Organic Letters

Papers
(The median citation count of Organic Letters is 5. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2022-01-01 to 2026-01-01.)
ArticleCitations
Visible-Light-Promoted Selenylative Radical Cyclization of 2-Vinyl-N-Aryl Imines to 3H-Indoles via Oxygen Photosensitization95
Ascomycotols A–C: Rare Sulfur/Sulfone-Containing Scaffolds from Mushroom Endophytes with Dual Anti-inflammatory and Antirenal Fibrosis Effects91
Deciphering Regulatory Proteins of Prenylated Protein via the FRET Technique Using Nitroso-Based Ene-Ligation and Sequential Azidation and Click Reaction85
Weak-Chelation Assisted Cobalt-Catalyzed C–H Bond Activation: An Approach Toward Regioselective Ethynylation of N-Aryl γ-Lactam84
Isolation and Bioinspired Total Synthesis of Rugosiformisin A, A Skeleton-Rearranged Abietane-Type Diterpenoid from Isodon rugosiformis80
Organocalcium-Complex-Catalyzed Dehydrogenative Silylation and Mono/Dihydrosilylation Tandem Reactions of Terminal Alkynes80
Nickel/SKP-Catalyzed Markovnikov Regio- and Enantioselective Hydroamination of Vinylarenes with Hydroxylamines79
Selective C–H Iodination of Weinreb Amides and Benzamides through Iridium Catalysis in Solution and under Mechanochemical Conditions78
Enantioselective Annulation of α,β-Unsaturated N-Acyliminium Ions with β-Keto Ester Enolates via Cooperative Palladium and Brønsted Acid Catalysis75
Deprotonative Generation and Trapping of Haloaryllithium in a Batch Reactor74
Asymmetric Synthesis of β-Aminoboronates via Copper-Catalyzed Reductive Coupling of Vinyl Boronates with Imines71
Photoredox-Catalyzed Synthesis of β-Amino Alcohols: Hydroxymethylation of Imines with α-Silyl Ether as Hydroxymethyl Radical Precursor70
Visible-Light-Induced Difunctionalization of 3-Butenoic Acid with Bromodifluoromethyl Heteroarylsulfones69
Intramolecular Friedel–Crafts Reactions of Sulfamoyl Fluorides, Fluorosulfates, and Sulfuramidimidoyl Fluorides67
Nickel-Catalyzed Deaminative Allenylation of Amino Acid Derivatives: Catalytic Activity Enhanced by an Amide-Type NN2 Pincer Ligand66
On-DNA Deoxygenative C(sp 2 )–C(sp 3 ) Coupling Facilitated by Surfactant–DNA (Surf-DNA) Workflow64
Syntheses and Properties of Hole-Transporting Biindenofluorenes64
Palladium-Catalyzed Asymmetric (3 + 2) Cycloaddition of 5-Allenyloxazolidine-2,4-Diones with Barbiturate-Derived Alkenes: Synthesis of Spirobarbiturate-γ-Lactams63
Palladium-Catalyzed Double ipso-Defluoroetherification of Allylic gem-Difluorides with Phenols or Alcohols61
Boron-Catalyzed Michael Reaction of Donor–Acceptor Carboxylic Acid Pairs Enabling Direct Synthesis of 1,5-Dicarboxylic Acids61
Photochemical “Cut and Sew” Transformations of Ethynylbenziodoxolone Reagents and Diazo Compounds61
Synthesis of a Phosphate-Bridged Photoaffinity Labeling Probe via Transesterification of Phenols and Alcohols60
Iridium-Catalyzed Regio- and Enantioselective C7-Allylic Alkylation of 4-Aminoindoles60
Copper-Catalyzed Chan–Lam Reaction and Sequential Oxidative Fischer Indole Synthesis to Prepare Indole Derivatives59
Domino Semipinacol/Iterative Aldol/Iso-Nazarov Cyclization to Triaryl-cyclopentenone: Enantioselective Synthesis of Combretastatin A-4 Analogues59
