Archiv der Pharmazie

Papers
(The TQCC of Archiv der Pharmazie is 7. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2022-08-01 to 2026-08-01.)
ArticleCitations
In vitro antiviral activity of favipiravir and its 6‐ and 3‐O‐substituted derivatives against coronavirus: Acetylation leads to improvement of antiviral activity74
Cover Picture: Arch Pharm (1/2024)60
What doesn't fit is made to fit: Pim‐1 kinase adapts to the configuration of stilbene‐based inhibitors54
Isoxazole‐Based Compounds Targeting the Taxane‐Binding Site of Tubulin50
Synthesis and Biological Evaluation of Novel 2‐(Piperidin‐4‐yl)‐1,2,3,4‐tetrahydroisoquinoline and 2‐(Piperidin‐4‐yl)decahydroisoquinoline Antimycotics48
Investigating the Hepatoprotective Properties of Entresto in Hepatic Ischemia‐Reperfusion Injury in Rats: The Implication of TLR4/MYD88/NF‐KB p‐65 and PPAR‐γ/HO‐1/Nrf2 Pathways47
GOAT rs10096097 and CREB1 rs6740584 single nucleotide polymorphisms are associated with type 2 diabetes mellitus in Egyptians40
NorA Efflux Pump Inhibitors: Expanding SAR Knowledge of Pyrazolo[4,3‐c][1,2]benzothiazine 5,5‐Dioxide Derivatives36
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Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review35
Synthesis, antimycobacterial, cytotoxicity, anti‐inflammatory, in silico studies and molecular dynamics of pyrazole‐embedded thiazolidin‐4‐one hybrids32
Carboline Hybrids as Potential Multitarget‐Directed Anti‐Alzheimer's Disease Agents: A Comprehensive Analysis of Design Strategies and Structure–Activity Relationships32
Ultra‐Fast UPLC‐MS/MS Method for the Ripretinib Quantification in the HLMs Matrix With Metabolic Stability Assessment: In‐Silico Study for Toxic Alerts and the Metabolic Lability32
Structure‐guided identification of a selective sulfonamide‐based inhibitor targeting the human carbonic anhydrase VA isoform28
Issue Information: Arch Pharm (1/2026)28
Tamoxifen‐Based Dimers: Design, Synthesis, Cell Viability Evaluation on Breast Cancer Cells, and Computational Insights26
Review on the pharmacological effects and pharmacokinetics of scutellarein26
Unraveling the Anticancer Activity of Sunitinib Derivatives Through Modifications in Solvent‐Exposed Regions: Synthesis, In Vitro Evaluation, and Computational Studies25
AI‐Based Prediction of PROTAC‐ and Molecular Glue‐Mediated Ternary Complexes: A Comparative Evaluation of AlphaFold 3 and Boltz‐225
Combating DC‐SIGN‐mediated SARS‐CoV‐2 dissemination by glycan‐mimicking polymers24
Synthesis of novel pyrimido[4,5‐b]quinoline derivatives as dual EGFR/HER2 inhibitors as anticancer agents24
Aripiprazole as an Inhibitor of the EGFR/PI3K/AKT Signaling Pathway and Sensitizer of MPA Suppressed Progestin‐Resistant Endometrial Cancer Cells24
Fabrication of sulfobutylether‐β‐cyclodextrin/glabridin inclusion complex for promoting bioactivities24
Sustainable RP‐HPLC Method Development for Simultaneous Estimation of Fampridine and Monomethyl Fumarate in Lipid Nanocarriers and Biological Fluids: Application of AQbd Principles23
Structure–Activity Relationship Study on Ligands Activating the Voltage‐Gated Potassium Channel K V 7.123
DCAF16‐Based Covalent Molecular Glues for Targeted Protein Degradation of Histone Deacetylases23
Discovery of xanthone‐based nitric oxide donors targeting biofilm clearance23
Functional combination of resveratrol and tamoxifen to overcome tamoxifen‐resistance in breast cancer cells23
Design, synthesis, and activity evaluation of novel multitargeted l‐tryptophan derivatives with powerful antioxidant activity against Alzheimer's disease23
