OOIR: Observatory of International Research

Papers

(The median citation count of Molecular Pharmaceutics is 3. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-05-01 to 2025-05-01.)

Article	Citations
High Molecular Weight Poly(glutamic acid) to Improve BMP2-Induced Osteogenic Differentiation	138
Microemulsion for Prolonged Release of Fenretinide in the Mammary Tissue and Prevention of Breast Cancer Development	107
Highly Soluble Dacarbazine Multicomponent Crystals Less Prone to Photodegradation	104
Development of Broad-Spectrum Nanobodies for the Therapy and Diagnosis of SARS-CoV-2 and Its Multiple Variants	78
A Model Study to Assess Fibrillation and Product Stability to Support Peptide Drug Design	74
Understanding the Roles of Excipients in Moisture Management in Solid Dosage Forms	72
Correlating Differences in the Surface Activity to Interface-Induced Particle Formation in Different Protein Modalities: IgG mAb Versus Fc-Fusion Protein	65
Coupled Discrete Phase and Eulerian Wall Film Models for Drug Deposition Efficacy Analysis in Human Respiratory Airways	62
Construction and Preclinical Evaluation of a ^124/125I-Labeled Specific Antibody Targeting PD-L2 in Lung Cancer	62
pH-Responsive Liposomes Loaded with Targeting Procoagulant Proteins as Potential Embolic Agents for Solid Tumor-Targeted Therapy	62
Computational-Based Polyphenol Therapy for Nonsmall Cell Lung Cancer: Naringin Coamorphous Systems for Solubility and Bioavailability Enhancement	62
NIR-II Navigation with an EGFR-Targeted Probe Improves Imaging Resolution and Sensitivity of Detecting Micrometastases in Esophageal Squamous Cell Carcinoma Xenograft Models	60
A Positron Emission Tomography Tracer Targeting the S2 Subunit of SARS-CoV-2 in Extrapulmonary Infections	58
Fluorophore-Conjugated Anti-ICOS Antibody Enables Precise Prediction of Therapeutic Response of the STING Agonist in Colorectal Cancer via NIRF Imaging	58
Analysis of Cimetidine Crystal Polymorphs by X-ray Absorption Near-Edge Spectroscopy	57
Evaluation of a Tumor-Targeting Oligosaccharide Nanosystem in BNCT on an Orthotopic Hepatocellular Carcinoma Model	55
Defining the Intravital Renal Disposition of Fluorescence-Quenched Exenatide	54
Quantitative Characterization of Clinically Relevant Drug-Metabolizing Enzymes and Transporters in Rat Liver and Intestinal Segments for Applications in PBPK Modeling	54
The Potency of Cowpea Mosaic Virus Particles for Cancer In Situ Vaccination Is Unaffected by the Specific Encapsidated Viral RNA	52
Stem Cell-Derived Extracellular Vesicles for Cancer Therapy and Tissue Engineering Applications	52
Lactoferrin-Modified Gambogic Acid Liposomes for Colorectal Cancer Treatment	52
Issue Editorial Masthead	52
Investigating Key Molecular Descriptors Affecting Particle Size: A Predictive Exemplary Approach for Self-Emulsifying System	49
Exploring Bimetallic Nanoparticles in Alzheimer’s Therapy: A Novel Bio-Assisted Synthesis with Multitarget Potential	49
Pharmacokinetic Bioequivalence between Generic and Originator Orally Inhaled Drug Products: Validity of Administration of Doses above the Approved Single Maximum Dose	48

Issue Publication Information	47
Structured Sponsorship: An Option for Improved Workplace Inclusion in the Pharmaceutical Sciences	47
Mechanical Extrusion of the Plasma Membrane to Generate Ectosome-Mimetic Nanovesicles for Lung Targeting	45
Issue Editorial Masthead	44
Exploration of Verticillins in High-Grade Serous Ovarian Cancer and Evaluation of Multiple Formulations in Preclinical In Vitro and In Vivo Models	43
Bridging the Gap between Food Effects under Clinical Trial Conditions and Real Life: Modeling Delayed Gastric Emptying of Drug Substances and Gastric Content Volume Based on Meal Characteristics	43
