chemodynamic Therapy and Chemotherapy”	26
Radiation-Activated Cobalamin-Kinase Inhibitors for Treatment of Pancreatic Ductal Adenocarcinoma	26
Molecular Recognition Study toward the Mitochondrial Electron Transport Chain Inhibitor Mubritinib and Human Serum Albumin	26
Can Continuous Manufacturing of Topical Semisolids by Hot Melt Extrusion Soon Be a Reality?	25
Self-Delivery Nanoplatform Based on Amphiphilic Apoptosis Peptide for Precise Mitochondria-Targeting Photothermal Therapy	25
Utilizing Monocarboxylate Transporter 1-Mediated Blood–Brain Barrier Penetration for Glioblastoma Positron Emission Tomography Imaging with 6-[¹⁸F]Fluoronicotinic Acid	25
AF4 and PEG Precipitation as Predictive Assays for Antibody Self-Association	25
The pH-Dependent Microspecies Dissociations in the Trade-Off of Solubility and Permeability of Vitamin B2 Eutectic Solids	25
Top Cited Articles in Molecular Pharmaceutics: Leading Trends in Pharmaceutical Research	25
Liposomal Copermeation Assay Reveals Unexpected Membrane Interactions of Commonly Prescribed Drugs	24
Voices in Molecular Pharmaceutics: Meet Yan Shan Loo, a Graduate Student Exploring Nanoformulations of Natural Products	24
Glatiramer Acetate Complexes CpG Oligodeoxynucleotides into Nanoparticles and Boosts Their TLR9-Driven Immunity	24
Investigation of Tumor Cells and Receptor-Ligand Simulation Models for the Development of PET Imaging Probes Targeting PSMA and GRPR and a Possible Crosstalk between the Two Receptors	24
Voices in Molecular Pharmaceutics: Meet Dr. Weijun Wei Who Is Developing Theranostic Nuclear Medicine Agents for Clinical Use	24
Propionic Acid Groups and Multiple Aromatic Rings Induce Binding of Ketoprofen and Naproxen to the Hydrophobic Core of Bovine Serum Albumin	24
Advances in Structure Pharmaceutics from Discovery to Evaluation and Design	24
Issue Editorial Masthead	23
Issue Publication Information	23
In Vitro and In Vivo Study of Novel PSMA-Targeted Radioligands: Enhancing Tumor Uptake and Therapeutic Efficacy through Zwitterionization and Albumin-Binding Strategies	23
Issue Publication Information	23
Bile Salts Trigger Deformability in Liposomal Vesicles through Edge-Activating Action	23
Issue Editorial Masthead	23
Folate Receptor-Targeted Liposomes Loaded with Actinomycin X2 Enhance Antitumor Potency for HCCLM3 Hepatocellular Carcinoma Both In Vitro and In Vivo	23
Structural Similarity of Biological Drugs Using Statistical Signal Processing and Nuclear Magnetic Resonance Spectral Pattern Analysis	22
Mechanisms and Extent of Enhanced Passive Permeation by Colloidal Drug Particles	22
An Insight on Pillararene-Functionalized Mesoporous Silica Nanoparticles for Targeted Drug Delivery and Theranostics in Cancer	22
Dual Tumor-Selective β-Carboline-Based Fluorescent Probe for High-Contrast/Rapid Diagnosis of Clinical Tumor Tissues	22
Kinase Drug Discovery: Impact of Open Science and Artificial Intelligence	22
Transdermal Drug Delivery Systems (TDDS): Recent Advances and Failure Modes	22
A Pectin-Based Delivery Nanoplatform with an Optimized Tradeoff between Active Targeting and Drug Loading for Hepatocellular Carcinoma Treatment	22
Magnetic Resonance Imaging of Fibroblast Activation Protein Using a Targeted Gadolinium-Based Contrast Agent	22
Physiologically Based Pharmacokinetic Modeling of Phosphate Prodrugs─Case Studies: Fostemsavir and Fostamatinib	22
Nanoparticle-Reinforced Tough Hydrogel as a Versatile Platform for Pharmaceutical Drug Delivery: Preparation and in Vitro Characterization	22
Stimuli-Responsive and Receptor-Targeted Carbon Nanotubes for Multimodal Cancer Therapy and Diagnosis	22
Investigation of Praziquantel/Cyclodextrin Inclusion Complexation by NMR and LC-HRMS/MS: Mechanism, Solubility, Chemical Stability, and Degradation Products	22