Piperlongumine and its derivatives against cancer: A recent update and future prospective23
Medicinal Chemistry, SAR, and Molecular Insights Into 2,4‐Thiazolidinediones as Antidiabetic Agents (2020–2025)23
Synthesis and biological evaluation of salophen nickel(II) and cobalt(III) complexes as potential anticancer compounds23
Design, synthesis and biological evaluation of (E)‐kojyl‐styryl‐sulfones: Novel recilisib hybrids as promising radioprotectors22
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Cover Picture: Arch Pharm (7/2023)21
Aromatic linker variations in novel dopamine D2 and D3 receptor ligands21
Editorial Board: Arch Pharm (10/2023)20
Microwave‐Enhanced Synthesis of 2‐Styrylquinoline‐4‐Carboxamides With Promising Anti‐Lymphoma Activity20
Optimization of 4‐amino‐pyridazin‐3(2H)‐one as a valid core scaffold for FABP4 inhibitors20
Cover Picture: Arch Pharm (2/2024)20
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Discover the Power of Lithospermic Acid as Human Carbonic Anhydrase VA and Pancreatic Lipase Inhibitor Through In Silico and In Vitro Studies20
Issue Information: Arch Pharm (5/2025)20
The Therapeutic Potential of Berberine in Lung Cancer20
Novel tetrahydropyran‐triazole hybrids with antiproliferative activity against human tumor cells19
Fully Synthetic Non‐Carbohydrate Heparin Mimetics—Perspectives for Therapeutic Anticoagulation and Beyond?19
New chimeric HDAC inhibitors for the treatment of colorectal cancer19
Design, synthesis, biological evaluation, and molecular modeling simulations of new phthalazine‐1,4‐dione derivatives as anti‐Alzheimer's agents19
Unveiling the Therapeutic Potential of Dulaglutide in Mitigating Tacrolimus‐Induced Nephrotoxicity Through Targeting the miR‐22/HMGB‐1/TLR4/MyD88/NF‐κB Trajectory19
Green Synthetic Strategies for Pyrazole Derivatives: A Comprehensive Review19
The discovery of a new nonbile acid modulator of Takeda G protein‐coupled receptor 5: An integrated computational approach18
Unprecedented carbonic anhydrase inhibition mechanism: Targeting histidine 64 side chain through a halogen bond18
Structural determinants of sphingosine‐1‐phosphate receptor selectivity18
Liposomal formulation of model pentathiepin improves solubility and stability toward glutathione while preserving anticancer activity18
Design, synthesis, and evaluation of dual‐target inhibitors for the treatment of Alzheimer's disease18
Exploration of 3‐aryl pyrazole‐tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors18
Uncovering chemical profiles, biological potentials, and protection effect against ECM destruction in H2O2‐treated HDF cells of the extracts of Stachys tundjeliensis18
Novel therapeutic strategies and drugs for idiopathic pulmonary fibrosis18
Discovery of novel pyrazole and pyrazolo[1,5‐a]pyrimidine derivatives as cyclooxygenase inhibitors (COX‐1 and COX‐2) using molecular modeling simulation17
Evaluation of the effect of carvedilol orodispersible tablets on ischemia–reperfusion injury and flap viability in rats: An in vivo study17
Replacing the oxidation‐sensitive triaminoaryl chemotype of problematic KV7 channel openers: Exploration of a nicotinamide scaffold17
Novel benzothiazole/benzothiazole thiazolidine‐2,4‐dione derivatives as potential FOXM1 inhibitors: In silico, synthesis, and in vitro studies17
Spirooxadiazoline‐oxindoles derived from imatinib show antimyeloproliferative potential in K562 cells17
Efficient Radiosynthesis of 99m Tc‐Amygdalin for Tumor Imaging Using a 99 Mo/ 16
Combining chemical profiles and biological abilities of different extracts from Tanacetum nitens (Boiss. & NoëGrierson using network pharmacology15