Invisible Bridges: Unveiling the Role and Prospects of Tunneling Nanotubes in Cancer Therapy	43
Predicting Experimental B₂₂ Values and the Effects of Histidine Charge States for Monoclonal Antibodies Using Coarse-Grained Molecular Simulations	42
Influence of Nucleation on Relaxation, Molecular Cooperativity, and Physical Stability of Celecoxib Glass	41
⁶⁴Cu Radiolabeled PDGFRβ-Targeting Affibody for PET Imaging in Pancreatic Cancer	41
Pharmacokinetics in Penguins Compared to Other Avian Species: A Review of Enrofloxacin and Voriconazole	40
The Dawn of a New Era: Tumor-Targeting Boron Agents for Neutron Capture Therapy	40
Delivery and Expression of mRNA in the Secondary Lymphoid Organs Drive Immune Responses to Lipid Nanoparticle-mRNA Vaccines after Intramuscular Injection	40
Options of Therapeutics and Novel Delivery Systems of Drugs for the Treatment of Melanoma	40
Pterostilbene-Loaded Soluplus/Poloxamer 188 Mixed Micelles for Protection against Acetaminophen-Induced Acute Liver Injury	38
A Biopharmaceutical Perspective on Higher-Order Structure and Thermal Stability of mRNA Vaccines	38
Monoclonal Antibody Delivery Using 3D Printed Biobased Hollow μNe3dle Arrays for the Treatment of Osteoporosis	38
Co-amorphous Systems of Sinomenine with Platensimycin or Sulfasalazine: Physical Stability and Excipient-Adjusted Release Behavior	36
Preparation of a Self-Assembled Rhein–Doxorubicin Nanogel Targeting Mitochondria and Investigation on Its Antihepatoma Activity	36
Fluorescent Self-Reporting Lipid Nanoparticles for Nitric Oxide/Gene Co-Delivery and Combination Therapy	36
Knowledge Gaps in Generating Cell-Based Drug Delivery Systems and a Possible Meeting with Artificial Intelligence	36
Deconstructing Annealing Phenomena in Modified Release Lipid Multiparticulates	35
Effect of Moisture Sorption and Lactose Type on Tablet Quality: A Hygroscopicity Study between Lactose Powder and Tablets	35
Immuno-PET Imaging of TNF-α in Colitis Using ⁸⁹Zr-DFO-infliximab	35
In Vitro Release from Polymeric Core/Shell Nanoparticles through the Lens of Multiscale Modeling	33
Issue Publication Information	33
Difference in Endocytosis Pathways Used by Differentiated Versus Nondifferentiated Epithelial Caco-2 Cells to Internalize Nanosized Particles	33
Transition Metal (Molybdenum)-Doped Drug-like Conformational Nanoarchitectonics with Altered Valence States (Mn²⁺/Mn⁴⁺ and Mo⁵⁺/Mo⁶⁺) for Augmented Cancer T	33
Mesoporous Matrices as a Promising New Generation of Carriers for Multipolymorphic Active Pharmaceutical Ingredient Aripiprazole	33
Gold Nanoparticle-Decorated Drug Nanocrystals for Enhancing Anticancer Efficacy and Reversing Drug Resistance Through Chemo-/Photothermal Therapy	33
Enhanced Therapeutic Efficacy Against Melanoma through Exosomal Delivery of Hesperidin	33
Voices in Molecular Pharmaceutics: Meet Dr. Weijun Wei Who Is Developing Theranostic Nuclear Medicine Agents for Clinical Use	32
Voices in Molecular Pharmaceutics: Meet Yan Shan Loo, a Graduate Student Exploring Nanoformulations of Natural Products	32
Top Cited Articles in Molecular Pharmaceutics: Leading Trends in Pharmaceutical Research	32
[⁶⁴Cu]Cu(DDC)₂ NPs: A Novel PET Probe for Noninvasive Visualization of NPL4 Expression in Tumors In Vivo	32
Issue Editorial Masthead	31
Issue Publication Information	31
The pH-Dependent Microspecies Dissociations in the Trade-Off of Solubility and Permeability of Vitamin B2 Eutectic Solids	30
Clinical and Preclinical Methods of Heat-Stabilization of Human Vaccines	30
iBCS: 1. Principles and Framework of an Inhalation-Based Biopharmaceutics Classification System	30