Preclinical Evaluation and First-in-Human Study of [⁶⁸Ga]Ga-αvβ6–2: A Novel Dimeric Integrin αvβ6-Targeted PET Probe for Pancreatic Cancer Imaging	22
Correction to “Selecting Counterions to Improve Ionized Hydrophilic Drug Encapsulation in Polymeric Nanoparticles”	21
Dimeric Artesunate–Phosphatidylcholine-Based Liposomes for Irinotecan Delivery as a Combination Therapy Approach	21
Impact of Storage Conditions on the Physical Stability of Amorphous Solid Dispersions Containing Two Structurally Similar Drugs	21
Exploring the Predictive Power of the In Situ Perfusion Technique towards Drug Absorption: Theory, Practice, and Applications	21
Implications of the Digestion of Milk-Based Formulations for the Solubilization of Lopinavir/Ritonavir in a Combination Therapy	21
A CAIX Dual-Targeting Small-Molecule Probe for Noninvasive Imaging of ccRCC	21
An Artificial Gut/Absorption Simulator: Understanding the Impact of Absorption on In Vitro Dissolution, Speciation, and Precipitation of Amorphous Solid Dispersions	21
Compatibility between Proteins and Polysaccharide Excipients in Oral Delivery Tablets	21
Regional Transcriptomics and Proteomics of Pharmacokinetics-Related Genes in Human Intestine	21
Imaging Very Late Antigen-4 on MOLT4 Leukemia Tumors with Cysteine Site-Specific ⁸⁹Zr-Labeled Natalizumab Immuno-Positron Emission Tomography	21
CD7-Targeted Cytotoxic Potency of Diphtheria Toxin- and Ricin-Based Immunotoxins in Targeted Therapy for T-Cell Acute Lymphoblastic Leukemia	21
Impact of Polymers on the Kinetics of the Solid-State Phase Transition of Piracetam Polymorphs	21
Development of an ¹¹¹In-Labeled Glucagon-Like Peptide-1 Receptor-Targeting Exendin-4 Derivative that Exhibits Reduced Renal Uptake	20
Tumor-Repopulating Cell-Derived Microparticle-Based Therapeutics Amplify the Antitumor Effect through Synergistic Inhibition of Chemoresistance and Immune Evasion	20
Voices in Molecular Pharmaceutics: Meet Dr. Zahari Vinarov, Who Unites Physical Chemistry and Pharmacy to Tackle Fundamental and Industrial Biopharmaceutical Challenges	20
Networking in the Pharmaceutical Sciences	20
Pharmacokinetic–Pharmacodynamic Analysis of pH-Responsive Doxorubicin-Releasing Micelles with Anticancer Activity	20
Endogenous Iron(II) Self-Enriched Fenton Nanocatalyst via FTH1 Activity Inhibition and Iron(III) Reduction for Amplified Cancer Ferroptosis Therapy	20
Dynamic Phase Behavior of Amorphous Solid Dispersions Revealed with In Situ Stimulated Raman Scattering Microscopy	20
Experimental and Numerical Integrated Strategy for the Optimization of Microfluidic Parameters for Eudragit L100 Nanoparticles and Microparticles	20
Combined Probe Strategy to Increase the Enzymatic Digestion Rate and Accelerate the Renal Radioactivity Clearance of Peptide Radiotracers	20
Bootstrap Statistics and Its Application in Disintegration and Dissolution Data Analysis	20
Utility of Intravenous Curcumin Nanodelivery Systems for Improving In Vivo Pharmacokinetics and Anticancer Pharmacodynamics	20
Research Progress on Nanoplatforms and Nanotherapeutic Strategies in Treating Glioma	20
Construction of SLC16A1/3 Targeted Gallic Acid-Iron-Embelin Nanoparticles for Regulating Glycolysis and Redox Pathways in Cervical Cancer	20
Development of an Injectable Formulation of a Water-Insoluble Glycyrrhizin Derivative That Potently Inhibits High-Mobility Group Box 1 in Murine Intracerebral Hemorrhage	20
Small Scale, Big Impact: Nanotechnology-Enhanced Drug Delivery for Brain Diseases	20
Fe(II)-Targeted PET/¹⁹F MRI Dual-Modal Molecular Imaging Probe for Early Evaluation of Anticancer Drug-Induced Acute Kidney Injury	19