Identification of 3‐(5‐cyano‐6‐oxo‐pyridin‐2‐yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity15
Implication of Central β2 Adrenergic Receptor for the Development of Novel Drugs Against Alzheimer's Disease15
N‐[4‐(Benzyloxy)‐3‐methoxybenzyl)]adamantane‐1‐amine (DZH2), a dual CCR5 and CXCR4 inhibitor as a potential agent against triple negative breast cancer15
Small Molecules, Big Impact: Structural Innovations Driving PD‐L1 Checkpoint Modulation15
Synthesis of new phenothiazine derivatives: Molecular docking, assessment of cytotoxic activity and oxidant–antioxidant properties on PCS‐201‐012, HT‐29, and SH‐SY5Y cell lines15
Exploring the Antidiabetic Potential of Heterophylliin A From Elaeocarpus grandis15
Harnessing Hybrid Chemistry: Novel Ethyl Ferulate Ester of Niflumic Acid for Enhanced Therapeutic Benefits15
Peripheral (E)‐2‐[(4‐hydroxybenzylidene)‐3,4‐dihydronaphthalen‐1(2H)‐one)]‐coordinated phthalocyanines with improved enzyme inhibition properties and photophysicochemical behaviors15
Design, synthesis, and biological evaluation of simplified tetrahydroisoquinoline analogs15
Identification of Novel β ‐Lactam Derivatives as Proteasome Inhibitors for Antitumor Therapy15
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Cytotoxic derivatives of dichloroacetic acid and some metal complexes14
Hydrazinated geraniol derivatives as potential broad‐spectrum antiprotozoal agents14
New benzimidazole‐oxadiazole derivatives: Synthesis, α‐glucosidase, α‐amylase activity, and molecular modeling studies as potential antidiabetic agents14
Algal–Bacterial Interaction‐Driven Secondary Metabolites From Phaeobacter inhibens and Their Anti‐Allergic Effects on Th2 Cell Immune Response14
5‐methyl‐2‐carboxamidepyrrole‐based novel dual mPGES‐1/sEH inhibitors as promising anticancer candidates14
Current scenario of fused pyrimidines with in vivo anticancer therapeutic potential14
Unveiling the chemistry of 1,3,4‐oxadiazoles and thiadiazols: A comprehensive review14
Recent updates on 1,2,3‐, 1,2,4‐, and 1,3,5‐triazine hybrids (2017–present): The anticancer activity, structure–activity relationships, and mechanisms of action14
Synthesis, Characterization and Evaluation of Antioxidant and Antimicrobial Activities of Novel Isatin Derivatives14
Investigating the Telomerase Downregulatory Potential of Steroidal Drugs Following Pharmacophore‐Based Rational; Computational and In Vitro Assessments14
Synthesis of novel benzylamine antimycotics and evaluation of their antimycotic potency13
A literature review on pharmacological aspects, docking studies, and synthetic approaches of quinazoline and quinazolinone derivatives13
Discovery of potent CSK inhibitors through integrated virtual screening and molecular dynamic simulation13
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Cover Picture: Arch Pharm (6/2023)13
New PEPPSI‐Pd‐NHC complexes bearing 4‐hydroxyphenylethyl group: Synthesis, characterization, molecular docking, and bioactivity properties13
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Piperazine‐based P2X4 receptor antagonists13
Conjugates of amiridine and thiouracil derivatives as effective inhibitors of butyrylcholinesterase with the potential to block β‐amyloid aggregation13
In Vitro, In Silico and Structure–Activity Relationship Evaluation of 3‐Amino‐thiophene‐2‐carbohydrazides as Lactoperoxidase Inhibitors13
Synthesis, Antituberculosis Evaluation and Structure–Activity Relationships of New SQ109 Analogs13
Review of β‐carboline and its derivatives as selective MAO‐A inhibitors13