Physiologically Based Pharmacokinetic Modeling of Phosphate Prodrugs─Case Studies: Fostemsavir and Fostamatinib	30
Liposomal Copermeation Assay Reveals Unexpected Membrane Interactions of Commonly Prescribed Drugs	29
Structural Similarity of Biological Drugs Using Statistical Signal Processing and Nuclear Magnetic Resonance Spectral Pattern Analysis	29
Nanoparticle-Reinforced Tough Hydrogel as a Versatile Platform for Pharmaceutical Drug Delivery: Preparation and in Vitro Characterization	29
Radiation-Activated Cobalamin-Kinase Inhibitors for Treatment of Pancreatic Ductal Adenocarcinoma	29
New Model to Predict the Concentration-Dependent Viscosity of Monoclonal Antibody Solutions	29
Phytochemical-Based Nanomedicine for Targeting Tumor Microenvironment and Inhibiting Cancer Chemoresistance: Recent Advances and Pharmacological Insights	28
Mechanisms and Extent of Enhanced Passive Permeation by Colloidal Drug Particles	28
Glatiramer Acetate Complexes CpG Oligodeoxynucleotides into Nanoparticles and Boosts Their TLR9-Driven Immunity	28
Propionic Acid Groups and Multiple Aromatic Rings Induce Binding of Ketoprofen and Naproxen to the Hydrophobic Core of Bovine Serum Albumin	28

Transdermal Drug Delivery Systems (TDDS): Recent Advances and Failure Modes	28
Development of a Specifically Labeled ⁸⁹Zr Antibody for the Noninvasive Imaging of Tumors Overexpressing B7-H3	28
Preclinical Evaluation and First-in-Human Study of [⁶⁸Ga]Ga-αvβ6–2: A Novel Dimeric Integrin αvβ6-Targeted PET Probe for Pancreatic Cancer Imaging	28
Investigation of Praziquantel/Cyclodextrin Inclusion Complexation by NMR and LC-HRMS/MS: Mechanism, Solubility, Chemical Stability, and Degradation Products	28
Magnetic Resonance Imaging of Fibroblast Activation Protein Using a Targeted Gadolinium-Based Contrast Agent	28
Targeted Hyperbranched Nanoparticles for Delivery of Doxorubicin in Breast Cancer Brain Metastasis	28
Therapeutic Immunomodulation of Tumor-Lymphatic Crosstalk via Intratumoral Immunotherapy	27
Azide-Locked Prodrug Co-Assembly into Nanoparticles with Indocyanine Green for Chemophotothermal Therapy	27
Prediction of Multi-Pharmacokinetics Property in Multi-Species: Bayesian Neural Network Stacking Model with Uncertainty	27
Intradermal Injection of a Thermoresponsive Polymeric Dexamethasone Prodrug (ProGel-Dex) Ameliorate Dermatitis in an Imiquimod (IMQ)-Induced Psoriasis-like Mouse Model	27
Longitudinal MicroSPECT Imaging of Systemic Sclerosis Model Mice with [^99mTc]Tc-HYNFA via Folate Receptor Targeting	27
Quantitative Analysis of Drug Supersaturation Region by Temperature-Variable Nuclear Magnetic Resonance Measurements, Part 2: Effects of Solubilizer	26
Biomimetic Nanoparticles Loaded with Ulinastatin for the Targeted Treatment of Acute Pancreatitis	26
Mechanism-Based Pharmacokinetic Modeling of Absorption and Disposition of a Deferoxamine-Based Nanochelator in Rats	26
Functional Characterization of Six SLCO1B1 (OATP1B1) Variants Observed in Finnish Individuals with a Psychotic Disorder	26
Advances in Structure Pharmaceutics from Discovery to Evaluation and Design	25
Molecular Recognition Study toward the Mitochondrial Electron Transport Chain Inhibitor Mubritinib and Human Serum Albumin	25
Can Continuous Manufacturing of Topical Semisolids by Hot Melt Extrusion Soon Be a Reality?	25
Correction to “H₂O₂ Self-Supplying and GSH-Depleting Nanocatalyst for Copper Metabolism-Based Synergistic Chemodynamic Therapy and Chemotherapy”	25
Correction to “Novel HER2-Targeted Peptide for NIR-II Imaging of Tumor”	25
Polymeric Iron Chelators Enhancing Pro-Oxidant Antitumor Efficacy of Vitamin C by Inhibiting the Extracellular Fenton Reaction	24
