OOIR: Observatory of International Research

Papers

(The H4-Index of Bioorganic & Medicinal Chemistry is 30. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-05-01 to 2025-05-01.)

Article	Citations
Discovery of 3-hydroxymethyl-azetidine derivatives as potent polymerase theta inhibitors	91
Synthesis and antiproliferative activity of (−)-cleistenolide, (6S)-cleistenolide and 4-substituted cleistenolide analogues	87
Synthesis and biological evaluation of pyrazole-fused oleanolic acid derivatives as novel inhibitors of inflammatory and osteoclast differentiation	83
Novel hybrid conjugates with dual estrogen receptor α degradation and histone deacetylase inhibitory activities for breast cancer therapy	79
DNA-encoded C H functionality via photoredox-mediated hydrogen atom transformation catalysis	76
Production and synthesis of a novel 191Pt-labeled platinum complex and evaluation of its biodistribution in healthy mice	64
Crescent-shaped meta-substituted benzene derivatives as a new class of non-nucleoside ribonuclease A inhibitors	56
Synthesis and medicinal chemistry of tetronamides: Promising agrochemicals and antitumoral compounds	54
A DNA-encoded library special issue	45
Discovery of novel 2,8-diazaspiro[4.5]decan-1-one derivatives as potent RIPK1 kinase inhibitors	44
Sustainable electrochemical C(sp3) − H oxygenation using water as the oxygen source	42
Discovery of 5-methylpyrimidopyridone analogues as selective antimycobacterial agents	40
Targeting prolidase. A survey of the literature data to depict a structure-activity relationship frame and to address future studies for drug development	39
Multiple approaches to repurposing drugs for neuroblastoma	36
Design, synthesis and evaluation the bioactivities of novel 1,3-dimethyl-6-amino-1H-indazole derivatives as anticancer agents	35
Graphical abstract TOC	33
Current Japanese pharmaceutical chemistry	33
Design, synthesis and validation of a new Crimped Head-Piece for DNA-Encoded libraries generation	33
Janus dendritic ionizable lipids with fine designed headgroup and tails to improve mRNA delivery efficiency	33
Site-specific construction of triptolide-based antibody-drug conjugates	33
Graphical abstract TOC	32
Contents continued	32
Development of delivery carriers for plasmid DNA by conjugation of a helical template to oligoarginine	31
Selective targeting of human TET1 by cyclic peptide inhibitors: Insights from biochemical profiling	31
Diterpenoids from the whole plants of Croton yunnanensis and their bioactivities	31

Editorial Board	31
Exploring novel A2AAR antagonists: Design, synthesis, and evaluation of 2,6,9-trisubstituted purine derivatives as promising antifibrotic agents	31
Targeting m6A binding protein YTHDFs for cancer therapy	30
RNA-templated chemical synthesis of proapoptotic L- and d-peptides	30
Design, synthesis and antibacterial evaluation of oxazolidinone derivatives containing N-methylglycyl or quaternary ammonium salts	30
Antimycobacterial and anti-inflammatory activities of thiourea derivatives focusing on treatment approaches for severe pulmonary tuberculosis	30