Bioorganic & Medicinal Chemistry Letters

Article	Citations
Editorial Board	112
Pyrazolo-1-carbothioamides as EGR-1–DNA binding disruptors	77
Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor	64
Armeniaspirol analogues disrupt the electrical potential (ΔΨ) of the proton motive force	53
Graphical Abstract TOC	44
Editorial Board	40
Neuropilin 1-targeted near-infrared fluorescence probes for tumor diagnosis	38
Contents continued	34
Synthesis and biological evaluation of novel 1,2,3,4-tetrahydro-β-carboline derivatives as potential antibacterial agents	33
Design, synthesis and biological evaluation of alginate oligosaccharide derivatives	32
Studies on in vitro modulatory effects to base excision repair enzymes induced by small molecule binding to Deaminated CAG repeat hairpin	31
Discovery of DS-1093a: An oral hypoxia-inducible factor prolyl hydroxylase inhibitor for the treatment of renal anemia	30
Phytochemical investigation of Asarum sieboldii var. seoulense and the phenotypic profiles of its constituents against a Parkinson’s Disease olfactory cell line	30
Design and evaluation of anaplastic lymphoma kinase degraders using a covalent fumarate handle	30
Epigallocatechin and epigallocatechin-3-gallate are not inhibitors of tyrosinase	29
Discovery of a macrocyclic FAK inhibitor GZD-257 for treatment of glioblastoma	28
4′-O-methoxyethyl-2′-deoxy-uridine and cytidine ribonucleotides improve duplex stability, nuclease resistance, and elicit efficient knockdown of Bcl-2 expression	28
Synthesis of novel 5,6,6a,8-tetrahydro-1H-benzo[5,6]oxepino[2,3,4-de]quinoline fused iminosugars as uncompetitive inhibitors against α-glucosidase	27
Design and structural optimization of thiadiazole derivatives with potent GLS1 inhibitory activity	27
Discovery of structural diverse reversible BTK inhibitors utilized to develop a novel in vivo CD69 and CD86 PK/PD mouse model	25
Green synthesis and anti-biofilm activities of 3,5-disubstituted isoxazoline/isoxazole-linked secondary sulfonamide derivatives on Pseudomonas aeruginosa	25
New class of fused [3,2-b][1,2,4]triazolothiazoles for targeting glioma in vitro	25
Improved synthesis and anticancer activity of a potent neuronal nitric oxide synthase inhibitor	25
A concise review on MDM2 inhibitors and recent progress in radiopharmaceutical development for imaging MDM2 expression in tumors with PET or SPECT	24
Development of a highly potent and selective degrader of LRRK2	24

Recent progress in synthetic strategies to develop potent, HDAC8-selective, small-molecule inhibitors	24
Synthesis and evaluation of novel oxanthrene scaffold-derived oxazolidinone antibiotics with potent antitubercular activity and low cellular toxicity	24
Design, synthesis and characterizations of prodrugs of brexanolone	24
Design, synthesis and biological evaluation of tanshinone IIA derivatives as NLRP3 inflammasome inhibitors	23
SARS-CoV-2 papain-like protease (PLpro) inhibitory and antiviral activity of small molecule derivatives for drug leads	23
A PSMA-targeted doxorubicin small-molecule drug conjugate	23
Revisiting the dipeptidyl carboxypeptidase inhibitor captopril as a source of pan anti-trypanosomatid agents	23
Design and synthesis of Tetrahydroindeno[4,5-c]chromen-4(3H)-one derivatives as antiproliferative agents for prostate Cancer cells	22
A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation	22
Discovery of multitargeting single agents as a novel route to the potential treatment of neurodegenerative diseases	22
Contents continued	21
Contents continued	21
Contents continued	21
Design and activity evaluation of new EGFR tyrosine kinase inhibitors containing cyclic polyamines	20
Design, synthesis, and biological evaluation of 5ʹ-deoxy (N)-methanocarbanucleoside derivatives as A3 adenosine receptor ligands	20
Photocrosslinking and capture for the analysis of carbohydrate-dependent interactions	20
α-Fluorination of tropane compounds and its impact on physicochemical and ADME properties	19