Dual Tumor-Selective β-Carboline-Based Fluorescent Probe for High-Contrast/Rapid Diagnosis of Clinical Tumor Tissues	24
Self-Delivery Nanoplatform Based on Amphiphilic Apoptosis Peptide for Precise Mitochondria-Targeting Photothermal Therapy	24
Issue Editorial Masthead	24
Isothermal Crystallization and Time–Temperature Transformation of Amorphous Nifedipine: A Case of Polymorphism Formation and Conversion	24
Assessment of In Vitro Models of the Human Buccal Mucosa for Vaccine and Adjuvant Development	23
Development of PLGA Nanoparticles with a Glycosylated Myelin Oligodendrocyte Glycoprotein Epitope (MOG_35–55) against Experimental Autoimmune Encephalomyelitis (EAE)	23
Development of Edaravone Ionic Liquids and Their Application for the Treatment of Cerebral Ischemia/Reperfusion Injury	23
Cytidinyl/Cationic Lipid Encapsulating Insulin-Like Growth Factor 1 Receptor siRNA for Hepatocellular Carcinoma Therapy	23
Kinase Drug Discovery: Impact of Open Science and Artificial Intelligence	23
The Effect of Lipid Composition on the Liposomal Delivery of Camptothecin Developed by Active Click Loading	23
Opto-Laser-Responsive Smart NanoGel with Mild Hyperthermia, Vascularization, and Anti-Inflammatory Potential for Boosting Hard-to-Heal Wounds in a Diabetic Mice Model	23
AF4 and PEG Precipitation as Predictive Assays for Antibody Self-Association	23
Investigation of Tumor Cells and Receptor-Ligand Simulation Models for the Development of PET Imaging Probes Targeting PSMA and GRPR and a Possible Crosstalk between the Two Receptors	23
Exploring the Predictive Power of the In Situ Perfusion Technique towards Drug Absorption: Theory, Practice, and Applications	22
Construction of SLC16A1/3 Targeted Gallic Acid-Iron-Embelin Nanoparticles for Regulating Glycolysis and Redox Pathways in Cervical Cancer	22
Nanostructured Valsartan Microparticles with Enhanced Bioavailability Produced by High-Throughput Electrohydrodynamic Room-Temperature Atomization	22
Implications of the Digestion of Milk-Based Formulations for the Solubilization of Lopinavir/Ritonavir in a Combination Therapy	22
Developing an In Vitro to In Vivo Extrapolation (IVIVE) Model to Predict Human Milk-to-Plasma Drug Concentration Ratios	22
Non-Viral RNA Therapies for Non-Small Cell Lung Cancer and Their Corresponding Clinical Trials	22
Optimizing Drug Development: Harnessing the Sustainability of Pharmaceutical Cocrystals	22
An Artificial Gut/Absorption Simulator: Understanding the Impact of Absorption on In Vitro Dissolution, Speciation, and Precipitation of Amorphous Solid Dispersions	22
Regional Transcriptomics and Proteomics of Pharmacokinetics-Related Genes in Human Intestine	22
GSH-Responsive Prodrug Nanoassembly as a Carrier-Free Nanoplatform for Tumor-Targeting Delivery and Chemo-Photothermal Therapy	21
Sweet Battle of the Epimers─Continued Exploration of Monosaccharide-Derived Delivery Agents for Boron Neutron Capture Therapy	21
Ultrasound-Driven Nitric Oxide Generation for Enhanced Sonodynamic–Photothermal Therapy	21
Correction to “Selecting Counterions to Improve Ionized Hydrophilic Drug Encapsulation in Polymeric Nanoparticles”	21
Combined Probe Strategy to Increase the Enzymatic Digestion Rate and Accelerate the Renal Radioactivity Clearance of Peptide Radiotracers	21
Development of an ¹¹¹In-Labeled Glucagon-Like Peptide-1 Receptor-Targeting Exendin-4 Derivative that Exhibits Reduced Renal Uptake	21
Fe(II)-Targeted PET/¹⁹F MRI Dual-Modal Molecular Imaging Probe for Early Evaluation of Anticancer Drug-Induced Acute Kidney Injury	21
¹²⁴I-Labeled Immuno-PET Targeting hTREM2 for the Diagnosis of Gastric Carcinoma	21
Smart SPIONs for Multimodal Cancer Theranostics: A Review	21
Small Scale, Big Impact: Nanotechnology-Enhanced Drug Delivery for Brain Diseases	21