Cobalt-Catalyzed Intramolecular [4 + 2] Cycloaddition of Cyclopropyl-Capped Dienes with Alkynes/Alkenes/Allene and Reaction Mechanism59
Synthesis of the Tetracyclic Core of the Daphlongeranines58
Synthesis of Tertiary Amines through Extrusive Alkylation of Carbamates58
Asymmetric Synthesis of Chiral Aza-macrodiolides via Iridium-Catalyzed Cascade Allylation/Macrolactonization58
A Tsuji–Trost Reaction Using Free Carbenes as Nucleophiles: Palladium-Catalyzed Photoinduced Coupling of Acylsilanes with Allylic Alcohol Derivatives57
Lewis Acid-Catalyzed Annulations of Geminally Disubstituted Cyclopropanes with Aldehydes or 1,3,5-Triazinanes57
Hydrophilic Azide-Containing Amino Acid to Enhance the Solubility of Peptides for SPAAC Reactions56
Base Metal-Controlled Chemodivergent Cyclization of Propargylamines for the Atom-Economic Synthesis of Nitrogen Heterocycles56
Pd-Catalyzed Asymmetric Allylic Substitution Cascade of Substituted 4-Hydroxy-2H-pyrones with meso-Allyl Dicarbonates56
Ligand-Controlled Diastereodivergency in Propargylic Alkylation of Vinylogous Aza-Enamines: Construction of 1,3-Stereocenters55
Enantioselective Total Synthesis of (+)-Lucidumone via Organocatalytic Double Michael Addition55
Diversity-Oriented Synthesis of ERα Modulators via Mitsunobu Macrocyclization55
Copper-Catalyzed Coupling of N-Acyl-N′-Substituted Hydrazines with (Hetero)aryl Chlorides/Bromides55
Enantioselective Organocatalytic Conjugate Addition of Malonates to β,β-Disubstituted β-Trifluoromethyl Enones under High Pressure55
Conformationally Fluxional Pseudo-C2 Symmetric Decaphyrins (1.0.0.0.0.1.0.0.0.0) with Multiple m-Phenylene Subunits and Their Cyclic Bis-BODIPYs55
Photocatalyzed Aerobic Cross-Dehydrogenative Coupling of Diarylphosphine Oxides with Alcohols and Phenols55
Fluoranthene-Containing Distorted Nanographenes Exhibiting Two-Photon Absorption Response53
Palladium-Catalyzed Synthesis of Amino β-Lactones Using Aryl Amines and Alkenyl Carboxylic Acids53
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Vitamin B12 and Micellar Solution Enable Regioselective Ring Opening of Epoxides and Aziridines with Electrophilic Olefins50
Ni-Catalyzed Reductive Coupling of Acetals with Anhydrides and Vinyl Triflates via Single-Electron C–O Activation50
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Ruthenium(II)-Catalyzed C–H Activation/Annulation of 5-Phenyl-pyrroline-2-carboxylates with Alkynes: Synthesis of 2,3-Diphenylspiro-[indene-1,2′pyrrolidine]carboxylate Derivatives50
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New Approach to Assembling Nucleic Acid Dendrons on a Solid Phase50
Systematic Route to Construct the 5–5–6 Tricyclic Core of Furanobutenolide-Derived Cembranoids and Norcembranoids49
Visible-Light-Promoted Reduction of Epoxides, Hydroxysulfonates, and Halohydrines with Alkyltitanium Alkoxides49
Palladium-Catalyzed Domino Conversion of Aryl–Thianthreniums with Anhydrides: Rapidly Building Highly Functionalized Fluorenones49
Palladium-Catalyzed 1,2-Alkynylarylation of Vinyl Arenes with Haloalkynes and Arylboronic Acids49
Photochemical Organocatalytic Aerobic Cleavage of C═C Bonds Enabled by Charge-Transfer Complex Formation49
Regioselective Divergent Benzannulations of Vinyl Sulfoxonium Ylides with Electron-Deficient Alkynes49