Design, synthesis, and biological evaluation of cytochrome P450 CYP11A1 inhibitors	19
Design, synthesis, and anti-tumor evaluation of indolin-2-one derivatives based on 3D-QSAR	19
Combined antitumor efficacy of a new tanshinone IIA analog and irinotecan with alleviating gastrointestinal side effect	19
11C-labeling of 20(S)-protopanaxadiol, an aglycon of ginsenoside, based on the use of Pd(0)-mediated rapid C-[11C]methylation of boronic precursors	18
PEG-lipid-modified agonistic antibody against tumor necrosis factor receptor family elicits superior apoptosis-inducing activity against human carcinoma	17
Synthesis and evaluation of 3-hydroxyquinolin-2(1H)-one derivatives as inhibitors of tyrosinase	17
Design, synthesis and properties of peptide inhibitors based on BRCA1856-871	17
Editorial Board	16
Graphical abstract TOC	16
Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase	16
Ultrasound-dependent RNAi using TatU1A-rose bengal conjugate	16
Exploratory study of oxatomide derivatives with high P2X7 receptor inhibitory activity	16
Design, synthesis and biological evaluation of pyrimidine base hydroxamic acid derivatives as dual JMJD3 and HDAC inhibitors	16
DDD-028: A potent, neuroprotective, non-opioid compound for the treatment of diabetic neuropathy	16
Graphical abstract TOC	16
Graphical abstract TOC	16
Biocatalytic synthesis and evaluation of antioxidant and antibacterial activities of hydroxyequols	16
Graphical abstract TOC	15
Stereochemical inversion at a 1,4-cyclohexyl PROTAC linker fine-tunes conformation and binding affinity	15
Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity	15
Design, synthesis and biological evaluation of pteridine-7(8H)-one derivatives as potent and selective CDK4/6 inhibitors	15
A photoactivatable self-localizing ligand with improved photosensitivity for chemo-optogenetic control of protein localization in living cells	15
Synthesis and evaluation of lipoic acid – donepezil hybrids for Alzheimer’s disease using a straightforward strategy	15
Design, synthesis, and activity evaluation of RET protein degradation based on PROTAC and HyTTD techniques	15
Natural products targeting the NF-κB signaling pathway:Potential therapeutic drug candidates	15
An overview of cyclopropenone derivatives as promising bioactive molecules	15
Retraction notice to “Preclinical metabolism of LB42908, a novel farnesyl transferase inhibitor, and its effects on the cytochrome P450 isozyme activities” [Bioorg. Med. Chem. Lett. 22(9) (2012) 3067–	14
Lysine-reactive tag system for cell-surface protein labeling via N-acyl-N-alkyl sulfonamide chemistry	14
Discovery and optimization of (2-naphthylthio)acetic acid derivative as selective Bfl-1 inhibitor	14
Pharmacokinetic analysis of 6-O-[18F]FEE for PET imaging of EGFR mutation	14
Synthesis and pharmacological characterization of multiply substituted 2H-chromene derivatives as P2Y6 receptor antagonists	14
Comparative analysis of p-terphenylquinone and seriniquinone derivatives as reactive oxygen species-modulating agents	14
Biological evaluation of newly synthesized α-benzil monoxime thiocarbohydrazide derivatives as an antimicrobial and anticancer agent: In vitro screening and ADMET predictions	14

Structure-based discovery of sulfamoyl-ethyl-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidine amides and sulfonamides as potent B-Cell Lymphoma 6 (BCL6)-BTB inhibitors	14
Discovery and optimization of 2,3-Dihydroindole derivatives as STING receptor allosteric agonists	13
Design, synthesis, and evaluation of 1,3,4-oxadiazole-based EGFR inhibitors	13
Graphical abstract TOC	13
Editorial Board	13
Rational design, synthesis and biological evaluation of novel HIV-1 protease inhibitors containing 2-phenylacetamide derivatives as P2 ligands with potent activity against DRV-Resistant HIV-1 variants	13
Structure-activity relationship study of HIF-2α inhibitors with tricyclic scaffold	13
Design, synthesis and biological evaluation of novel cyano-cinnamate derivatives as mitochondrial pyruvate carrier inhibitors	13