Quantum dots in the biomedical world: A smart advanced nanocarrier for multiple venues application13
Issue Information: Arch Pharm (4/2025)13
Screening of Chelidonium majus isoquinoline alkaloids reveals berberine and chelidonine as selective ligands for the nuclear receptors RORβ and HNF4α, respectively13
Tetrazole Derivatives as Multiclass Inhibitors of Bacterial Carbonic Anhydrases12
Role of Brusatol in Preventing Gastrointestinal Cancer: Recent Trends and Future Perspectives12
Synthesis and evaluation of novel almazole D analogs as anticancer agents12
Silybin loaded Ag‐nanoparticles as a drug delivery system for solid tumor theragnosis: Extraction, radioiodination, and biodistribution study12
Design, synthesis, and evaluation of novel 3,4‐isoxazolediamide derivatives for the combination treatment of azole‐resistant candidiasis12
Unlocking the potential of edible Ulva sp. seaweeds: Metabolomic profiling, neuroprotective mechanisms, and implications for Parkinson's disease management12
Design, synthesis, acetylcholinesterase, butyrylcholinesterase, and amyloid‐β aggregation inhibition studies of substituted 4,4ʹ‐diimine/4,4ʹ‐diazobiphenyl derivatives12
Solvent and Catalyst‐Free One‐Pot Synthesis of Tetrahydropyrimidine Analogs for Their Larvicidal Activity and Structural Insights12
A new series of hydrazones as small‐molecule aldose reductase inhibitors12
Current Landscape of Hydroxamic Acid Hybrids With Anti‐Colorectal Cancer Potential12
Design and Synthesis of Novel Pyridazinone Derivatives as Cardiac Myosin Activator for the Systolic Heart Failure12
Decoding MYC Targeted Inhibition in Cancer: Integrating Medicinal Insights With Computational Design Approaches12
Recent Advancements and Developments of Anti‐Malarial Agents Reported in 202312
Synthesis and photodynamic activity of new 5‐[(E)‐2‐(3‐alkoxy‐1‐phenyl‐1H‐pyrazol‐4‐yl)ethenyl]‐2‐phenyl‐3H‐indoles12
Identification of novel sulfathiazole‐triazolo‐chalcone hybrids as VEGFR‐2/EGFR dual inhibitors with antiangiogenic activity and apoptotic induction12
A Multifaceted Mechanistic Approach to Assess the Inhibitory Potential of Broccoli‐Derived Glucosinolates Against Tumor‐Associated Carbonic Anhydrase IX12
Therapeutic Horizons in Targeting EZH2 With Dual and Non‐PROTAC Inhibitor Molecules: Recent Achievements, Comparative Analysis, and Future Perspectives12
Current Scenario of Hydroxamic Acid Derivatives With In Vivo Antitumor Therapeutic Potential11
Advances in polysaccharide‐based materials for biomedical and pharmaceutical applications: A comprehensive review11
The therapeutic potential of indole hybrids, dimers, and trimers against drug‐resistant ESKAPE pathogens11
Editorial Board: Arch Pharm (9/2023)11
Xanthenone Orchestrates the Renin–Angiotensin System/Ferroptosis Crosstalk: A Novel AT2R‐Dependent Strategy Against Lower Limb Transient Ischemia‐Induced Liver Injury11
Тhio‐containing pteridines: Synthesis, modification, and biological activity11
Development of New Thiadiazole Derivatives as VEGFR‐2 Inhibitors With Anticancer and Proapoptotic Activities‏11
5,6‐Dihydrotetrazolo[1,5‐c]quinazolines: Toxicity prediction, synthesis, antimicrobial activity, molecular docking, and perspectives11
Electro‐Mechanical Uncoupling of K V 7.1 Voltage Sensor and Pore by 1,4‐Benzodiazepines Is Modulated by Decoration of Position 111
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Discovery of C2: A Novel Lead Compound for the Treatment of Gout and Hyperuricemia via Multi‐Pathway Inhibition11
Discovery of 4‐(isopentyloxy)‐3‐nitrobenzamide derivatives as xanthine oxidase inhibitors through a non‐anthraquinone exploration11