Regioselective Alkylacylation of 1,3-Dienes by Merging N-Heterocyclic Carbene Catalysis with Photoinduced Palladium Catalysis48
DNA-Compatible Diversification of Indole π-Activated Alcohols via a Direct Dehydrative Coupling Strategy48
Stereoselective Double Spirocyclization of 2-Benzyl-3-alkynyl Chromone with Nitrone via Gold-Catalyzed Cascade Reactions48
Solid-Phase Total Synthesis of Plusbacin A348
Photocatalytic Regioselective Alkoxycarbonylation/Cyclization of 3-Aza-1,5-dienes: Access to Ester-Containing Pyrrolin-2-ones48
Electrochemical Cyanation of Alcohols Enabled by an Iodide-Mediated Phosphine P(V/III) Redox Couple47
Synthesis of Sulfur-Substituted Bicyclo[1.1.1]pentanes by Iodo-Sulfenylation of [1.1.1]Propellane47
Palladium-Catalyzed Synthesis of Esters from Arenes through C–H Thianthrenation47
Enantioselective Cobalt-Catalyzed Remote Hydroboration of Alkenylboronates46
On-DNA Synthesis of Privileged Dihydropteridinones via Diboron-Mediated Cyclizations46
Visible-Light-Induced NHC-Catalyzed Carboacylation Reaction of Alkenes from Aryl Thianthrenium Salts and Aldehydes46
Cobalt-Catalyzed Asymmetric 1,4-Reduction of α,β-Unsaturated Nitriles with HBpin45
Formal Syntheses of (−)-Quinocarcinamide and (−)-Quinocarcin45
Synthesis of 1-Substituted Bicyclo[2.1.1]hexan-2-ones via a Sequential SmI2-Mediated Pinacol Coupling and Acid-Catalyzed Pinacol Rearrangement Reaction45
Chiral Squaramide Catalyzed Asymmetric Spiroketalization toward Aromatic [6,5] Spiroketals45
1,3-Butadiene Dicarbofunctionalization Enabled by the Dual Role of Diaryl Ketone in Photo-HAT/Chromium Catalysis45
DalPhos/Nickel-Catalyzed C2–H Arylation of 1,3-Azoles Using a Dual-Base System45
Spirochrains A–D, Four Caged [5,6,5] Spirocyclic Amides from an Antarctic Fungus Aspergillus ochraceopetaliformis SCSIO 05702 with Anti-RSV Activities45
My Discovery of Science45
Tosylazide as N1-Synthon: Iron-Catalyzed Nitrogenative Dimerization of Indoles to p-Bisindolopyrazine Derivatives45
Hydrazone Activation in the Aminocatalytic Cascade Reaction for the Synthesis of Tetrahydroindolizines45
Mild Installation of Piperidines on 4-Alkylpyridines45
Manipulating Crystal Packing and Self-Assembly by π-Extended and Isomeric Fused Strategies in Thiophene Ring-Terminated Polycyclic Aromatic Hydrocarbons45
Rh-Catalyzed Carbonylative Cyclization of Propargylic Alcohols with Aryl Boronic Acids45
Aromatic Amine and Chiral Phosphoric Acid Synergistic Catalyzed Cascade Reaction of Alkynylnaphthols with Aldehydes45
Regiochemical Switching in Ir-Catalyzed C–H Borylation by Altering Ligand Loadings of N,B-Type Diboron Species44
From Nitrogen to Sulfur: Investigating the Effect of Core Modification within Azaacene-Fused 21,23-Dithiaporphyrins44
Photocatalytic Strecker-Type Reaction for the Synthesis of Primary α-Aminonitriles44
Organic Chemistry in Argentina and the Genesis of SAIQO44
Sequential Strategies to Trigger Mild Dearomative Diels–Alder Cyclizations44
Cope-Type Hydroamination of Vinylboronates44
Synthesis of α-Aryl Secondary Amides via Nickel-Catalyzed Reductive Coupling of Redox-Active Esters44
Charge-Enhanced Reactivity of Esters by a Cationic Substituent44
Correction to “Access to 6-Deoxy-heptose Constructs by One Carbon Homologation of Hexoses with Malononitrile: Divergent Synthesis of Campylobacter jejuni Strain 81-176 Capsular Trisaccharide Re44