Structure-activity relationship of dual inhibitors containing maleimide and imidazole motifs against glutaminyl cyclase and glycogen synthase kinase-3β	13
6-Aryl-quinazolines as novel GABAB receptor positive allosteric modulators	13
Graphical abstract TOC	13
Discovery of 3-phenyl-1H-5-pyrazolylamides as PLpro inhibitors through virtual screening and structure optimization	13
High-yield and high-purity amide bond formation using DMTMM PF6 for DNA-encoded libraries	13
(E)-3-(3-([1,1′-Biphenyl]-4-yl)-1-phenyl-1H-pyrazol-4-yl)-1-phenylprop-2-en-1-ones inducing reactive oxygen species generation through glutathione depletion	13
Design, synthesis, and antitumor activity study of novel oleanolic acid structural derivatives targeting c-Kit	13
Graphical abstract TOC	12
Neratinib derivative 7A induces apoptosis in colon cancer cells via the p53 pathway	12
Graphical abstract TOC	12
Discovery of sinomenine/8-Bis(benzylthio)octanoic acid hybrids as potential anti-leukemia drug candidate via mitochondrial pathway	12
Graphical abstract TOC	12
Editorial Board	12
Phenyl urea based adjuvants for β-lactam antibiotics against methicillin resistant Staphylococcus aureus	12
Syntheses and antitumor activities of neorautenol and shinpterocarpin analogs	12
Discovery of triazenyl triazoles as Nav1.1 channel blockers for treatment of epilepsy	12
Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma brucei	12
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides	12
Editorial Board	12
Graphical abstract TOC	12
Contents continued	12
Reinvestigation of clopidogrel bioactivation unveils new cytochrome P450-catalyzed thioester cleavage mechanism	12
Synthesis of a tricyclic hexapeptide –via two consecutive ruthenium-catalyzed macrocyclization steps– with a constrained topology to mimic vancomycin's binding properties toward D-Ala-D-Ala dipeptide	12
Design, synthesis and anti-pneumonic activity evaluation of shikonin ester derivatives	11
Enzymatic reconstitution of salicylate formation in promysalin biosynthesis	11
Identification of potent and selective inhibitors of PKR via virtual screening and traditional design	11
Design, synthesis and biological evaluation of novel cationic liposomes loaded with melphalan for the treatment of cancer	11
Discovery of novel N-(1-benzyl-1H-imidazol-2-yl)amide derivatives as melanocortin 1 receptor agonists	11
Discovery and characterization a new collagenase from Hathewaya massiliensis for effective subcutaneous adipolysis	11
Exploration of imidazothiazole and imidazopyrimidine carboxamides for enhanced antitubercular activity	11
Design, synthesis and activity evaluation of Hedgehog inhibitor Itraconazole derivatives in A549 cells	11
Direct-to-biology platform: From synthesis to biological evaluation of SHP2 allosteric inhibitors	11
Synthesis of dolutegravir derivatives modified by 1,2,3-triazole structure and their anti-inflammatory activity in LPS-induced BV2 cells	11
Recent advances and perspectives in therapeutics for mpox	11
Design, synthesis, in silico studies, and antiproliferative evaluations of novel indolin-2-one derivatives containing 3-hydroxy-4-pyridinone fragment	11
Synthesis of a new series of quinoline/pyridine indole-3-sulfonamide hybrids as selective carbonic anhydrase IX inhibitors	11
Discovery of N-Ts-3-benzylidene-indolin-2-imines as potent anti-colorectal cancer agents through suppression of the PI3K-AKT pathway	11
Design, synthesis and evaluation of clickable photoaffinity probes for nuclear lamins	11
Design, synthesis and evaluation of pterostilbene-indole hybrids as potential anticancer agents	11
Study of the reversal of metallo-β-lactamase-mediated resistance in Gram-negative bacteria by EDTMP	11
Discovery of novel 4-aminobenzamide derivatives as small molecule CBX2 inhibitors	11
Strengths and limitations of Ba/F3 cells in modelling FLT3-driven AML resistance	11
Design, synthesis and biological evaluation of cajanonic acid A analogues as potent PPAR γ antagonists	11
