OOIR: Observatory of International Research

Papers

(The TQCC of Bioconjugate Chemistry is 8. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-01-01 to 2025-01-01.)

Article	Citations
Issue Publication Information	203
Correction to Development of an Effective Functional Lipid Anchor for Membranes (FLAME) for the Bioorthogonal Modification of the Lipid Bilayer of Mesenchymal Stromal Cells	137
Tyrosinase-Related Protein2 Peptide with Replacement of N-Terminus Residue by Cysteine Binds to H-2K^b and Induces Antigen-Specific Cytotoxic T Lymphocytes after Conjugation with CpG-DNA	82
Copper-Free Click Enabled Triazabutadiene for Bioorthogonal Protein Functionalization	69
Multiple Applications of a Novel Biarsenical Imaging Probe in Fluorescence and PET Imaging of Melanoma	65
Issue Editorial Masthead	62
Issue Editorial Masthead	51
Issue Editorial Masthead	48
Preparation of Maleimide-Modified Oligonucleotides from the Corresponding Amines Using N-Methoxycarbonylmaleimide	47
Hydrolytically Stable Maleimide-End-Functionalized Polymers for Site-Specific Protein Conjugation	46
Camouflaged Fluorescent Silica Nanoparticles Target Aggregates and Condensates of the Amyloidogenic Protein Tau	41
DNA Origami–Platelet Adducts: Nanoconstruct Binding without Platelet Activation	41
Site-Specific Chemical Modification of a Cytokine Mimic for Small Molecule-Based Tumor Targeting	39
Therapeutic Targeting of Tumor Cells Rich in LGR Stem Cell Receptors	38
Design and Optimization of an α-Helical Bundle Dimer Cell-Penetrating Peptide for In Vivo Drug Delivery	37
Structure-Dependent Nontraditional Intrinsic Fluorescence of Aliphatic Hyperbranched Polyureas	34
Copper-Containing Artificial Polyenzymes as a Clickase for Bioorthogonal Chemistry	34
Natural and Synthetic Sortase A Substrates Are Processed by Staphylococcus aureus via Different Pathways	33
Issue Publication Information	33
Issue Editorial Masthead	32
Issue Editorial Masthead	32
Issue Editorial Masthead	31
Correction to “Oral Delivery of Peptide Drugs Using Nanoparticles Self-Assembled by Poly(γ-glutamic acid) and a Chitosan Derivative Functionalized by Trimethylation”	31
Issue Editorial Masthead	31
Issue Publication Information	31

Transthyretin-Penetratin: A Potent Fusion Protein Inhibitor against Alzheimer’s Amyloid-β Fibrillogenesis with High Blood Brain Barrier Crossing Capability	29
Near-Infrared Photoresponsive Nanotransducers for Precise Regulation of Gene Expression	29
Site-Specific ⁶⁸Ga Radiolabeling of Trastuzumab Fab via Methionine for ImmunoPET Imaging	29
Modular PET Agent Construction Strategy through Strain-Promoted Double-Click Reagent with Efficient Photoclick Step	28
Duo-Chol: A Photoconvertible Live Cell Imaging Tool for Tracking Cholesterol	27
Formal [4 + 2] Cycloadditions of Maleimides on Duplex DNA	27
Live-Cell Mitochondrial Targeted NIR Fluorescent Covalent Labeling of Specific Proteins Using a Dual Localization Effect	27
Facile Synthesis of a Redox-Responsive Hyperbranched Polymer Prodrug as a Unimolecular Micelle for the Tumor-Selective Drug Delivery	25
A Functionalizable Analog of the Yariv Reagent for AGP Imaging using Fluorescence Microscopy	25
Characterization of an N-Allylglyoxylamide-Based Bioorthogonal Nitrone Trap	24
Issue Editorial Masthead	24
DOTAM-Based, Targeted, Activatable Fluorescent Probes for the Highly Sensitive and Selective Detection of Cancer Cells	24
Tandem-Cleavage Linkers Improve the In Vivo Stability and Tolerability of Antibody–Drug Conjugates	24
Efficient Chemical Synthesis of Multi-Monoubiquitylated and Diubiquitylated Histones by the α-Halogen Ketone-Mediated Strategy	24
