Archiv der Pharmazie

Article	Citations
Cover Picture: Arch Pharm (4/2024)	193
Combating DC‐SIGN‐mediated SARS‐CoV‐2 dissemination by glycan‐mimicking polymers	179
On the hunt for metalloenzyme inhibitors: Investigating the presence of metal‐coordinating compounds in screening libraries and chemical spaces	69
Synthesis and evaluation of febrifugine derivatives as anticoccidial agents	63
Editorial Board: Arch Pharm (2/2021)	61
SC‐560 and mofezolac isosteres as new potent COX‐1 selective inhibitors with antiplatelet effect	49
Issue Information: Arch Pharm (8/2024)	46
GOAT rs10096097 and CREB1 rs6740584 single nucleotide polymorphisms are associated with type 2 diabetes mellitus in Egyptians	39
Fabrication of sulfobutylether‐β‐cyclodextrin/glabridin inclusion complex for promoting bioactivities	39
1,2,3‐Triazole‐based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition	36
New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzo[4,5]imidazo[1,2‐a][1,3,5]triazine scaffold: Synthesis and pharmacological effects	35
Synthesis and antimicrobial testing of 5‐fluorouracil derivatives	33
Cover Picture: Arch Pharm (1/2022)	33
Editorial Board: Arch Pharm (1/2022)	32
In vitro and in vivo evaluation of a water‐in‐oil microemulsion of platycodin D	31
Analysis of histamine and sisomicin in gentamicin: Search for the causative agents of adverse effects	31
Pioneering first‐in‐class FAAH‐HDAC inhibitors as potential multitarget neuroprotective agents	31
	30
Archiv der Pharmazie—200 years	30
Natural cyclic polypeptides as vital phytochemical constituents from seeds of selected medicinal plants	28
	27
Issue Information: Arch Pharm (5/2024)	27
Extracting binding energies and binding modes from biomolecular simulations of fragment binding to endothiapepsin	26
Design, synthesis, and activity evaluation of novel multitargeted l‐tryptophan derivatives with powerful antioxidant activity against Alzheimer's disease	25
Implication of in silico studies in the search for novel inhibitors against SARS‐CoV‐2	24