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Novel quinazoline–chromene hybrids as anticancer agents: Synthesis, biological activity, molecular docking, dynamics and ADME studies11
Design, Synthesis, and Molecular Evaluation of SNAr‐Reactive N‐(6‐Fluoro‐3‐Nitropyridin‐2‐yl)Isoquinolin‐3‐Amines as Covalent USP7 Inhibitors Reveals an Unconventional Binding Mode11
Issue Information: Arch Pharm (4/2024)11
Development of 1‐(2‐aminophenyl)pyrrole‐based amides acting as human topoisomerase I inhibitors11
Beyond the Shadow of Indole: Medicinal Chemistry of Indolizines and Isoindolinones in the Fight Against Infectious Diseases11
A virtual library of small molecules mimicking dipeptides11
Targeting the binding pocket of the fluorophore 8‐anilinonaphthalene‐1‐sulfonic acid in the bacterial enzyme MurA10
An overview of the latest outlook of sulfamate derivatives as anticancer candidates (2020–2024)10
Design, synthesis, and structure–activity studies of new rhodanine derivatives as carbonic anhydrase II, IX inhibitors10
New paracetamol hybrids as anticancer and COX‐2 inhibitors: Synthesis, biological evaluation and docking studies10
Inhibitory effects of 190 compounds against SARS‐CoV‐2 Mpro protein: Molecular docking interactions10
Synthesis, structure–activity relationship, and biological evaluation of quinolines for development of anticancer agents10
Research progress on the pathogenesis of psoriasis and its small molecule inhibitors10
Structure Characterization and Antibacterial, Antifungal, and Antiquorum‐Sensing Activity of New Metabolites From the Lipophilic Fractions of Platycodon grandiflorum 10
Synthesis, characterization, biochemical, and molecular modeling studies of carvacrol‐based new thiosemicarbazide and 1,3,4‐thiadiazole derivatives10
Issue Information: Arch Pharm (1/2025)10
Health benefits of fraxetin: From chemistry to medicine10
A novel indole derivative, 2‐{3‐[1‐(benzylsulfonyl)piperidin‐4‐yl]‐2‐methyl‐1H‐indol‐1‐yl}‐1‐(pyrrolidin‐1‐yl)ethenone, suppresses hedgehog signaling and drug‐resistant tumor growth10
Deciphering Anticoagulant Active Substances and Mechanisms in Guanxinjing Formula Through Phenotype‐Anchored Hierarchical Strategy and Topological Network Analysis10
Rational Design of 6‐Amino‐2‐Piperazinylpyridine‐Based ROCK2 Inhibitors With Anti‐Breast Cancer Metastatic Efficiency10
Medicinal Insights Into FLT3 Inhibitors as Anticancer Agents: Current Status and Future Direction10
Various pharmacological agents in the pipeline against intractable epilepsy10
Synthesis and biological evaluation of benzamide‐chalcone hybrids as potential c‐Met kinase and COX‐2 inhibitors10
Structural Advances in Non‐Sulfonamide Carbonic Anhydrase Inhibitors: Insights Into Design, Bioactivity, and Binding Mechanism10
Multitargeted inhibition of key enzymes associated with diabetes and Alzheimer's disease by 1,3,4‐oxadiazole derivatives: Synthesis, in vitro screening, and computational studies10
Greenness‐by‐design approach for developing novel UV spectrophotometric methodologies resolving a quaternary overlapping mixture10
Synthesis, anticholinesterase activity, molecular docking, and molecular dynamic simulation studies of 1,3,4‐oxadiazole derivatives10
Design, synthesis of novel thiazole‐thiomorpholine derivatives and evaluation of their anticancer activity via in vitro and in silico studies10
New 1,3,4‐Thiadiazole‐Based Dual B‐Raf/VEGFR‐2 Inhibitors With Potential Anti‐Breast Activity: Design, Synthesis, In Vitro and In Silico Evaluations10