Bioresorbable Depot for Sustained Release of Immunostimulatory Resiquimod in Suppressing Both Primary Triple-Negative Breast Tumors and Metastatic Occurrence	24
Correction to “Direct Loading and Tunable Release of Antibiotics from Polyelectrolyte Multilayers To Reduce Bacterial Adhesion and Biofilm Formation”	23
Correction to “Multifunctional Nanoflowers for Simultaneous Multimodal Imaging and High-Sensitivity Chemo-Photothermal Treatment”	23
Issue Publication Information	23
Solid-Phase Synthesis of Caged Luminescent Peptides via Side Chain Anchoring	23
A β-Cyclodextrin-Albumin Conjugate for Enhancing Therapeutic Efficacy of Cytotoxic Drugs	23
Exo-Enzymatic Addition of Diazirine-Modified Sialic Acid to Cell Surfaces Enables Photocrosslinking of Glycoproteins	23
Development of Radiopharmaceuticals for NPY Receptor-5 (Y5) Nuclear Imaging in Tumors by Synthesis of Specific Agonists and Investigation of Their Binding Mode	22
Issue Publication Information	22
Synthesis of Isolated DNA Aptamer and Its Application of AC-Electrothermal Flow-Based Rapid Biosensor for the Detection of Dengue Virus in a Spiked Sample	21
Monitoring Human Neutrophil Activation by a Proteinase 3 Near-Infrared Fluorescence Substrate-Based Probe	21
A Series of Furimazine Derivatives for Sustained Live-Cell Bioluminescence Imaging and Application to the Monitoring of Myogenesis at the Single-Cell Level	21
Design, Mechanical Properties, and Dynamics of Synthetic DNA Filaments	21
Synthesis and Evaluation of Three Azide-Modified Disaccharide Oxazolines as Enzyme Substrates for Single-Step Fc Glycan-Mediated Antibody-Drug Conjugation	20
Tumor-Derived PD-L1⁺ Exosomes with Natural Inflammation Tropism for Psoriasis-Targeted Treatment	20
Optimization of Enzymolysis Clearance Strategy To Enhance Renal Clearance of Radioligands	20
Issue Publication Information	20
Albumin Biomolecular Drug Designs Stabilized through Improved Thiol Conjugation and a Modular Locked Nucleic Acid Functionalized Assembly	20
Issue Publication Information	19
Gene Regulation Using Nanodiscs Modified with HIF-1-α Antisense Oligonucleotides	19
Conjugation of Hemoglobin and Mannan Markedly Improves the Immunogenicity of Domain III of the Zika Virus E Protein: Structural and Immunological Study	19
Editorial for January	19
Issue Editorial Masthead	19
Xylose Dehydrogenase Immobilized on Ferromagnetic Nanoparticles for Bioconversion of Xylose to Xylonic Acid	19
Sculpting a Uniquely Reactive Cysteine Residue for Site-Specific Antibody Conjugation	19
Issue Publication Information	19
Bioorthogonal PEGylation Prolongs the Elimination Half-Life of N-TIMP2 While Retaining MMP Inhibition	19
Palladium-Mediated S-Arylation of Cysteine Residues with 4-[¹⁸F]Fluoroiodobenzene ([¹⁸F]FIB)	18
A Cysteine-Maleimide-Based Design for Hemostatic, Antibacterial, and Biodegradable Wound Dressing	18
Targeted Anti-Cancer Provascular Therapy Using Ultrasound, Microbubbles, and Nitrite to Increase Radiotherapy Efficacy	18
Issue Publication Information	18
Rational Approach to Improve Detergent Efficacy for Membrane Protein Stabilization	18
Click Chemistry Enables Rapid Amplification of Full-Length Reverse Transcripts for Long-Read Third Generation Sequencing	18
Cyanine Masking: A Strategy to Test Functional Group Effects on Antibody Conjugate Targeting	18
Synthetic Pept-Ins as a Generic Amyloid-Like Aggregation-Based Platform for In Vivo PET Imaging of Intracellular Targets	18
Site-Specific Modification of Single Domain Antibodies by Enzyme-Immobilized Magnetic Beads	17