Asymmetric Synthesis of CF3-Substituted β-Hydroxyketones and 1,3-Diols by Engineered Ketoreductases44
Staudinger Cleavages of Amides on Naphthalene for the Ipsilateral Effect of 1,8-Substituents44
Gold-Catalyzed Regioselective Synthesis of Crowded Cyclopentadienes by Migratory Cycloisomerization of Vinylallenes44
Asymmetric Organocatalysis Enables Rapid Assembly of Portimine Precursor Chains44
Conformational Effects in Intramolecular C(sp3)–H Bond Functionalization: Gold(I)-Catalyzed Cycloisomerization of Aliphatic 1-Bromoalkynes as Benchmark Reaction43
Palladium-Catalyzed Chemo- and Regiocontrolled Tandem Cyclization/Cross-Coupling of 2-Benzyl-3-alkynyl Chromones with Aryl Iodides for the Synthesis of 4H-Furo[3,2-c]chromenes and Xantho43
Formation and Rearrangement of a Congested Spiropentane from the Trapping of Dibenzonorcarynyliden(e/oid) by Phencyclone43
Enantioselective [3 + 3] Annulation–Deoxalation Strategy for Rapid Access to δ-Oxoesters via N-Heterocyclic Carbene Catalysis43
Sc-Catalyzed Asymmetric [2 + 2] Annulation of 2-Alkynylnaphthols with Dienes to Access Cyclobutene Frameworks43
Chromium-Catalyzed Diastereoselective Synthesis of Conformationally Constrained Spirotetrahydroquinolines43
P(O)Me2–Alkenes: From Synthesis to Applications43
Synthesis of 3-Benzazepines via Cobalt-Catalyzed C–H Bond Functionalization with CaC2 as the Acetylene Source43
Domino Synthesis of Thioindirubin via Aldol Condensation/C–S Cross-Coupling/Cyclization Reaction Using Xanthate as a Sulfur Surrogate43
Application of Ni/Zr-Mediated Ketone Coupling for the Scalable Synthesis of Homohalichondrin B43
Deciphering the δ-Lactam Formation and lron-Reducing Activity of Spinactins from Saccharopolyspora spinosa42
Collective Syntheses of Corynanthe Alkaloids Based on a Chirality-Tunable Structure Unit42
Rhodium-Catalyzed Selective C( sp 2 )–H Activation/Annulation of tert -Buty42
Polysubstituted Indole Synthesis via Palladium/Norbornene Cooperative Catalysis of Oxime Esters42
Photoredox Fe-Catalyzed Truce–Smiles Rearrangement of N -Arylsulfonyl Acrylamides with Aliphatic Carboxylic Acids42
Preparation of 3,5-Methanobenzo[ b ]azepines: An sp 3 -Rich Quinolone Isostere42
Environmentally Friendly Synthesis of Highly Substituted Phenols Using Enallenoates and Grignard Reagents42
Diarylamine Synthesis via Desulfinylative Smiles Rearrangement42
Triflylpyridinium as Coupling Reagent for Rapid Amide and Ester Synthesis42
Highly Contorted Rigid Nitrogen-Rich Nanographene with Four Heptagons42
Radical Alkynylthiolation with Visible-Light-Sensitive S-Alkynylthio Sulfonates41
Isolation and Total Synthesis of Beru’amide, an Antitrypanosomal Polyketide from a Marine Cyanobacterium Okeania sp.41
Biocatalytically Generated Library of Chiral Building Blocks Containing a Quaternary Stereocenter41
Aryl Carboxylic Acids as Structure-Tunable HAT Agents for Photochemical Site-Selective C(sp 3 )–H gem 41
Amidophosphine Boranes as Hydroboration Reagents for Nitriles, Alkynes, and Carboxylic Acids41
Construction of Oxo-Bridged Diazocines via Rhodium-Catalyzed (4+3) Cycloaddition of Carbonyl Ylides with Azoalkenes41
Pd-Catalyzed Asymmetric Intramolecular Dearomatizing Reductive Heck Reaction of Indoles41
