OOIR: Observatory of International Research

Papers

(The H4-Index of Bioorganic & Medicinal Chemistry is 27. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-11-01 to 2025-11-01.)

Article	Citations
Synthesis and antiproliferative activity of (−)-cleistenolide, (6S)-cleistenolide and 4-substituted cleistenolide analogues	127
Current Japanese pharmaceutical chemistry	115
Targeting prolidase. A survey of the literature data to depict a structure-activity relationship frame and to address future studies for drug development	87
Sulfadoxine derivatization through multicomponent reactions to obtain new antiplasmodial compounds	71
Innovative synthesis and purification method of fluorescent and bifunctional substrates for self-labelling protein tags	71
Diterpenoids from the whole plants of Croton yunnanensis and their bioactivities	44
Targeting m6A binding protein YTHDFs for cancer therapy	42
Site-specific construction of triptolide-based antibody-drug conjugates	42
Sustainable electrochemical C(sp3) − H oxygenation using water as the oxygen source	41
Development of delivery carriers for plasmid DNA by conjugation of a helical template to oligoarginine	40
Synthesis and medicinal chemistry of tetronamides: Promising agrochemicals and antitumoral compounds	39
Synthesis and biological evaluation of pyrazole-fused oleanolic acid derivatives as novel inhibitors of inflammatory and osteoclast differentiation	37
Graphical abstract TOC	37
Graphical abstract TOC	36
RNA-templated chemical synthesis of proapoptotic L- and d-peptides	35
Contents continued	34
Design, synthesis and validation of a new Crimped Head-Piece for DNA-Encoded libraries generation	34
Production and synthesis of a novel 191Pt-labeled platinum complex and evaluation of its biodistribution in healthy mice	33
Research progress of STAT3-based dual inhibitors for cancer therapy	32
Discovery of novel 2,8-diazaspiro[4.5]decan-1-one derivatives as potent RIPK1 kinase inhibitors	32
Crescent-shaped meta-substituted benzene derivatives as a new class of non-nucleoside ribonuclease A inhibitors	30
Editorial Board	30
A DNA-encoded library special issue	30
Design, synthesis and antibacterial evaluation of oxazolidinone derivatives containing N-methylglycyl or quaternary ammonium salts	30
Discovery of trisubstituted meta-carboranes as T cell activators by regulating CD28 cytoplasmic region and SH2 domains of Grb2 and PI3K interactions	29

Design, synthesis and evaluation the bioactivities of novel 1,3-dimethyl-6-amino-1H-indazole derivatives as anticancer agents	28
Discovery of 5-methylpyrimidopyridone analogues as selective antimycobacterial agents	28
Discovery of 3-hydroxymethyl-azetidine derivatives as potent polymerase theta inhibitors	27