A Synergistically Enhanced Near-Infrared ESIPT Fluorescent Probe for High-Performance In Situ Imaging of Cellular Apoptosis	19
Radioactive and Fluorescent Dual Modality Cysteine Cathepsin B Activity-Based Probe for Cancer Theranostics	19
Issue Publication Information	19
Improvement in Inhalation Properties of Theophylline and Levofloxacin by Co-Amorphization and Enhancement in Its Stability by Addition of Amino Acid as a Third Component	19

Magnetic Nanoworm-Based Screening of Yeast Library for Anti-PEG Nanobodies	19
Sensitive Positron Emission Tomography Imaging of PD-L1 Expression in Human Breast and Lung Carcinoma Xenografts Using the Radiometalated Peptide Ga-68-TRAP-WL12	19
Smart SPIONs for Multimodal Cancer Theranostics: A Review	19
GSH-Responsive Prodrug Nanoassembly as a Carrier-Free Nanoplatform for Tumor-Targeting Delivery and Chemo-Photothermal Therapy	19
Tumor Microenvironment Responsive RNA Drug Delivery Systems: Intelligent Platforms for Sophisticated Release	19
Hydrogels as a Potential Biomaterial for Multimodal Therapeutic Applications	19
Insights into Factors Affecting Ethylene-Vinyl Acetate Copolymer Crystallinity in Islatravir Implant	19
Thermodynamic Perspectives on the Impact of a Second Drug on Amorphous Drug Solubility	19
New Radiolabeled Exendin Analogues Show Reduced Renal Retention	19
Tranexamic Acid-Based Polymeric Micellar Hydrogel for Enhanced Dermal Delivery and Melanin Reduction	19
Non-Viral RNA Therapies for Non-Small Cell Lung Cancer and Their Corresponding Clinical Trials	18
Insights into the Structure of Sucralfate by Advanced Solid- and Liquid-State NMR	18
Issue Publication Information	18
Preparation of Compound Salvia miltiorrhiza–Blumea balsamifera Nanoemulsion Gel and Its Effect on Hypertrophic Scars in the Rabbit Ear Model	18
Caffeic Acid-Grafted PLGA as a Novel Material for the Design of Fluvastatin-Eluting Nanoparticles for the Prevention of Neointimal Hyperplasia	18
Systematic Evaluation of Local and Global Machine Learning Models for the Prediction of ADME Properties	18
Recent Updates on Viral Oncogenesis: Available Preventive and Therapeutic Entities	18
Dumbbell-Shaped Antisense Oligonucleotide Prodrugs Showed Improved Antinuclease Stability and Anticancer Efficacy	18
Multimodal Imaging Response after the Singular or Combination Treatments of Vascular Endothelial Growth Factor Inhibitor and Immune Checkpoint Inhibitor	18
Ultrasound-Driven Nitric Oxide Generation for Enhanced Sonodynamic–Photothermal Therapy	18
¹²⁴I-Labeled Immuno-PET Targeting hTREM2 for the Diagnosis of Gastric Carcinoma	18
Cocrystallization Enables Ensitrelvir to Overcome Anomalous Low Solubility Caused by Strong Intermolecular Interactions between Triazine–Triazole Groups in Stable Crystal Form	18
Developing an In Vitro to In Vivo Extrapolation (IVIVE) Model to Predict Human Milk-to-Plasma Drug Concentration Ratios	18
Gallium Mesoporphyrin IX-Mediated Photodestruction: A Pharmacological Trojan Horse Strategy To Eliminate Multidrug-Resistant Staphylococcus aureus	18
Bimetallic Gold/Silver and Bioactive Camptothecin Hybrid Nanoparticles for Eradication of Cancer Stem Cells in a Combination Manner	18
Novel Oxygen-Dependent Degradable Immunotoxin Regulated by the Ubiquitin–Proteasome System Reduces Nonspecific Cytotoxicity	18
Systemic and Local Administration of a Dual-siRNA Complex Efficiently Inhibits Tumor Growth and Bone Invasion in Oral Squamous Cell Carcinoma	18
Delivery of Anticancer Drugs Using Microbubble-Assisted Ultrasound in a 3D Spheroid Model	18
Design of Biopharmaceutical Formulations Accelerated by Machine Learning	18
Sweet Battle of the Epimers─Continued Exploration of Monosaccharide-Derived Delivery Agents for Boron Neutron Capture Therapy	18