Imaging Very Late Antigen-4 on MOLT4 Leukemia Tumors with Cysteine Site-Specific ⁸⁹Zr-Labeled Natalizumab Immuno-Positron Emission Tomography	21
Development of an Injectable Formulation of a Water-Insoluble Glycyrrhizin Derivative That Potently Inhibits High-Mobility Group Box 1 in Murine Intracerebral Hemorrhage	21
A CAIX Dual-Targeting Small-Molecule Probe for Noninvasive Imaging of ccRCC	21
Insights into Factors Affecting Ethylene-Vinyl Acetate Copolymer Crystallinity in Islatravir Implant	21
Tumor Microenvironment Responsive RNA Drug Delivery Systems: Intelligent Platforms for Sophisticated Release	20
Sensitive Positron Emission Tomography Imaging of PD-L1 Expression in Human Breast and Lung Carcinoma Xenografts Using the Radiometalated Peptide Ga-68-TRAP-WL12	20
Caffeic Acid-Grafted PLGA as a Novel Material for the Design of Fluvastatin-Eluting Nanoparticles for the Prevention of Neointimal Hyperplasia	20
Systematic Evaluation of Local and Global Machine Learning Models for the Prediction of ADME Properties	20
Gallium Mesoporphyrin IX-Mediated Photodestruction: A Pharmacological Trojan Horse Strategy To Eliminate Multidrug-Resistant Staphylococcus aureus	20
Impact of Storage Conditions on the Physical Stability of Amorphous Solid Dispersions Containing Two Structurally Similar Drugs	20
Utility of Intravenous Curcumin Nanodelivery Systems for Improving In Vivo Pharmacokinetics and Anticancer Pharmacodynamics	20
Recent Updates on Viral Oncogenesis: Available Preventive and Therapeutic Entities	20
NMR Reveals Functionally Relevant Thermally Induced Structural Changes within the Native Ensemble of G-CSF	19
Tumor-Repopulating Cell-Derived Microparticle-Based Therapeutics Amplify the Antitumor Effect through Synergistic Inhibition of Chemoresistance and Immune Evasion	19
In Vivo Induction of P-Glycoprotein Function can be Measured with [¹⁸F]MC225 and PET	19
Halogenation at the Phenylalanine Residue of Monomethyl Auristatin F Leads to a Favorable cis/trans Equilibrium and Retained Cytotoxicity	19
Radioactive and Fluorescent Dual Modality Cysteine Cathepsin B Activity-Based Probe for Cancer Theranostics	19
Dynamic Phase Behavior of Amorphous Solid Dispersions Revealed with In Situ Stimulated Raman Scattering Microscopy	19
Issue Publication Information	19
Cocrystallization Enables Ensitrelvir to Overcome Anomalous Low Solubility Caused by Strong Intermolecular Interactions between Triazine–Triazole Groups in Stable Crystal Form	19
Impact of Polymers on the Kinetics of the Solid-State Phase Transition of Piracetam Polymorphs	19
Pharmacokinetic–Pharmacodynamic Analysis of pH-Responsive Doxorubicin-Releasing Micelles with Anticancer Activity	19
New Radiolabeled Exendin Analogues Show Reduced Renal Retention	19
Bimetallic Gold/Silver and Bioactive Camptothecin Hybrid Nanoparticles for Eradication of Cancer Stem Cells in a Combination Manner	19
Networking in the Pharmaceutical Sciences	19
Dimeric Artesunate–Phosphatidylcholine-Based Liposomes for Irinotecan Delivery as a Combination Therapy Approach	19
Experimental and Numerical Integrated Strategy for the Optimization of Microfluidic Parameters for Eudragit L100 Nanoparticles and Microparticles	19

Voices in Molecular Pharmaceutics: Meet Dr. Zahari Vinarov, Who Unites Physical Chemistry and Pharmacy to Tackle Fundamental and Industrial Biopharmaceutical Challenges	19
Endogenous Iron(II) Self-Enriched Fenton Nanocatalyst via FTH1 Activity Inhibition and Iron(III) Reduction for Amplified Cancer Ferroptosis Therapy	19
Bootstrap Statistics and Its Application in Disintegration and Dissolution Data Analysis	18
Hydrogels as a Potential Biomaterial for Multimodal Therapeutic Applications	18