Investigation of the site 2 pocket of Grp94 with KUNG65 benzamide derivatives	11
Hydrazinecarbonyl-thiazol-2-acetamides with pronounced apoptotic behavior: synthesis, in vitro/in vivo anti-proliferative activity and molecular modeling simulations	10
Contents continued	10
Improving reactivity of naphthalimide-based GST probe by imparting TPP cation: Development and application for live cell imaging	10
Permeation behavior of porphyrin derivatives with different functional group positions across cancer cell membranes	10
Graphical abstract TOC	10
Synthesis, in vitro antimicrobial activity and docking studies of novel 1,2,4-oxadiazole based piperidin-1-yl-methanone analogues	10
A small molecule binding to TGGAA pentanucleotide repeats that cause spinocerebellar ataxia type 31	10
Synthesis of substrate peptides incorporating non-natural amino acids and screening study using BACE1	10
A guanidinium group is an effective mimic of the tertiary carbocation formed by isopentenyl diphosphate isomerase	10
Synthesis and biological evaluation of biotinylated ZJ-101	10
Contents continued	10
Further structural optimization and SAR study of sungsanpin derivatives as cell-invasion inhibitors	10
Synthesis of mizoribine prodrugs and their in vivo evaluation as immunosuppressive agents	10
Harnessing dual-mode RIPK1 ligands for cross-species anti-necroptosis inhibitor compounds	10
Iodophenyl-conjugated closo-dodecaborate as a promising small boron molecule that binds to serum albumin and accumulates in tumor	10
PSMA-targeted SMART molecules outfitted with SN38	10
Methyl N-(tert-butoxycarbonyl)pyridine-2-carbimidothioate: A new reagent for the synthesis of N-phenylpyridinecarboxamidine (“arylimidamide”) DNA-minor groove binders from poorly nucleophilic amines	10
Synthesis and functional evaluation of tetrahydroisoquinoline and polysubstituted benzylamine derivatives as sigma-2 receptor-targeted small-molecule probes	10
Graphical abstract TOC	10
The Pyrimidinyl Hydrazones: Selective for anti-Cancer cytotoxicity	10
Graphical abstract TOC	10
Evaluation of an ester-linked immunosuppressive payload: A case study in understanding the stability and cleavability of ester-containing ADC linkers	10
Discovery of 3-acyl-2-anilino-1,4-dihydroquinolin-4-one derivatives as potential inhibitors of methicillin-resistant Staphylococcus aureus	10
Graphical abstract TOC	10
Synthesis, modeling, and biological evaluation of anti-tubulin indole-substituted furanones	10
Highly potent anti-inflammatory, analgesic and antioxidant activities of 3,5-disubstituted tetrahydro-2H-1,3,5-thiadiazine thiones	9
Zinc-dependent deacetylases (HDACs) as potential targets for treating Alzheimer’s disease	9
Discovery of a proteolysis targeting chimera (PROTAC) as a potent regulator of FOXP3	9

Synthesis of esters and amides of 2-aryl-1-hydroxy-4-methyl-1H-imidazole-5-carboxylic acids and study of their antiviral activity against orthopoxviruses	9
Discovery of an ellipticine derivative as TLR3 inhibitor against influenza A virus and SARS-CoV-2	9
Discovery of a potent and subtype-selective TYK2 degrader based on an allosteric TYK2 inhibitor	9
Design, synthesis, and biological evaluation of 2,4-diaminopyrimidine inhibitors of hematopoietic progenitor kinase 1	9
Discovery of a potent orally available pyrazolopyridone derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor	9
A potent and selective RORγ inhibitor for the treatment of autoimmune diseases	9
Cyano-Hydrol green derivatives: Expanding the 9-cyanopyronin-based resonance Raman vibrational palette	9
Corrigendum to “Discovery of 4-aminopyrimidine analogs as highly potent dual P70S6K/Akt inhibitors” [Bioorgan. Med. Chem. Lett. 50 (2021) 128352]	9
Novel drug discovery approaches for MMP-13 inhibitors in the treatment of osteoarthritis	9
Synthesis, in vitro cytotoxicity evaluation and mechanism of 5′ monosubstituted chalcone derivatives as antitumor agents	9