Nickel-Catalyzed Photoredox Allenylation of Alkyl Halides41
Protecting-Group Free Total Synthesis of β-Levantenolide through Late Stage Bromo-Spirocyclization41
A Sterically Tuned 2-Fluoropyridinium Salt for the Catalyst-Free, Visible-Light-Mediated Deoxygenation of Alcohols via an Electron Donor–Acceptor Complex41
Asymmetric Intramolecular Hydroamination to Construct Diverse N–N/C–N Indole Atropisomers via Cooperative Pd(0) and Chiral Phosphoric Acid Catalysis40
Synthesis of γ-Butyrolactones with Chiral Quaternary–Tertiary Stereocenters via Catalytic Asymmetric Mukaiyama–Michael Addition40
Paired Electrocatalysis-Enabled Cross Coupling of Sulfinamides with Olefins toward the Synthesis of Vinyl Sulfoximines40
Electrochemical Allylic C(sp3)–H Isothiocyanation via [3,3]-Sigmatropic Rearrangement40
Photochemical Carbene-Transfer Reaction of Vinyldiazo Compounds: Synthesis of 1-Pyrrolines via Methylenation/[2+3] Annulation40
Free Amine-Directed Redox Neutral Ruthenium(II) Catalysis toward Regioselective Synthesis of Heterobiaryls40
Fluorous Phase-Enhanced Fluorescent Sensitivity for Enantioselective Recognition of Lysine40
Gold-Catalyzed C–O Cross-Coupling Reactions of Aryl Iodides with Silver Carboxylates40
Biocatalytic Synthesis of Metaxalone and Its Analogues40
Aldehydes as O-Nucleophiles in Cobalt Hydride Hydrogen Atom Transfer Catalysis: Overriding the Innate Somophilicity39
Annulative π-Extension by Cp*Co(III)-Catalyzed Ketone-Directed peri-Annulation: An Approach to Access Fused Arenes39
Access to SCF3-Substituted Indolizines via a Photocatalytic Late-Stage Functionalization Protocol39
Diphenylsilylsilanolates Enable the Transfer of a Wide Range of Silyl Groups39
Ligand- and Substrate-Controlled para C–H Borylation of Anilines at Room Temperature39
N-Heterocyclic Carbene Catalysis for Polycyclic Benzazepines Assembly: Regioselective Intramolecular Tandem Radical Cyclization39
Light-Induced Activation of C–X Bond via Carbonate-Assisted Anion−π Interactions: Applications to C–P and C–B Bond Formation39
Photocatalytic Synthesis of α-Ketonyl Glycosyl Compounds from Glycosyl Thiols and Silyl Enol Ethers39
Pd-Catalyzed Asymmetric Allylic Alkylation of Carboxylic Acids for the Synthesis of Chiral Butenolidyl Ester Prodrugs and Peptide–Drug Conjugates39
Shuttle Hydrogen Atom Transfer for Hydro-Fluorosulfonylation of Haloalkynes without β-Scission39
Dinickel-Catalyzed Asymmetric Allylic Alkylation of Cyclic Ketones with Allylic Amine Derivatives38
Palladium-Catalyzed “Cut-and-Sew” Reaction of C(sp3)–NC: Direct Synthesis of Bulky Nitriles Containing an All-Carbon Quaternary Center38
Biosynthesis of Dolastatin 10 in Marine Cyanobacteria, a Prototype for Multiple Approved Cancer Drugs38
Divergent Access to Polycyclic N-Heterocyclic Compounds through Büchner-Type Dearomatization Enabled Cycloisomerization of Diynamides under Gold Catalysis38
Synthesis and Structural Revision of the Cyclic Hexapeptide Dimers Antatollamides A and B38
Synergistic [4 + 1] Spiroannulation and Selective Ring-Opening Strategy toward γ-Spirolactams38
Kinetic Resolution of BINOLs and Biphenols by Atroposelective, Cu–H-Catalyzed Si–O Coupling with Hydrosilanes38