The carbonic anhydrase enzymes as new targets for the management of neglected tropical diseases10
3‐[3‐(Phenalkylamino)cyclohexyl]phenols: Synthesis, biological activity, and in silico investigation of a naltrexone‐derived novel class of MOR‐antagonists10
Issue Information: Arch Pharm (12/2024)10
Nature‐Inspired Compounds Targeting Escherichia coli WrbA as Biofilm‐Modulating Agents: Computational Design, Synthesis, and Biological Evaluation9
Design, Synthesis and Evaluation of Indole‐Based 1,2,3‐Triazoles as Potential Quorum Sensing and Biofilm Inhibitors Against Pseudomonas aeruginosa9
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Proapoptotic effects of halogenated bis‐phenylthiourea derivatives in cancer cells9
Metabolic profiling of Verbena bonariensis L. extract by LC/MS and evaluation of the hepatoprotective potential with isoniazid‐ and rifampicin‐induced hepatotoxicity in rats9
MCC950 as a promising candidate for blocking NLRP3 inflammasome activation: A review of preclinical research and future directions9
Indoles—A Targeting the PI3K/Akt/mTOR Pathway: Recent Advances in Strategic Design, Mechanism, and Future Perspectives9
Development of new pyrazoles as class I HDAC inhibitors: Synthesis, molecular modeling, and biological characterization in leukemia cells9
Dihydropyrimidinones as potent anticancer agents: Insight into the structure–activity relationship9
Harnessing Fragment Merging and Chain Extension Approaches for Designing Phthalimidoalkyl‐Arylidene Thiazolidinedione Hybrids: New Frontiers in Apoptosis‐Inducing Cancer Treatment9
In‐vitro and in‐silico investigations of SLC‐0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors9
The current landscape of coumarin hybrids with antibreast cancer therapeutic applications: An updated review9
Self‐microemulsifying drug delivery system‐based gastroretentive in situ raft of pazopanib with enhanced solubility and bioavailability9
Innovative Pyrazole–Thiazole–Oxadiazole Hybrid Compounds for Targeted EGFR/VEGFR2 Inhibition in Cancer Treatment9
Development and Synthesis of Bioactive (3‐Arylediene‐1‐phenyl‐1 H ‐pyrazol‐4‐yl)acryloyl‐4‐hydroxy‐6‐methyl‐2 H 9
1,3,4‐Thiadiazole and 1,2,4‐triazole‐5‐thione derivatives bearing 2‐pentyl‐5‐phenyl‐2,4‐dihydro‐3H‐1,2,4‐triazole‐3‐one ring: Synthesis, molecular docking, urease inhibition, and crystal struct9
Bruceantin and Brusatol: Molecular Insights and Therapeutic Promise of Quassinoids in Cancer Drug Discovery9
Editorial Board: Arch Pharm (9/2022)9
Pyrazole scaffold‐based derivatives: A glimpse of α‐glucosidase inhibitory activity, SAR, and route of synthesis9
New phenylthiosemicarbazide‐phenoxy‐1,2,3‐triazole‐N‐phenylacetamides as dual inhibitors against α‐glucosidase and PTP‐1B for the treatment of type 2 diabetes9
Design, Synthesis, and Selective Antiproliferative Activity of Indolizine Derivatives as Microtubule Destabilizers9
The anti‐breast cancer potential of indole/isatin hybrids9
Eco‐friendly approaches to 1,3,4‐oxadiazole derivatives: A comprehensive review of green synthetic strategies9
Design and synthesis of benzofuran‐ and naphthalene‐fused thiazinones as antimycobacterial agents9
Novel RP‐HPLC method for estimation of a newly developed combination of tizanidine and etoricoxib in rat plasma: Eight criteria for greens evaluation8
Development and in vitro antiviral activity of ivermectin liposomes as a potential drug carrier system8
Cover Picture: Arch Pharm (8/2023)8
Cover Picture: Arch Pharm (10/2023)8
Morpholinodiazenyl chalcone blocks influenza A virus capsid uncoating by perturbing the clathrin‐mediated vesicular trafficking pathway8