Imidazo[2,1-b]thiazole based indoleamine-2,3-dioxygenase 1 (IDO1) inhibitor: Structure based design, synthesis, bio-evaluation and docking studies	9
Design, synthesis and biological evaluation of novel indole-piperazine derivatives as antibacterial agents	9
New diarylpentanoids and chalcones as potential antimicrobial adjuvants	9
Synthesis of triazolopyrimidinone- and imidazotriazinone-based tankyrase inhibitors: Identification of Basroparib (STP1002) as a clinical candidate	9
A small-molecule pretargeting approach for PSMA-targeted conjugates	9
Design, synthesis and antitumor evaluation of a novel nectin-4 targeting bicyclic toxin conjugate	9
Conversion of oxadiazolo[3,4-b]pyrazines to imidazo[4,5-b]pyrazines via a tandem reduction-cyclization sequence generates new mitochondrial uncouplers	9
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido[2,3-d]pyrimidin-7-one-based SOS1 inhibitor	9
Discovery of imidazole-based apo-IDO1 inhibitors: rational design, synthesis, and biological evaluation	9
Photo-regulated PROTACs: A novel tool for temporal control of targeted protein degradation	9
Thiamine analogues featuring amino-oxetanes as potent and selective inhibitors of pyruvate dehydrogenase	8
Multifaceted roles of HDAC7 in disease and the evolving chemical toolkit for its modulation	8
Graphical abstract TOC	8
Synthesis and properties of PNA containing a dicationic nucleobase based on N4-benzoylated cytosine	8
Graphical abstract TOC	8
Recent developments of benzimidazole based analogs as potential tubulin polymerization inhibitors: A critical review	8
Graphical Abstract TOC	8
Azolo[5′,1′,2,3]pyrimido[5,4-e]tetrazolo[1,5-c]pyrimidines as dual-action antiglycators and α-glucosidase inhibitors	8
Editorial Board	8
Graphical abstract TOC	8
Synthesis and antitumor activity of a series of novel N-aryl-5-(2,2,2-trifluoroethoxy)-1,5-dihydro-2H-pyrrol-2-ones derivatives	8
Editorial Board	8
Targeted design, synthesis, molecular simulation, ADME-T and in-vitro anticancer assessment of phenyl-substituted-thioxo-tetrahydro-pyrimidin-benzenesulfonamide derivatives as potential BRAFV600E/WT i	8
Design, synthesis and antitumor activity of novel 4-oxobutanamide derivatives	8
Discovery of novel imidazo[4,5-b]pyridine derivatives as noncovalent reversible Bruton’s tyrosine kinase inhibitors	8
Design, synthesis, and biological evaluation of novel HDAC inhibitors with a 3-(benzazol-2-yl)quinoxaline framework	8
Development of chromone-thiazolidine-2,4-dione Knoevenagel conjugates as apoptosis inducing agents	8
Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM	8
The lipidation and glycosylation enabling bioactivity enhancement and structural change of antibacterial peptide G3	8
Design, synthesis and biological evaluation of sulfonylurea derivatives as NLRP3 inflammasome inhibitors	8
Contents continued	8
Discovery of BI-9787, a potent zwitterionic ketohexokinase inhibitor with oral bioavailability	8
Synthesis and preliminary immunologic properties of di-/trisaccharide-conjugates related to Bacillus anthracis	8
Graphical Abstract TOC	8
Design, synthesis, and antibacterial activity evaluation of tryptanthrin derivatives	8
SAR study of niclosamide derivatives for neuroprotective function in SH-SY5Y neuroblastoma	8
Short synthesis of a broadly Reactive, cell permeable serine hydrolase Fluorophosphonate-Alkyne probe	8
Synthesis of proposed structure of ledebourin A	8
Synthesis and evaluation of catecholamine derivatives as amyloid-beta aggregation inhibitors	8
5-Fluoro-2′-deoxyuridine as an efficient 19F NMR reporter for G-quadruplex and i-motif structures	8
Graphical Abstract Contents Continued	8
Graphical abstract TOC	8
Development of novel GI-centric prostaglandin E2 receptor type 4 (EP4) agonist prodrugs as treatment for ulcerative colitis and other intestinal inflammatory diseases	8
Synthesis of drimanyl indole fragments of drimentine alkaloids and their antibacterial activities	8