Minisci-Type Dehydrogenative Coupling of C(sp3)–H and N-Heteroaromatics Enabled by Photoelectrochemical Hydrogen Atom Transfer38
Asymmetric Total Synthesis of (+)-Spiroapplanatumine G38
Stereoselective Synthesis of Conjugated Dienes via Aryl-to-Vinyl 1,4-Nickel Migration and Reductive Cross-Coupling38
Copper-Catalyzed Asymmetric Propargylic [3 + 2] Cycloaddition: Synthesis of Enantioenriched Dihydrofuro[3,2-c]coumarins and its Quinolinone and Thiocoumarin Analogues38
Visible-Light-Induced Selective α-Fluoroarylation of Secondary N-Alkyl Anilines with Polyfluoroarenes via Direct C–H/C–F Coupling37
Electrochemical Desaturation and β-Thiocyanation of Cyclic Amides37
Photoinduced Difluoromethylation Cyclization to Generate Medium-Sized Difluoro-benzo[b]azepines37
Environmentally Responsible and Cost-Effective Synthesis of the Antimalarial Drug Pyronaridine37
C–C Bond Cleavage-Induced C- to N-Acyl Transfer for Synthesis of Amides37
Visible-Light-Driven C,N-Selective Heteroarylation of N-Fluoroalkyl Hydroxylamine Reagents with Quinoxalin-2(1H)-ones37
Transformation-Guided Genome Mining Provides Access to Brominated Lanthipeptides37
Total Synthesis of the Phenolic Steroid Myrmenaphthol A37
Enantioselective Palladium-Catalyzed Domino Carbonylative Heck Esterification of o-Iodoalkenylbenzenes with Arylboronic Acids37
Iridium-Catalyzed Double Asymmetric Hydrogenation of 2,5-Dialkylienecyclopentanones for the Synthesis of Chiral Cyclopentanones37
Nonactivated Aziridine Synthesis by Intermolecular Polarity-Mismatched Carboamination of Unactivated Alkenes with Unactivated Alkyl Halides37
Intramolecular Appel Reaction of Trifluoromethylated β-Keto Diazos Enabling Assembly of Trifluoromethylpyrazoles37
Nickel-Catalyzed Domino Reaction of α-Aryloxyacetonitriles with Arylboronic Acids: Synthesis of 2-Aroylbenzo[b]furans36
Tertiary Amine-Mediated Reductions of Phosphine Oxides to Phosphines36
Ring-Enlargement of in Situ Generated Cyclopropanones by the Reaction with Sulfonium Ylides: One-Pot Synthesis of Cyclobutanones36
Nickel-Catalyzed Regioselective Markovnikov Hydrosilylation of Vinylarenes via Hydrogen Atom Transfer36
Photoredox Catalytic Approach for Difluoroallylation of Electron-Deficient sp3 C–H Bonds36
A Synthetic Strategy for the Preparation of Fused [5,6,5,5]-Tetracyclic Energetic Compounds36
Computationally Assisted Analysis of NMR Chemical Shifts as a Tool in Conformational Analysis36
Strain-Release Glycosylation of Thio- and Selenoglycosides Enabled by Activation of Donor–Acceptor Oxiranes with Catalytic TfOH36
Reductive Hydrodehalogenation of Halogenated Carboxylic Acid Derivatives Using a DMSO/HCOONa·2H2O System36
Multiselective Diels–Alder Reaction of α-Arylacroleins Catalyzed by Boron Tribromide-Assisted Chiral Phosphoric Acids36
Photocatalytic Borylation of Imines and Alkenes via Decarboxylation of Trimethylamine Carboxyborane: A New Approach for Generating Boryl Radicals36
Visible-Light-Induced Cascade Cyclization of 3-(2-(Ethynyl)phenyl)quinazolinones to Phosphorylated Quinolino[2,1-b]quinazolinones36
A Catalytic Enantioselective Suzuki Coupling for the Modular Construction of Axially Chiral BODIPYs with Bright Solid-State Emission36
Macrocyclization of Unprotected Peptides via Cycloaddition between o-Diones and Furan-2(3H)-one36