Binding of the B-Raf Inhibitors Dabrafenib and Vemurafenib to Human Serum Albumin: A Biophysical and Molecular Simulation Study	18
Comparative Evaluation of Dissolution Performance in a USP 2 Setup and Alternative Stirrers and Vessel Designs: A Systematic Computational Investigation	18
mPEG_2k-PCL_x Polymeric Micelles Influence Pharmacokinetics and Hypoglycemic Efficacy of Metformin through Inhibition of Organic Cation Transporters in Rats	18
Improvement in Inhalation Properties of Theophylline and Levofloxacin by Co-Amorphization and Enhancement in Its Stability by Addition of Amino Acid as a Third Component	18
Design of Biopharmaceutical Formulations Accelerated by Machine Learning	18
Prospective Study Comparing [^99mTc]Tc-DP-FAPI Quantitative SPECT/CT with [⁶⁸Ga]Ga-FAPI-04 PET/CT in Patients with Gastrointestinal Tumors	18
Systemic and Local Administration of a Dual-siRNA Complex Efficiently Inhibits Tumor Growth and Bone Invasion in Oral Squamous Cell Carcinoma	18
Insights into the Structure of Sucralfate by Advanced Solid- and Liquid-State NMR	18
Enhanced Detection of Early Pulmonary Fibrosis Disease Using ⁶⁸Ga-FAPI-LM3 PET	18
Research Progress on Nanoplatforms and Nanotherapeutic Strategies in Treating Glioma	18
Preparation of Compound Salvia miltiorrhiza–Blumea balsamifera Nanoemulsion Gel and Its Effect on Hypertrophic Scars in the Rabbit Ear Model	18
Effects of Polymers on Cocrystal Growth in a Drug–Drug Coamorphous System: Relations between Glass-to-Crystal Growth and Surface-Enhanced Crystal Growth	18
Delivery of Anticancer Drugs Using Microbubble-Assisted Ultrasound in a 3D Spheroid Model	18
Oligomerization of Pharmaceutically Relevant Insulin Analogues for Varying Concentration and Salinity Revealed by Small-Angle X-ray Scattering	18
Study of Disordered Mesoporous Silica Regarding Intrinsic Compound Affinity to the Carrier and Drug-Accessible Surface Area	18
Novel Oxygen-Dependent Degradable Immunotoxin Regulated by the Ubiquitin–Proteasome System Reduces Nonspecific Cytotoxicity	17
Early Prediction of Radiation-Induced Pulmonary Fibrosis Using Gastrin-Releasing Peptide Receptor-Targeted PET Imaging	17
Issue Editorial Masthead	17
Application of a CYP1B1-Targeted NIR Probe for Breast Cancer Diagnosis, Surgical Navigation, and CYP1B1-Associated Chemotherapy Resistance Monitoring	17
Issue Editorial Masthead	17
Miniaturized High-Throughput Amorphous Solid Dispersion Screening via Picoliter Volume 2D-Inkjet Printing of Formulation Microarrays	17
In Silico Modeling Approaches Coupled with In Vitro Characterization in Predicting In Vivo Performance of Drug Delivery System Formulations	17
Dumbbell-Shaped Antisense Oligonucleotide Prodrugs Showed Improved Antinuclease Stability and Anticancer Efficacy	17
Inhomogeneous Phase Significantly Reduces Oral Bioavailability of Felodipine/PVPVA Amorphous Solid Dispersion	17
Issue Publication Information	17
The Molecular Size of Bioengineered Oxygen Carriers Determines Tissue Oxygenation in a Hypercholesterolemia Guinea Pig Model of Hemorrhagic Shock and Resuscitation	17
Combining β-Carotene with 5-FU via Polymeric Nanoparticles as a Novel Therapeutic Strategy to Overcome uL3-Mediated Chemoresistance in p53-Deleted Colorectal Cancer Cells	17
Multimodal Imaging Response after the Singular or Combination Treatments of Vascular Endothelial Growth Factor Inhibitor and Immune Checkpoint Inhibitor	17
Recent Advancement of Indocyanine Green Based Nanotheranostics for Imaging and Therapy of Coronary Atherosclerosis	17
Solid Dispersion Incorporated into Dissolving Microneedles for Improved Antifungal Activity of Amphotericin B: In Vivo Study in a Fungal Keratitis Model	17