Azobenzene-Based Amino Acids for the Photocontrol of Coiled-Coil Peptides	17
Spherical Nucleic Acid Mediated Functionalization of Polydopamine-Coated Nanoparticles for Selective DNA Extraction and Detection	17
Non-Genetic Generation of Antibody Conjugates Based on Chemoenzymatic Tyrosine Click Chemistry	17
PEGylation of anti-MerTK Antibody Modulates Ocular Biodistribution	17
Advances in Optical Sensors of N-Acetyl-β-d-hexosaminidase (N-Acetyl-β-d-glucosaminidase)	17
Peptide Amphiphile Hydrogels Based on Homoternary Cucurbit[8]uril Host-Guest Complexes	17
Impact of Drug Conjugation on Thermal and Metabolic Stabilities of Aglycosylated and N-Glycosylated Antibodies	17
Designing Functional Bionanoconstructs for Effective In Vivo Targeting	17
Rapid Production of Bispecific Antibodies from Off-the-Shelf IgGs with High Yield and Purity	17
Hollow Cobalt Sulfide Nanospheres with Highly Enzyme-like Antibacterial Activities to Accelerate Infected Wound Healing	17
Synthesis and Characterization of a Positron Emission Tomography Imaging Probe Selectively Targeting the Second Bromodomain of Bromodomain Protein BRD4	17
One-Pot Conversion of Free Sialoglycans to Functionalized Glycan Oxazolines and Efficient Synthesis of Homogeneous Antibody–Drug Conjugates through Site-Specific Chemoenzymatic Glycan Remodeling	17
Incorporation of Intracellular NanoSIMS Tracers to Oligonucleotide Conjugates via Strain Promoted Sydnone–Alkyne Cycloaddition	16
Gallic Acid-Encapsulated PAMAM Dendrimers as an Antioxidant Delivery System for Controlled Release and Reduced Cytotoxicity against ARPE-19 Cells	16
Strategies to Control or Mimic Growth Factor Activity for Bone, Cartilage, and Osteochondral Tissue Engineering	16
Cysteine-Based Coupling: Challenges and Solutions	16
Bioconjugate Biomaterials: Leveraging Biology for the Next Generation of Active Materials	16
Pathologic Tissue Injury and Inflammation in Mice Immunized with Plasmid DNA-Encapsulated DOTAP-Based Lipid Nanoparticles	16
Polysaccharide-Based Coacervate Microgel Bearing Cationic Peptides That Achieve Dynamic Cell-Membrane Structure Alteration and Facile Cytosolic Infusion of IgGs	16
CD22L Conjugation to Insulin Attenuates Insulin-Specific B Cell Activation	16
Modular Click Assembly DNA-Encoded Glycoconjugate Libraries with on-DNA Functional Group Transformations	16
“On-Demand” Antimicrobial Photodynamic Activity through Supramolecular Photosensitizers Built with Rose Bengal and (p-Vinylbenzyl)triethylammomium Polycation Derivatives	16
Hypoxia-Activated Prodrug Enabling Synchronous Chemotherapy and HIF-1α Downregulation for Tumor Treatment	16
S9.6 Antibody–Enzyme Conjugates for the Detection of DNA–RNA Hybrids	16
Development of a Micellar-Promoted Heck Reaction for the Synthesis of DNA-Encoded Libraries	15
Environment-Sensitive Nucleoside Probe Unravels the Complex Structural Dynamics of i-Motif DNAs	15
Issue Publication Information	14
Biomedical Application of Porphyrin-Based Amphiphiles and Their Self-Assembled Nanomaterials	14
Chemoselective Reagents for the Traceless Bioreversible Modification of Native Proteins	14
Issue Editorial Masthead	14
Cyclopentadiene as a Multifunctional Reagent for Normal- and Inverse-Electron Demand Diels–Alder Bioconjugation	14
New Phenol Esters for Efficient pH-Controlled Amine Acylation of Peptides, Proteins, and Sepharose Beads in Aqueous Media	14
Therapeutic Potential of MF-TTZ-MMAE, a Site-Specifically Conjugated Antibody-Drug Conjugate, for the Treatment of HER2-Overexpressing Breast Cancer	14