Visible-Light Catalyzed Desulfurative Cyclization for Synthesis of 3-Amino-[1,2,4]-triazolo Pyridine36
Ir-Catalyzed Asymmetric Cascade Allylation/Spiroketalization Reaction for Stereoselective Synthesis of Oxazoline-Spiroketals36
Photocatalytic Umpolung Strategy for the Synthesis of α-Amino Phosphine Oxides and Deuterated Derivatives36
Stereodivergent 3,4-Hydroalkoxylation of 1,3-Dienes Via Dual Photo and Copper Catalysis36
Synthesis of ortho-Phosphated (Hetero)Arylamines through Cascade Atherton–Todd Reaction/[3,3]-Rearrangement from Arylhydroxylamines and Dialkyl Phosphites36
Photochemical Construction of Trifluoromethyl Bicyclo[1.1.1]pentyl-heterocycles36
Cobalt-Catalyzed Enantioselective Reductive Amination of Ketones with Hydrazides36
Photochemical Reduction of Quinolines with γ-Terpinene36
Chiral Brønsted Acid Catalyzed Enantioselective Synthesis of Spiro-Isoindolinone-Indolines via Formal [3 + 2] Cycloaddition36
Synthesis of ortho-Methylated Benzamides via Palladium-Catalyzed Denitrogenative Cross-Coupling Reaction of [1,2,3]-Benzotriazin-4(3H)-ones with DABAL-Me336
Rhodium(III)-Catalyzed Synthesis of Diverse Fluorescent Polycyclic Purinium Salts from 6-Arylpurine Nucleosides and Alkynes36
Biomimetic Total Synthesis of Clavicipitic Acid: A DDQ-Mediated Intramolecular Cross-Dehydrogenative Coupling Approach36
Relay Annulation of Ammonium Ylides with Oxindole-Derived α,β-Unsaturated Ketimines: Catalytic Construction of Spiro-polycyclic Oxindoles35
Direct Synthesis of α-Methylated Arylacetamides from Arylacetonitriles via Ir-Catalyzed Cascade α-Methylation and Selective Hydration35
Ru(II)-Catalyzed Divergent C–H Annulations of Propargyl Cyclic Carbonates35
Conia-Ene Cyclization of Pyrazolones with o -Alkynyl Aldehydes: A Strategic Shift from Classical Condensation to Spiroannulation35
Photocatalytic Bicyclization of Indole-Tethered 1,6-Enynes for Diastereoselective Synthesis of Pyrrolo[3,2,1-jk]carbazoles35
Nickel-Catalyzed Cross-Electrophile Ring Opening/gem-Difluoroallylation of Aziridines35
Solvent-Driven Room-Temperature Curtius Rearrangements to Access Nucleotides Bearing Substituted Fused Pyridones35
Sequential One-Pot Transformation to R–CF2-Embedded 1,5-Diketones Enabled by Nickel: Access to 4-Perfluoroalkylpyridines35
Supramolecular Polymerization of Biphenyl-Cyanostilbenes. Triggering Circularly Polarized Luminescence by Self-Assembly35
Biocatalytic Enantioselective Oxidation of N -Acyl- S -Methyl Sulfenamides for the Asymmetric Synthesis of35
Cobalt/Rhodium-Catalyzed Diversified Amidation of Benzocyclobutenols via C–C Cleavage under Catalyst and Condition Control35
Dual 1,2-Migration-Enabled β-Boryl Amide Synthesis35
A Donor–Acceptor 10-Cycloparaphenylene and Its Use as an Emitter in an Organic Light-Emitting Diode34
Dichloromethyl(diaryl) Sulfonium Salts as gem-Dichlorocyclopropanation Reagents34
AJICAP-M: Traceless Affinity Peptide Mediated Conjugation Technology for Site-Selective Antibody–Drug Conjugate Synthesis34
Expanded Access to Fluoroformamidines via a Modular Synthetic Pathway34
Stereoretentive Decarboxylative Amidation of α,β-Unsaturated Carboxylic Acids to Access Enamides34
Visible-Light-Induced Photocatalytic Deoxygenative Benzylation of Quinoxalin-2-(1H)-ones with Carboxylic Acid Anhydrides34