Harnessing PHGDH Inhibition for Cancer Therapy: Mechanisms, SAR, Computational Aspects, and Clinical Potential8
EGB761 ameliorates mild cognitive impairment by inhibiting the pyroptosis and apoptosis in both in vivo and in vitro experiments8
A review of recent advances in anticancer activity and SAR of pyrazole derivatives8
Synthesis of new dihydropyrimidine derivatives and investigation of their antimicrobial and DNA gyrase inhibitory activities8
Combating Drug‐Resistant Protozoal Infections: A Review of Emerging Therapeutics8
Synthesis of selenophene‐based chalcone analogs and assessment of their biological activity as anticancer agents8
Multi‐Angle Bioactivity Cartography for Computational Screening and Mechanistic Analysis of AChE Inhibitors From Yellow Gastrodia elata8
Exosomal miR‐122, miR‐128, miR‐200, miR‐298, and miR‐342 as novel diagnostic biomarkers in NAFL/NASH: Impact of LPS/TLR‐4/FoxO3 pathway8
Exploring Novel Nitrofuryl‐1,3,4‐Thiadiazole‐Based Derivatives: Design, Synthesis, and Evaluation of In Vitro Leishmanicidal and Trypanocidal Activity8
Quinolinone Derivatives Suppress Angiogenesis in Human Umbilical Vein Endothelial Cells by Blocking the VEGF‐Induced VEGFR2 Signaling Pathway8
Design, synthesis, and biological evaluation of naphthalene imidazo[1,2‐b]pyridazine hybrid derivatives as VEGFR selective inhibitors8
Revealing a Gold Mine of Bioactive Compounds From Natural Sources Using In Vitro, In Silico, and Network Pharmacology: A Case Study on Cachrys cristata8
Rational Design, Green Synthesis, and Biological Evaluation of Novel Imidazole Derivatives as Potent EGFR Inhibitors via One‐Pot Four‐Component Reaction8
Synthesis and evaluation of febrifugine derivatives as anticoccidial agents8
Emerging green synthetic routes for thiazole and its derivatives: Current perspectives8
4‐{3‐[(Pyridin‐4‐ylmethyl)amino]‐[1,2,4]triazolo[4,3‐b][1,2,4]triazin‐6‐yl}phenol: An improved anticancer agent in hepatocellular carcinoma and a selective MDR1/MRP modulator8
Current Landscape of Indole Hybrids in the Design and Development of Anti‐Alzheimer Agents: Structural Insights, Therapeutic Potential and In Silico Studies8
New azaaurone derivatives as potential multitarget agents in HIV‐TB coinfection8
Corrigendum to “Design, Synthesis, Biological Evaluation, and In Silico Studies of Quinoxaline Derivatives as Potent p38αMAPK Inhibitors”8
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Recent Progress and Therapeutic Potential of Indole Hybrids Against Colorectal Cancer8
Design, Synthesis, and Biological Evaluation of Novel Benzimidazole/Schiff Base Hybrid Derivatives With Potential Biological Activities7
Soft drug inhibitors for the epigenetic targets lysine‐specific demethylase 1 and histone deacetylases7
6‐Aminocoumarin oxime‐ether/sulfonamides as selective hCA IX and XII inhibitors: Synthesis, evaluation, and molecular dynamics studies7
The anti‐Acinetobacter baumannii therapeutic potential of azole hybrids: A mini‐review7
Sequential Optimization Approach Toward an Azapeptide‐Based SARS‐CoV‐2 Main Protease Inhibitor7
Discovery of Furopyrimidine‐Pyrazole Hybrid Compounds Targeting p53‐MDM2 Interaction as Anticancer Agents7
Radiosynthesis and whole‐body distribution in mice of a 18F‐labeled azepino[4,3‐b]indole‐1‐one derivative with multimodal activity for the treatment of Alzheimer's disease7
A decade of research effort in synthesis, biological activity assessments, and mechanistic investigations of sulfamethazine‐incorporating molecules7
Repurposing of 5‐nitrofuran‐3,5‐disubstituted isoxazoles: A thriving scaffold to antitrypanosomal agents7