Cyclohexanediamine Triazole (CHDT) Functionalization Enables Labeling of Target Molecules with Al¹⁸F/⁶⁸Ga/¹¹¹In	14
Engineering and Validation of a Peptide-Stabilized Poly(lactic-co-glycolic) Acid Nanoparticle for Targeted Delivery of a Vascular Disruptive Agent in Cancer Therapy	14
Chemical Synthesis of Interleukin-6 for Mirror-Image Screening	14
Issue Publication Information	14
Issue Editorial Masthead	14
Penetrating the Blood-Brain Barrier with New Peptide–Porphyrin Conjugates Having anti-HIV Activity	14
Evaluation of Cellular Targeting by Fab′ vs Full-Length Antibodies in Antibody–Nanoparticle Conjugates (ANCs) Using CD4 T-cells	14
Ultrastable PEGylated Calixarene-Coated Gold Nanoparticles with a Tunable Bioconjugation Density for Biosensing Applications	14
Guest-Induced Planar-Chiral Pillar[5]arene Surface for Selectively Adsorbing Protein Based on Host–Guest Chemistry	14
Design and Synthesis of Piperazine-Based Compounds Conjugated to Humanized Ferritin as Delivery System of siRNA in Cancer Cells	14
Highly Photoluminescent Nitrogen- and Zinc-Doped Carbon Dots for Efficient Delivery of CRISPR/Cas9 and mRNA	13
Equimolar Cross-Coupling Using Reactive Coiled Coils for Covalent Protein Assemblies	13
Antibody-Mediated Screening of Peptide Inhibitors for Monoamine Oxidase-B (MAO-B) from an Autodisplayed F_V Library	13
Positron Emission Tomography Tracer Design of Targeted Synthetic Peptides via ¹⁸F-Sydnone Alkyne Cycloaddition	13
Ligand-Modulated Catalytic Selectivity of Ag Clusterzyme for Relieving Multiorgan Injury via Inhabiting Acute Oxidative Stress	13
Identification of a Novel Transasparaginase Activity of Bacillus subtilis (bTG) for Sequence-Specific Bioconjugation	13
Efficiency and Safety of Dextran-PAMAM/siMMP-9 Complexes for Decreasing Matrix Metalloproteinase-9 Expression and Promoting Wound Healing in Diabetic Rats	13
Easy Surface Functionalization and Bioconjugation of Peptides as Capture Agents of a Microfluidic Biosensing Platform for Multiplex Assay in Serum	13
Sonotheranostics and Sonogenetics Special Issue	13
Supramolecular Bioconjugation Strategy for Antibody-Targeted Delivery of siRNA	13
3D-Printing Biodegradable PU/PAAM/Gel Hydrogel Scaffold with High Flexibility and Self-Adaptibility to Irregular Defects for Nonload-Bearing Bone Regeneration	13
Recent Advances in Bioorthogonal Click Chemistry for Enhanced PET and SPECT Radiochemistry	12
Bioderived Lipoic Acid-Based Dynamic Covalent Nanonetworks of Poly(disulfide)s: Enhanced Encapsulation Stability and Cancer Cell-Selective Delivery of Drugs	12
Insight into the Covalently Oriented Immobilization of Antibodies on Gold Nanoparticle Probes to Improve Sensitivity in the Colorimetric Detection of Listeria monocytogenes	12
6-Iodopurine as a Versatile Building Block for RNA Purine Architecture Modifications	12
Discovery of Bivalent GalNAc-Conjugated Betulin as a Potent ASGPR-Directed Agent against Hepatocellular Carcinoma	12
Modular Adapters Utilizing Binders of Different Molecular Types Expand Cell-Targeting Options for Adenovirus Gene Delivery	12
Enolate–Azide [3 + 2]-Cycloaddition Reaction Suitable for DNA-Encoded Library Synthesis	12
Dimeric Metal-Salphen Complexes Which Target Multimeric G-Quadruplex DNA	12
Synthesis and Evaluation of Ubiquitin–Dioxetane Conjugate as a Chemiluminescent Probe for Monitoring Deubiquitinase Activity	12
Molecular Switch Engineering for Precise Genome Editing	12
Break to Build: Isothermal Assembly of Nucleic Acid Nanoparticles (NANPs) via Enzymatic Degradation	12