Genipin derivative induced the apoptosis and inhibited the invasion and migration of A549 cancer cells via regulation of EGFR/JAK1/STAT3 signaling	8
Graphical abstract TOC	8
Contents continued	8
Fragment-based discovery of novel phenyltriazolyl derivatives as allosteric type-I1/2 ALK inhibitors with promising antitumor effects	7
Design of cyclic peptides as novel inhibitors of ICOS/ICOSL interaction	7
Identification of sugar-containing natural products that interact with i-motif DNA	7
Design, synthesis and evaluation of the Brigatinib analogues as potent inhibitors against tertiary EGFR mutants (EGFRdel19/T790M/C797S and EGFRL858R/T790M/C797S)	7
Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease	7
An ascidian Polycarpa aurata-derived pan-inhibitor against coronaviruses targeting Mpro	7
Synthesis, antiproliferative activity, and biological profiling of C-19 trityl and silyl ether andrographolide analogs in colon cancer and breast cancer cells	7
Retraction notice to “Corrigendum to “Preclinical metabolism of LB42908, a novel farnesyl transferase inhibitor, and its effects on the cytochrome P450 isozyme activities” [Bioorg. Med. Chem. Lett. 22	7
Siderophores: Chemical tools for precise antibiotic delivery	7
Design, synthesis, and biological evaluation of novel aminopyrimidine derivatives as EGFR inhibitors	7
Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3	7
Structure-activity relationship study of antitrypanosomal analogues of gibbilimbol B using multivariate analysis and computation-aided drug design	7
The potential of Rhein's aromatic amines for Parkinson's disease prevention and treatment: α-Synuclein aggregation inhibition and disaggregation of preformed fibers	7
Identification of (−)-Epigallocateshin gallate derivatives promoting innate immune activation via 2′,3′-cyclic GMP-AMP-stimulator of interferon genes pathway	7
The structural modification and biological evaluation of tetrahydrothienopyridine derivatives as selective BChE inhibitors	7
A self-assembling peptide platform enables plasma membrane protein degradation	7
Diamino variants of piperazine-based tissue transglutaminase inhibitors	7
Discovery of L15 as a novel Vif PROTAC degrader with antiviral activity against HIV-1	7
Multigram-scale total synthesis of (±)-ambreinolide by a diastereoselective polyene cyclization	7
Editorial Board	7
Stanolone-1,2,3-Triazole derivatives: Synthesis, DNA damage in tumor cells and anti-prostate Cancer activity study	7
Rational design, synthesis, and biological evaluation of chalcone hybrids including benzoylpiperazin (phenylacetylpiperazin)-thiophene as anti- Alzheimer's agents	7
Diffusion of 1O2 along the PNA backbone diminishes the efficiency of photooxidation of PNA/DNA duplexes by biphenyl photosensitizer	7
Discovery of benzimidazole-2-amide BNZ-111 as new tubulin inhibitor	7
Graphical abstract TOC	7
Inhibitors for metallo-β-lactamases from the B1 and B3 subgroups provide an avenue to combat a major mechanism of antibiotic resistance	7
The association between oxidized low-density lipoprotein and cancer: An emerging targeted therapeutic approach?	7
Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors	7
Discovery of 4-((quinolin-8-ylthio)methyl)benzamide derivatives as a new class of SARS-CoV-2 nsp13 inhibitors	7
Graphical abstract TOC	7
Thermal treatment affects aptamers’ structural profiles	7
Design, synthesis, and activity evaluation of Asiatic acid derivatives as Survivin inhibitors	7
Discovery of a DCAF11-dependent cyanoacrylamide-containing covalent degrader of BET-proteins	7
Conformationally constrained potent inhibitors for enhancer of zeste homolog 2 (EZH2)	7
Synthesis and biological evaluation of novel 18F-labeled 2,4-diaminopyrimidine derivatives for detection of ghrelin receptor in the brain	7
Design, synthesis and antifungal activities of novel triazole derivatives with selenium-containing hydrophobic side chains	7
Inhibition of glutathione S-transferases by photoactive calix[4]arene α-ketophosphonic acids	7
Graphical abstract TOC	7