Distinctive Membrane Accommodation Traits Underpinning the Neutralization Activity of HIV-1 Antibody against MPER	17
Coacervation in Slow Motion: Kinetics of Complex Micelle Formation Induced by the Hydrolysis of an Antibiotic Prodrug	17
Voriconazole–Cyclodextrin Supramolecular Ternary Complex-Loaded Ocular Films for Management of Fungal Keratitis	16
Preclinical Evaluation of a Fluorescent Probe Targeting Receptor CDCP1 for Identification of Ovarian Cancer	16
Evaluation of a CD206-Targeted Peptide for PET Imaging of Macrophages in Syngeneic Mouse Models of Cancer	16
Hybrid Micelles of Carbon Quantum Dot–Doxorubicin Conjugates as Nanotheranostics for Tumor Therapy and Turn-On Fluorescence Imaging: Impact of Conjugated Structures and On–Off–On Mechanism	16
Interactions of Sucrose and Trehalose with Lysozyme in Different Media: A Perspective from Atomistic Molecular Dynamics Simulations	16
Quality by Design Considerations for Drop-on-Demand Point-of-Care Pharmaceutical Manufacturing of Precision Medicine	16
Reconstituted Lipid Nanoparticles from Cells/Tissues for Drug Delivery in Cancer	16
Reversing Hypoxia with PLGA-Encapsulated Manganese Dioxide Nanoparticles Improves Natural Killer Cell Response to Tumor Spheroids	16
Unlocking the Gates: Therapeutic Agents for Noninvasive Drug Delivery Across the Blood-Brain Barrier	16
ROS-Responsive Prodrug Micelle Co-Delivery System for Synergistic Antiatherosclerotic Therapy	16
Macropinocytosis-Inducible Extracellular Vesicles Modified with Antimicrobial Protein CAP18-Derived Cell-Penetrating Peptides for Efficient Intracellular Delivery	16
Aggregation Behavior of Structurally Similar Therapeutic Peptides Investigated by ¹H NMR and All-Atom Molecular Dynamics Simulations	16
Nanoparticle-Based Drug Delivery System: The Magic Bullet for the Treatment of Chronic Pulmonary Diseases	16
Oxygenated Wound Dressings for Hypoxia Mitigation and Enhanced Wound Healing	16
Synthesis and Preclinical Evaluation of a ⁶⁸Ga-Labeled Pyridine-Based Benzamide Dimer for Malignant Melanoma Imaging	16
Impact of Anti-PEG IgM Induced via the Topical Application of a Cosmetic Product Containing PEG Derivatives on the Antitumor Effects of PEGylated Liposomal Antitumor Drug Formulations in Mice	16
Extracellular Vesicles Derived from Human Umbilical Cord MSC Improve Vascular Endothelial Function in In Vitro and In Vivo Models of Preeclampsia through Activating Arginine Metabolism	16
Where Might Artificial Intelligence Be Going in Pharmaceutical Development?	16
Targeted Delivery Platforms for the Treatment of Multiple Sclerosis	16
Crystallinity: A Complex Critical Quality Attribute of Amorphous Solid Dispersions	16
Toward “CO in a Pill”: Silica-Immobilized Organic CO Prodrugs for Studying the Feasibility of Systemic Delivery of CO via In Situ Gastrointestinal CO Release	16
Fast-Disintegrating Nanofibrous Web of Pullulan/Griseofulvin–Cyclodextrin Inclusion Complexes	16
Development of a Deep Eutectic Solvent-Assisted Kaempferol Hydrogel: A Promising Therapeutic Approach for Psoriasis-like Skin Inflammation	16
Potentiation of Brain Bioavailability Using Thermoreversible Cubosomal Formulation	16
In Vivo Delivery of siRNAs Targeting EGFR and BRD4 Expression by Peptide-Modified Redox Responsive PEG–PEI Nanoparticles for the Treatment of Triple-Negative Breast Cancer	16
Correction to “Comparative Physical Study of Three Pharmaceutically Active Benzodiazepine Derivatives: Crystalline versus Amorphous State and Crystallization Tendency”	15
Comparison of the Anti-inflammatory Activity and Cellular Interaction of Brush Polymer–N-Acetyl Cysteine Conjugates in Human and Murine Microglial Cell Lines	15
Issue Publication Information	15