Clickable Albumin Nanoparticles for Pretargeted Drug Delivery toward PD-L1 Overexpressing Tumors in Combination Immunotherapy	12
Synthesis of First Coumarin Fluorescent Dye for Actin Visualization	12
RGD-Modified Titanium as an Improved Osteoinductive Biomaterial for Use in Dental and Orthopedic Implants	12
Tritium O-Methylation of N-Alkoxy Maleimide Derivatives as Labeling Reagents for Biomolecules	12
Stimuli-Responsive Regulation of Biocatalysis through Metallic Nanoparticle Interaction	12
Design, Heterologous Expression, and Application of an Immobilized Protein Kinase	11
Luciferase NLuc Site-Specific Conjugation to Generate Reporters for In Vitro Assays	11
Bioorthogonal Chemistry and Its Applications	11
Suppressing Pancreatic Cancer Survival and Immune Escape via Nanoparticle-Modulated STING/STAT3 Axis Regulation	11
A Dual-Mechanism Targeted Bioorthogonal Prodrug Therapy	11
3D Printed Multifunctional Ti₆Al₄V-Based Hybrid Scaffold for the Management of Osteosarcoma	11
Formation of Direction-Controllable Pseudorotaxane and Catenane Using Chemically Cyclized Oligodeoxynucleotides and Their Noncovalent RNA Labeling	11
Issue Publication Information	11
Large Protein Assemblies for High-Relaxivity Contrast Agents: The Case of Gadolinium-Labeled Asparaginase	11
Cholesterol-Modified Oligonucleotides as Internal Reaction Controls during DNA-Encoded Chemical Library Synthesis	11

Generation and Biological Evaluation of Fc Antigen Binding Fragment-Drug Conjugates as a Novel Antibody-Based Format for Targeted Drug Delivery	11
Linker Chemistry and Connectivity Fine-Tune the Immune Response and Kinetic Solubility of Conjugated NOD2/TLR7 Agonists	11
Development of a Versatile Cancer Vaccine Format Targeting Antigen-Presenting Cells Using Proximity-Based Sortase A-Mediated Ligation of T-Cell Epitopes	11
Drug Delivery Targeting Neuroinflammation to Treat Brain Diseases	11
Covalent and Oriented Immobilization of Antibodies through Systematic Modification of Photoactivatable RNA Hybrid Aptamers	11
Pretargeted PET Imaging with a TCO-Conjugated Anti-CD44v6 Chimeric mAb U36 and [⁸⁹Zr]Zr-DFO-PEG₅-Tz	11
Developing GLP-1 Conjugated Self-Assembling Nanofibers Using Copper-Catalyzed Alkyne–Azide Cycloaddition and Evaluation of Their Biological Activity	11
Dual-Function Antibody Conjugate-Enabled Photoimmunotherapy Complements Fluorescence and Photoacoustic Imaging of Head and Neck Cancer Spheroids	11
Development of [¹⁸F]AmBF₃ Tetrazine for Radiolabeling of Peptides: Preclinical Evaluation and PET Imaging of [¹⁸F]AmBF₃-PEG₇-Tyr³-Octr	11
Metal Polyphenol Nanoparticle-Based Chemo/Ferroptosis Synergistic Therapy for the Treatment of Oral Squamous Cell Carcinoma	11
Micropreparative Gel Electrophoresis for Purification of Nanoscale Bioconjugates	11
Human CD47-Derived Cyclic Peptides Enhance Engulfment of mAb-Targeted Melanoma by Primary Macrophages	11
Issue Editorial Masthead	11
Single Gold Nanostars Achieve Inherent Cascade Catalytic and Near-Infrared Photothermal Activities for Efficient Tumor Therapy	11
Supramolecular Assembly of Single-Tail ssDNA-Amphiphiles through π–π Interactions	11
Directly Quantifiable Biotinylation Using a Water-Soluble Isatoic Anhydride Platform	10
Issue Publication Information	10
New Triazacycloalkane Derivatives as Cytotoxic Agents for CLL Treatment: From Proof of Concept to the Targeting Biomolecule	10
Issue Editorial Masthead	10
2′-Modified Thymidines with Bioorthogonal Cyclopropene or Sydnone as Building Blocks for Copper-Free Postsynthetic Functionalization of Chemically Synthesized Oligonucleotides	10