Manganese-Catalyzed Regioselective C–H Lactonization and Hydroxylation of Fatty Acids with H2O234
Two Bioactive Compounds, Uniformides A and B, Isolated from a Culture of Nocardia uniformis IFM0856T in the Presence of Animal Cells34
Discovery, Characterization, and Anti-XOD Activity of Calcium Metallophore from Coix lacryma-jobi34
Asymmetric Synthesis of Axially Chiral Arylpyrazole via an Organocatalytic Arylation Reaction34
[60]Fullerene-Fused Cyclopentanes: Mechanosynthesis and Photovoltaic Application34
Photoredox 1,4-Hydroxysulfonylation of Methylenecyclobutane via Carbon-Radical-Mediated β-Scission of Cyclobutane34
Total Synthesis of (+)-Leucolusine and (−)-7-epi-Leucolusine34
Visible-Light-Induced Three-Component Selenofunctionalization of Alkenes: An Aerobic Selenol Oxidation Approach34
Total Synthesis of Daphenylline via Diels–Alder Cycloaddition and Rhodium-Catalyzed C–H Alkynylation34
Retraction of Activating Imides with Triflic Acid: A General Intramolecular Aldol Condensation Strategy Toward Indolizidine, Quinolizidine, and Valmerin Alkaloids33
Rhodium-Catalyzed Trifluoromethoxylation of Allenylic Trichloroacetimidates33
Correction to “Regioselective Synthesis of Highly Functionalized Pyrazoles from N-Tosylhydrazones”33
Asymmetric Synthesis of Hydrodibenzofurans from Norcaradienes: Kinetic Resolution via [3 + 2] Cycloaddition with Quinones33
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Photoactivation of Electron Donor–Acceptor Complexes for C(sp2)–H Amination of Arenes Using an Organocatalytic Acceptor33
Chemoselective Benzylic C–H Deuteration Using Deuterium Gas33
Synthesis and Characterization of Atropdiastereomeric Macrocyclic Metacyclophanes33
Dearomatization/Deiodination of o-Iodophenolic Compounds with α,β-Unsaturated Imines for Accessing Benzofuran Derivatives33
Studies towards the Enantioselective Synthesis of Cryptowolinol via Pd0-Catalyzed C(sp3)–H Arylation/Parallel Kinetic Resolution33
Rhodium-Catalyzed Synthesis of Peptide Polysulfides by Insertion of Sulfur into Unprotected Peptide Disulfides33
[Au]/[Ag]-Catalyzed Glycosidation of Ethynylcyclohexyl Glycosyl Carbonates Enables Direct Stereoselective Synthesis of 2-Azido-2-deoxy-β-mannopyranosides33
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Functional Crosstalk between Discrete Indole Terpenoid Gene Clusters in Tolypocladium album33
Asymmetric Synthesis of Bicyclic Isoxazolines via Dearomative Cycloaddition of 4-Nitroisoxazoles with Zwitterionic π-Allyl Palladium Species33
Co-Catalyzed Suzuki–Miyaura Coupling of Organoboronic Acids and Alkynyl Chlorides Using Potassium Bicarbonate as Base33
Regio- and Stereoselective anti-Hydroalumination of Internal and Terminal Alkynes Using a Mixed Reagent of Cesium Fluoride with Diisobutylaluminum Hydride33
Ruthenium(II)-Catalyzed Construction of 2,3-Disubstituted Benzo[b]thiophene-1,1-dioxides and Naphtho[1,2-b]thiophene-1,1-dioxides33
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DABCO-Catalyzed Reaction of 2-Naphthols with Aryl Isothiocyanates: Access to 2-Iminonaphtho-1,3-oxathioles32
(Methyl)thianthrenium Salt Enabled Monoselective N-Methylation and N-(13C-Methyl) Labeling: Late-Stage Functionalization of Arylamides32
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