OOIR: Observatory of International Research

Papers

(The H4-Index of Bioorganic & Medicinal Chemistry is 28. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2022-06-01 to 2026-06-01.)

Article	Citations
Current Japanese pharmaceutical chemistry	93
Targeting prolidase. A survey of the literature data to depict a structure-activity relationship frame and to address future studies for drug development	86
Synthesis and biological evaluation of pyrazole-fused oleanolic acid derivatives as novel inhibitors of inflammatory and osteoclast differentiation	70
Graphical abstract TOC	60
Contents continued	52
Production and synthesis of a novel 191Pt-labeled platinum complex and evaluation of its biodistribution in healthy mice	50
Crescent-shaped meta-substituted benzene derivatives as a new class of non-nucleoside ribonuclease A inhibitors	48
Editorial Board	45
Targeting m6A binding protein YTHDFs for cancer therapy	41
Selective targeting of human TET1 by cyclic peptide inhibitors: Insights from biochemical profiling	41
RNA-templated chemical synthesis of proapoptotic L- and d-peptides	40
Design, synthesis, biological activity and molecular docking studies of triazolopyridine derivatives as ASK1 inhibitors	38
Decades old glitazones still find niche in drug discoveries as PPAR-γ agonists: medicinal chemistry perspective, structure-activity relationships and therapeutic implications	37
Development of delivery carriers for plasmid DNA by conjugation of a helical template to oligoarginine	35
Design, synthesis and validation of a new Crimped Head-Piece for DNA-Encoded libraries generation	35
Graphical abstract TOC	33
Research progress of STAT3-based dual inhibitors for cancer therapy	33
Design, synthesis and evaluation the bioactivities of novel 1,3-dimethyl-6-amino-1H-indazole derivatives as anticancer agents	33
Discovery of 3-hydroxymethyl-azetidine derivatives as potent polymerase theta inhibitors	31
Natural product-derived antifungals against Candida albicans: Chemical diversity and mechanisms of action	31
Design, synthesis and antibacterial evaluation of oxazolidinone derivatives containing N-methylglycyl or quaternary ammonium salts	30
Synthesis and medicinal chemistry of tetronamides: Promising agrochemicals and antitumoral compounds	30
Sustainable electrochemical C(sp3) − H oxygenation using water as the oxygen source	30
Janus dendritic ionizable lipids with fine designed headgroup and tails to improve mRNA delivery efficiency	29
Synthesis and antiproliferative activity of (−)-cleistenolide, (6S)-cleistenolide and 4-substituted cleistenolide analogues	29

Exploring novel A2AAR antagonists: Design, synthesis, and evaluation of 2,6,9-trisubstituted purine derivatives as promising antifibrotic agents	28
A multifunctional hydrogel for synergistic dendritic cell activation and immunogenic cell death induction in enhanced chemoimmunotherapy	28
Innovative synthesis and purification method of fluorescent and bifunctional substrates for self-labelling protein tags	28