NMR Reveals Functionally Relevant Thermally Induced Structural Changes within the Native Ensemble of G-CSF	18
Application of a CYP1B1-Targeted NIR Probe for Breast Cancer Diagnosis, Surgical Navigation, and CYP1B1-Associated Chemotherapy Resistance Monitoring	17
Development of ¹⁸F-Labeled Positron Emission Tomography Agents Targeting Fibroblast Activation Protein	17
Actionable Predictions of Human Pharmacokinetics at the Drug Design Stage	17
Crystallinity: A Complex Critical Quality Attribute of Amorphous Solid Dispersions	17
ROS-Responsive Prodrug Micelle Co-Delivery System for Synergistic Antiatherosclerotic Therapy	17
Reconstituted Lipid Nanoparticles from Cells/Tissues for Drug Delivery in Cancer	17
Potentiation of Brain Bioavailability Using Thermoreversible Cubosomal Formulation	17
Study of Disordered Mesoporous Silica Regarding Intrinsic Compound Affinity to the Carrier and Drug-Accessible Surface Area	17
Effects of Polymers on Cocrystal Growth in a Drug–Drug Coamorphous System: Relations between Glass-to-Crystal Growth and Surface-Enhanced Crystal Growth	17
Miniaturized High-Throughput Amorphous Solid Dispersion Screening via Picoliter Volume 2D-Inkjet Printing of Formulation Microarrays	17
Early Prediction of Radiation-Induced Pulmonary Fibrosis Using Gastrin-Releasing Peptide Receptor-Targeted PET Imaging	17
Issue Editorial Masthead	17
Issue Publication Information	17
Distinctive Membrane Accommodation Traits Underpinning the Neutralization Activity of HIV-1 Antibody against MPER	17
Prospective Study Comparing [^99mTc]Tc-DP-FAPI Quantitative SPECT/CT with [⁶⁸Ga]Ga-FAPI-04 PET/CT in Patients with Gastrointestinal Tumors	17
In Vivo Delivery of siRNAs Targeting EGFR and BRD4 Expression by Peptide-Modified Redox Responsive PEG–PEI Nanoparticles for the Treatment of Triple-Negative Breast Cancer	17
Voriconazole–Cyclodextrin Supramolecular Ternary Complex-Loaded Ocular Films for Management of Fungal Keratitis	17
Polyphosphazene: A New Adjuvant Platform for Cocaine Vaccine Development	17
Evaluation of a CD206-Targeted Peptide for PET Imaging of Macrophages in Syngeneic Mouse Models of Cancer	17
Issue Editorial Masthead	17
Comparative Evaluation of Dissolution Performance in a USP 2 Setup and Alternative Stirrers and Vessel Designs: A Systematic Computational Investigation	17
Extracellular Vesicles Derived from Human Umbilical Cord MSC Improve Vascular Endothelial Function in In Vitro and In Vivo Models of Preeclampsia through Activating Arginine Metabolism	17
Targeted Delivery Platforms for the Treatment of Multiple Sclerosis	17
Effective Treatment of SSTR2-Positive Small Cell Lung Cancer Using ²¹¹At-Containing Targeted α-Particle Therapy Agent Which Promotes Endogenous Antitumor Immune Response	17
Fast-Disintegrating Nanofibrous Web of Pullulan/Griseofulvin–Cyclodextrin Inclusion Complexes	17
Engineered Fenofibrate as Oxidation-Sensitive Nanoparticles with ROS Scavenging and PPARα-Activating Bioactivity to Ameliorate Nonalcoholic Fatty Liver Disease	17
Toward “CO in a Pill”: Silica-Immobilized Organic CO Prodrugs for Studying the Feasibility of Systemic Delivery of CO via In Situ Gastrointestinal CO Release	17
Inhomogeneous Phase Significantly Reduces Oral Bioavailability of Felodipine/PVPVA Amorphous Solid Dispersion	17
Interactions of Sucrose and Trehalose with Lysozyme in Different Media: A Perspective from Atomistic Molecular Dynamics Simulations	16
Binding of the B-Raf Inhibitors Dabrafenib and Vemurafenib to Human Serum Albumin: A Biophysical and Molecular Simulation Study	16
3D-Printed Integrated Ultrasonic Microneedle Array for Rapid Transdermal Drug Delivery	16
Recent Advancement of Indocyanine Green Based Nanotheranostics for Imaging and Therapy of Coronary Atherosclerosis	16