A Peptide Nanocage Constructed by Self-Assembly of Oligoproline Conjugates	10
SARS-CoV-2 Peptide Bioconjugates Designed for Antibody Diagnostics	10
Fluorescent Investigation of Proteins Using DNA-Synthetic Ligand Conjugates	10
Issue Editorial Masthead	10
Amyloid β-Peptide Segment Conjugated Side-Chain Proline-Based Polymers as Potent Inhibitors in Lysozyme Amyloidosis	10
Discovery of Imaging and Therapeutic Integration Bifunctional Molecules Based on Bio-Orthogonal Reaction and Releasable Disulfide Bond	10
Issue Editorial Masthead	10
Correction to “Lactose-Modified Chitosan Gold(III)-PEGylated Complex-Bioconjugates: From Synthesis to Interaction with Targeted Galectin-1 Protein”	10
Issue Editorial Masthead	10
Focused Cluster: Synthetic Host–Guest Chemistry in Biology	10
Biotin–NeutrAvidin Mediated Immobilization of Polymer Micro- and Nanoparticles on T Lymphocytes	10
Delivery of Targeted Co(III)–DNA Inhibitors of Gli Proteins to Disrupt Hedgehog Signaling	10
Click Chemistry-Enabled Conjugation Strategy for Producing Dibenzodiazepinone-Type Fluorescent Probes To Target M₂Acetylcholine Receptors	10
Biofilm-Mediated Immobilization of a Multienzyme Complex for Accelerating Inositol Production from Starch	10
Structural Optimization of Decoy Oligonucleotide-Based PROTAC That Degrades the Estrogen Receptor	10
Issue Publication Information	10
Issue Publication Information	10
Issue Editorial Masthead	10
Real-Time Monitoring of CAR-T Cell Efficiency through a Biorthogonal Cycloaddition Labeling Strategy	10
An Overview of Recent Advances in Biomedical Applications of Click Chemistry	10
Bioconjugation of Au₂₅ Nanocluster to Monoclonal Antibody at Tryptophan	9
Photo-Controllable Phase Transition of Arylazopyrazole-Conjugated Oligonucleotides	9
Cationic Micelles Outperform Linear Polymers for Delivery of Antisense Oligonucleotides in Serum: An Exploration of Polymer Architecture, Cationic Moieties, and Cell Addition Order	9
Acoustically Detonated Microbubbles Coupled with Low Frequency Insonation: Multiparameter Evaluation of Low Energy Mechanical Ablation	9
Linker Architectures as Steric Auxiliaries for Altering Enzyme-Mediated Payload Release from Bioconjugates	9
γ-Functional Iminiumthiolactones for the Single and Double Modification of Peptides	9
Formulation and Preclinical Testing of Tc-99m-Labeled HYNIC-Glc-FAPT as a FAP-Targeting Tumor Radiotracer	9
Issue Editorial Masthead	9
Reconfigurable Nanopolygons Made of DNA Catenanes	9
DNA Compatible Oxidization and Amidation of Terminal Alkynes	9
In Situ Visualizing Nascent RNA by Exploring DNA-Templated Oxidative Amination of 4-Thiouridine	9
iFLinkC-X: A Scalable Framework to Assemble Bespoke Genetically Encoded Co-polymeric Linkers of Variable Lengths and Amino Acid Composition	9
Dual Blood–Brain Barrier–Glioma Targeting Peptide–Poly(levodopamine) Hybrid Nanoplatforms as Potential Near Infrared Phototheranostic Agents in Glioblastoma	9
Mirror-Image Human Serum Albumin Domain III as a Tool for Analyzing Site II-Dependent Molecular Recognition	9
Rapid Covalent Labeling of Membrane Proteins on Living Cells Using a Nanobody–Epitope Tag Pair	9
mCherry on Top: A Positive Read-Out Cellular Platform for Screening DMD Exon Skipping Xenopeptide–PMO Conjugates	9
Multivalent Display of Erythropoietin on Quantum Dots Enhances Aquaporin-4 Expression and Water Transport in Human Astrocytes In Vitro	9
Issue Editorial Masthead	9
Chemoselective Bioconjugation of Amyloidogenic Protein Antigens to PEGylated Microspheres Enables Detection of α-Synuclein Autoantibodies in Human Plasma	9