Drug Delivery Angle for Various Atherosclerosis and Aneurysm Percentages of the Carotid Artery	15
Polyphosphazene: A New Adjuvant Platform for Cocaine Vaccine Development	15
Issue Publication Information	15
Three Strikingly Different Crystal Habits of Tadalafil: Design, Characterization, Pharmaceutical Performance, and Computational Studies	15
Ionizable Drug Self-Associations and the Solubility Dependence on pH: Detection of Aggregates in Saturated Solutions Using Mass Spectrometry (ESI-Q-TOF-MS/MS)	15
Voices in Molecular Pharmaceutics: Meet Professor Keisuke Ueda, Who Scrutinizes the Molecular-Level Properties of Drugs and Formulations Using NMR Spectroscopy	15
Crystallization Risk Assessment of Amorphous Solid Dispersions by Physical Shelf-Life Modeling: A Practical Approach	15
Study on Sulfamethoxazole–Piperazine Salt: A Mechanistic Insight into Simultaneous Improvement of Physicochemical Properties	15
Lactosylated Chitosan Nanoparticles Potentiate the Anticancer Effects of Telmisartan In Vitro and in a N-Nitrosodiethylamine-Induced Mice Model of Hepatocellular Carcinoma	15
Issue Editorial Masthead	15
Introducing the Molecular Pharmaceutics Special Issue on “Emerging Trends in Molecular Pharmaceutics across Australasia”	15
Comment on: “Codelivery of Gemcitabine and MUC1 Inhibitor Using PEG-PCL Nanoparticles for Breast Cancer Therapy”	15
3D-Printed Integrated Ultrasonic Microneedle Array for Rapid Transdermal Drug Delivery	15
Actionable Predictions of Human Pharmacokinetics at the Drug Design Stage	15
Investigating Generation of Antibodies against the Lipid Nanoparticle Vector Following COVID-19 Vaccination with an mRNA Vaccine	15
Injectable Biodegradable Silica Depot for Controlled Subcutaneous Delivery of Antisense Oligonucleotides with beyond Monthly Administration	15
Nanoparticle Fraught Liposomes: A Platform for Increased Antibiotic Selectivity in Multidrug Resistant Bacteria	15
Opportunities for Bioactive Glass in Gastrointestinal Conditions: A Review of Production Methodologies, Morphology, Composition, and Performance	15
Complexation Mechanisms of Aqueous Amylose: Molecular Dynamics Study Using 3-Pentadecylphenol	15
Binding of the Dual-Action Anti-Parkinsonian Drug AG-0029 to Dopamine D₂ and Histamine H₃ Receptors: A PET Study in Healthy Rats	15
Enhancing Antituberculosis Treatment Nanoparticles Encapsulated with Catalase and Levofloxacin Under Ultrasound Stimulation: A 3D Spheroid Study	15
Insights into the Impact of Nanostructural Properties on Powder Tribocharging: The Case of Milled Salbutamol Sulfate	15
Engineered Fenofibrate as Oxidation-Sensitive Nanoparticles with ROS Scavenging and PPARα-Activating Bioactivity to Ameliorate Nonalcoholic Fatty Liver Disease	15
Effective Treatment of SSTR2-Positive Small Cell Lung Cancer Using ²¹¹At-Containing Targeted α-Particle Therapy Agent Which Promotes Endogenous Antitumor Immune Response	15
Noninvasive Assessment of Renal Fibrosis of Chronic Kidney Disease in Rats by [⁶⁸Ga]Ga-FAPI-04 Small Animal PET/CT and Biomarkers	15
Integrative Salt Selection and Formulation Optimization: Perspectives of Disproportionation and Microenvironmental pH Modulation	15
Effect of Pharmaceutical Excipients on Intestinal Absorption of Metformin via Organic Cation-Selective Transporters	15
Announcing the Winners of the 2025 Molecular Pharmaceutics Early Career Best Paper Award	14
Large-Scale Compartmental Model-Based Study of Preclinical Pharmacokinetic Data and Its Impact on Compound Triaging in Drug Discovery	14
Investigation of Copper-64-Based Host–Guest Chemistry Pretargeted Positron Emission Tomography	14
⁶⁸Ga-Labeled Cystine Knot Peptide Targeting Integrin α_vβ₆ for Lung Cancer PET Imaging	14