Coacervation in Slow Motion: Kinetics of Complex Micelle Formation Induced by the Hydrolysis of an Antibiotic Prodrug	16
Aggregation Behavior of Structurally Similar Therapeutic Peptides Investigated by ¹H NMR and All-Atom Molecular Dynamics Simulations	16
Oxygenated Wound Dressings for Hypoxia Mitigation and Enhanced Wound Healing	16
In Silico Modeling Approaches Coupled with In Vitro Characterization in Predicting In Vivo Performance of Drug Delivery System Formulations	16
Quality by Design Considerations for Drop-on-Demand Point-of-Care Pharmaceutical Manufacturing of Precision Medicine	16
Where Might Artificial Intelligence Be Going in Pharmaceutical Development?	16
Unlocking the Gates: Therapeutic Agents for Noninvasive Drug Delivery Across the Blood-Brain Barrier	16
Nanoparticle-Based Drug Delivery System: The Magic Bullet for the Treatment of Chronic Pulmonary Diseases	16
Insights into the Impact of Nanostructural Properties on Powder Tribocharging: The Case of Milled Salbutamol Sulfate	16
Hybrid Micelles of Carbon Quantum Dot–Doxorubicin Conjugates as Nanotheranostics for Tumor Therapy and Turn-On Fluorescence Imaging: Impact of Conjugated Structures and On–Off–On Mechanism	16
Development of a Deep Eutectic Solvent-Assisted Kaempferol Hydrogel: A Promising Therapeutic Approach for Psoriasis-like Skin Inflammation	16
The Molecular Size of Bioengineered Oxygen Carriers Determines Tissue Oxygenation in a Hypercholesterolemia Guinea Pig Model of Hemorrhagic Shock and Resuscitation	16
Enhanced Detection of Early Pulmonary Fibrosis Disease Using ⁶⁸Ga-FAPI-LM3 PET	16
Combining β-Carotene with 5-FU via Polymeric Nanoparticles as a Novel Therapeutic Strategy to Overcome uL3-Mediated Chemoresistance in p53-Deleted Colorectal Cancer Cells	16
Impact of Anti-PEG IgM Induced via the Topical Application of a Cosmetic Product Containing PEG Derivatives on the Antitumor Effects of PEGylated Liposomal Antitumor Drug Formulations in Mice	16
Synthesis and Preclinical Evaluation of a ⁶⁸Ga-Labeled Pyridine-Based Benzamide Dimer for Malignant Melanoma Imaging	16
Solid Dispersion Incorporated into Dissolving Microneedles for Improved Antifungal Activity of Amphotericin B: In Vivo Study in a Fungal Keratitis Model	16
Issue Publication Information	15
High-Density Lipoprotein Mimetic Peptide 4F Reduces Toxic Amyloid-Beta Exposure to the Blood-Brain Barrier Endothelium in Alzheimer’s Disease Transgenic Mice	15
Issue Publication Information	15
Leveraging a Dual Variable Domain Immunoglobulin to Create a Site-Specifically Modified Radioimmunoconjugate	15
Investigation of Optimum Production Conditions and the Stability of β-Cyclodextrin–Perfluorocarbon Nanocone Clusters for Histotripsy Applications	15
Enhanced Therapeutic Effect of Liposomal Doxorubicin via Bio-Orthogonal Chemical Reactions in Tumors	15
Synthesis and Preclinical Evaluation of PSMA-Targeted ¹¹¹In-Radioconjugates Containing a Mitochondria-Tropic Triphenylphosphonium Carrier	15
Issue Publication Information	15
Overcoming Resistance in Prostate Cancer Therapy Using a DZ-Simvastatin Conjugate	15
Hydrogen–Deuterium Exchange Dynamics of NISTmAb Measured by Small Angle Neutron Scattering	15
Injectable Biodegradable Silica Depot for Controlled Subcutaneous Delivery of Antisense Oligonucleotides with beyond Monthly Administration	15
Issue Editorial Masthead	15
Announcing the Winners of the 2025 Molecular Pharmaceutics Early Career Best Paper Award	15
Inductively Coupled Plasma Mass Spectrometry─A Valid Method for the Characterization of Metal Conjugates in View of the Development of Radiopharmaceuticals	15
In Vivo Profiling with ¹⁸F-YJH08 Reveals Diverse Tissue Patterns of Antagonist/Glucocorticoid Receptor Interactions	15