Novel Purine‐Based Natural Products as Inhibitors of Cholinesterases and Monoamine Oxidases Presenting Potential Multitarget Therapeutics Tackling Alzheimer's Disease7
New Benzimidazole Scaffolds Tagged With Isatin/Thiourea Motifs as Anti‐Cancer Agents: Promising Approach for VEGFR‐2 Inhibition7
Dual Anti‐Cancer and Anti‐Inflammatory Activity of Some New Benzofuran‐Thiazole Hybrids With Promising COX‐2 Inhibitory Potency: Cell‐Cycle Arrest, Apoptosis, and Safety Study7
Identification of vilazodone as a novel plasminogen activator inhibitor to overcome Alzheimer's disease through virtual screening, molecular dynamics simulation, and biological evaluation7
Synthesis of benzylated amine‐substituted xanthone derivatives and their antioxidant and anti‐inflammatory activities7
Novel N‐pyrocatechoyl and N‐pyrogalloyl hydrazone antioxidants endowed with cytotoxic and antibacterial activity7
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Recent advances in the development of celecoxib analogs as anticancer agents: A review7
The synergy between nucleotide biosynthesis inhibitors and antiviral nucleosides: New opportunities against viral infections?7
A Review on Curcumin: Pharmacological Promises and Biomedical Activities7
Facile one‐pot synthesis of N‐pyridinylaminonaphthol derivatives and their antibacterial evaluation against multidrug‐resistant Staphylococcus aureus7
The effects of morin and methotrexate on pentose phosphate pathway enzymes and GR/GST/TrxR enzyme activities: An in vivo and in silico study7
Uro‐Protective Role of Lacosamide Against Cyclophosphamide‐Induced Cystitis via Notch1/NICD/NF‐ κ B Pathway: Network Pharmacology, Molecular Docking, and7
Novel 2‐oxo‐2‐phenylethoxy and benzyloxy diaryl urea hybrids as VEGFR‐2 inhibitors: Design, synthesis, and anticancer evaluation7
Development of Potent Type V MAPK Inhibitors: Design, Synthesis, and Biological Evaluation of Benzothiazole Derivatives Targeting p38α MAPK in Breast Cancer Cells7
Design and synthesis of novel substituted s‐triazines tethered benzenesulfonamides as potential antimicrobial candidates: Antibiofilm and bacterial protein permeability assessments7
Inhibition of Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (ENPP1): A Medicinal Chemistry Approach at the Crossroad of Immunotherapy and Metabolic Modulation7
K v 7 and K 2P Potassium Channels in Thalamocortical Function and Their Therapeutic Potential in C7
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TERRA G‐quadruplex stabilization behind the anti‐multiple myeloma activity: Novel insights about resveratrol pleiotropic effects7
Exploring Micellar Systems for Intra‐Articular Delivery of Vanillic Acid in Management of Osteoarthritis7
Unraveling the chemical profile, antioxidant, enzyme inhibitory, cytotoxic potential of different extracts from Astragalus caraganae7
Natural products against tau hyperphosphorylation‐induced aggregates: Potential therapies for Alzheimer's disease7
Cover Picture: Arch Pharm (9/2023)7
Chicoric acid alleviates rotenone‐induced motor dysfunction in mice: Targeting PI3K/AKT/caspase‐3‐associated apoptosis and neuroinflammation7
Issue Information: Arch Pharm (2/2026)7
Support Vector Machine Identification of Small Molecule Binders to an Understudied Allosteric Site of SARS‐CoV‐2 Mpro for Next‐Generation PROTAC‐Based Therapeutics7
Structure‐Based Design of Chiral Thioureas as Anticholinesterase Inhibitors Using Enantiopure α‐Methylbenzylamines: Synthesis, Enzyme Inhibition, and In Silico Studies7
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