Rapid Electrophilic Cysteine Arylation with Pyridinium Salts	9
Evaluating the Effect of Dye–Dye Interactions of Xanthene-Based Fluorophores in the Fluorosequencing of Peptides	9
Issue Editorial Masthead	9
Enzymatic Spin-Labeling of Protein N- and C-Termini for Electron Paramagnetic Resonance Spectroscopy	9
Structure–Activity Relationship of Fluorinated Sialic Acid Inhibitors for Bacterial Sialylation	9
Luminescent Ruthenium(II) Complexes Used for the Detection of 8-Oxoguanine in the Human Telomeric Sequence	9
Scale up of Transmembrane NADH Oxidation in Synthetic Giant Vesicles	9
Evaluation of Efficient Non-reducing Enzymatic and Chemical Ligation Strategies for Complex Disulfide-Rich Peptides	9
Issue Publication Information	9
Passivating the Background of Living Microbes with a Zwitterionic Peptide for Therapies	9
Pentafulvene–Maleimide Cycloaddition for Bioorthogonal Ligation	9
Issue Editorial Masthead	9
Cucurbituril–Ferrocene: Host–Guest Based Pretargeted Positron Emission Tomography in a Xenograft Model	9
Development of a Modular NTA:His Tag Viral Vaccine for Co-delivery of Antigen and Adjuvant	9
Stearylated Macropinocytosis-Inducing Peptides Facilitating the Cellular Uptake of Small Extracellular Vesicles	8
Legumain-Triggered Macrocyclization of Radiofluorinated Tracer for Enhanced PET Imaging	8
Stable and Highly Efficient Antibody–Nanoparticles Conjugation	8
Issue Publication Information	8
Carbonic Anhydrase IX Targeting Mn(II)-Based Magnetic Resonance Molecular Imaging Probe for Hypoxia Tumors	8
Revival of Bioengineered Proteins as Carriers for Nucleic Acids	8
Synthesis and Structure Optimization of Star Copolymers as Tunable Macromolecular Carriers for Minimal Immunogen Vaccine Delivery	8
Fast and Selective Reaction of 2-Benzylacrylaldehyde with 1,2-Aminothiol for Stable N-Terminal Cysteine Modification and Peptide Cyclization	8
Site-Specific, Platform-Based Conjugation Strategy for the Synthesis of Dual-Labeled Immunoconjugates for Bimodal PET/NIRF Imaging of HER2-Positive Tumors	8
Artificial Nanocage Formed via Self-Assembly of β-Annulus Peptide for Delivering Biofunctional Proteins into Cell Interiors	8
A General Set of DNA-Compatible Reactions for Preparing DNA-Tagged Multisubstituted Pyrroles	8
Targeting Colon Cancer Cells with Enzyme-Triggered Casein-Gated Release of Cargo from Mesoporous Silica-Based Nanoparticles	8
Design and Biological Evaluation of the Long-Acting C5-Inhibited Ornithodoros moubata Complement Inhibitor (OmCI) Modified with Fatty Acid	8
Self-Immolative Carbamate Linkers for CD19-Budesonide Antibody–Drug Conjugates	8
Early Detection and Noninvasive Staging of Kidney Dysfunction by a PEGylated Conventional Fluorophore via GFR-Sensitive Renal Transport	8
Affinity-Based Kinase-Catalyzed Crosslinking to Study Kinase–Substrate Pairs	8
First Comparison Study of the In Vitro and In Vivo Properties of a Randomly and Site-Specifically Conjugated SPECT/NIRF Monomolecular Multimodal Imaging Probe (MOMIP) Based on an aza-BOD	8
Selective Reduction of Cysteine Mutant Antibodies for Site-Specific Antibody–Drug Conjugates	8
The Influence of a Polyethylene Glycol Linker on the Metabolism and Pharmacokinetics of a ⁸⁹Zr-Radiolabeled Antibody	8
Rose Bengal Labeled Bovine Serum Albumin for Protein Transport Imaging in Subcutaneous Tissues Using Computed Tomography and Fluorescence Microscopy	8
Light-Activated Nanodiamond-Based Drug Delivery Systems for Spatiotemporal Release of Antisense Oligonucleotides	8
Size-Dependent Glioblastoma Targeting by Polymeric Nanoruler with Prolonged Blood Circulation	8