N‐Substituted piperidine‐3‐carbohydrazide‐hydrazones against Alzheimer's disease: Synthesis and evaluation of cholinesterase, beta‐amyloid inhibitory activity, and antioxidant capacity	24
Recent green approaches for the synthesis of pyrazolo[3,4‐d]pyrimidines: A mini review	24
Structure–activity relationship study to improve cytotoxicity and selectivity of lonafarnib against breast cancer cells	23
Editorial Board: Arch Pharm (9/2022)	23
	23
New 3‐(1H‐benzo[d]imidazol‐2‐yl)quinolin‐2(1H)‐one‐based triazole derivatives: Design, synthesis, and biological evaluation as antiproliferative and apoptosis‐inducing agents	23
What doesn't fit is made to fit: Pim‐1 kinase adapts to the configuration of stilbene‐based inhibitors	23
New 1,2,4‐oxadiazole/pyrrolidine hybrids as topoisomerase IV and DNA gyrase inhibitors with promising antibacterial activity	21
Suppression of the TRIF‐dependent signaling pathway of TLRs by epoxomicin	21
Cover Picture: Arch Pharm (3/2022)	21
Indole derivatives targeting colchicine binding site as potential anticancer agents	19
The anti‐breast cancer therapeutic potential of 1,2,3‐triazole‐containing hybrids	19
Multitarget‐directed therapeutics: (Urea/thiourea)2 derivatives of diverse heterocyclic‐Lys conjugates	19
New [1,2,4]triazolo[4,3‐c]quinazoline derivatives as vascular endothelial growth factor receptor‐2 inhibitors and apoptosis inducers: Design, synthesis, docking, and antiproliferative evaluatio	18
Synthesis and biological profile of benzoxazolone derivatives	18
Synthesis and biological evaluation of sulfonamide‐based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae	18
An exploratory study on the effect of mechanical stress on particle formation in monoclonal antibody infusions	18
Editorial Board: Arch Pharm (1/2024)	17
Synthesis and evaluation of novel xanthene‐based thiazoles as potential antidiabetic agents	17
Cover Picture: Arch Pharm (1/2024)	17
Synthesis and screening of 6‐alkoxy purine analogs as cell type‐selective apoptotic inducers in Jurkat cells	16
Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐b][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors	16
Thiazole‐based SARS‐CoV‐2 protease (COV Mpro) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations	16
Synthesis of novel pyrimido[4,5‐b]quinoline derivatives as dual EGFR/HER2 inhibitors as anticancer agents	16
A novel class for carbonic anhydrases inhibitors and evaluation of their non‐zinc binding	16
Cover Picture: Arch Pharm (11/2023)	15
Structure‐guided identification of a selective sulfonamide‐based inhibitor targeting the human carbonic anhydrase VA isoform	15
Exploration of 1,2,3‐triazolo fused triterpenoids as inhibitors of human coronavirus 229E targeting the viral nsp15 protein	15
C5‐Iminosugar modification of casein kinase 1δ lead 3‐(4‐fluorophenyl)‐5‐isopropyl‐4‐(pyridin‐4‐yl)isoxazole promotes enhanced inhibitor affinity and selectivity	14
Discovery of novel α‐carboline derivatives as glycogen synthase kinase‐3β inhibitors for the treatment of Alzheimer's disease	14
Synthesis and evaluation of carbamate derivatives as fatty acid amide hydrolase and monoacylglycerol lipase inhibitors	14
Curcumin‐based bioactive heterocycles derived via multicomponent reactions	14
	14
	14
Aminoalkoxy‐substituted coumarins: Synthesis and evaluation for reactivation of inhibited human acetylcholinesterase	14
Emerging green synthetic routes for thiazole and its derivatives: Current perspectives	13
Design, synthesis, and evaluation of 4′‐phosphonomethoxy pyrimidine ribonucleosides as potential anti‐influenza agents	13
Synthesis and biological evaluation of coumarin‐thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors	13
Strategies in synthetic design and structure–activity relationship studies of novel heterocyclic scaffolds as aldose reductase‐2 inhibitors	13
Biological functions of kojic acid and its derivatives in medicine, cosmetics, and food industry: Insights into health aspects	13
Microwave‐induced one‐pot synthesis of 3‐imidazolyl indole clubbed 1,2,3‐triazole hybrids as antiproliferative agents and density functional theory study	13
Synthesis and biological evaluation of new 4‐oxo‐thiazolidin‐2‐ylidene derivatives as antimicrobial agents	13
In vitro antiviral activity of favipiravir and its 6‐ and 3‐O‐substituted derivatives against coronavirus: Acetylation leads to improvement of antiviral activity	13
Absolute configuration of cytotoxic anthraquinones from a Brazilian cave soil‐derived fungus, Aspergillus sp. SDC28	12
Design and development of novel series of indole‐3‐sulfonamide ureido derivatives as selective carbonic anhydrase II inhibitors	12
Piperlongumine and its derivatives against cancer: A recent update and future prospective	12
Oxadiazole: A highly versatile scaffold in drug discovery	12
Synthesis and biological evaluation of new coumarin derivatives as cytotoxic agents	12
	12
Synthesis, characterization, and biological study of new synthetic opioid hemorphin‐4 peptides containing sterically restricted nonnatural amino acids	12

hERG stereoselective modulation by mexiletine‐derived ureas: Molecular docking study, synthesis, and biological evaluation	12
Benzotriazole scaffold: An overview of antiproliferative potential, mechanisms of action, and structure–activity relationships	12
Comparative analysis of apocarotenoids and phenolic constituents of Crocus sativus stigmas from 11 countries: Ecological impact	12
Biosynthesized metallic nanoparticles: A new era in cancer therapy	12
Design, synthesis, cytotoxicity, and molecular docking studies of novel thiazolyl–hydrazone derivatives as histone lysine acetyl‐transferase inhibitors and apoptosis inducers	12
Synthesis of 3‐hydroxy‐2‐naphthohydrazide‐based hydrazones and their implications in diabetic management via in vitro and in silico approaches	11
The C‐terminally shortened analogs of a hexapeptide derived from Lingzhi hydrolysate with enhanced tyrosinase‐inhibitory activity	11
Synthesis, density functional theory calculation, molecular docking studies, and evaluation of novel 5‐nitrothiophene derivatives for anticancer activity	11
Triazole derivatives as potential xanthine oxidase inhibitors: Design, enzyme inhibition potential, and docking studies	11
New 1,3,4‐oxadiazole‐chalcone/benzimidazole hybrids as potent antiproliferative agents	11
Synthesis and antimalarial and anticancer evaluation of 7‐chlorquinoline‐4‐thiazoleacetic derivatives containing aryl hydrazide moieties	11
Synthesis, antimycobacterial, cytotoxicity, anti‐inflammatory, in silico studies and molecular dynamics of pyrazole‐embedded thiazolidin‐4‐one hybrids	11
Isobavachalcone suppresses the TRIF‐dependent signaling pathway of Toll‐like receptors	10
5‐Fluoro/(trifluoromethoxy)‐2‐indolinone derivatives with anti‐interleukin‐1 activity	10
Discovery of N,N'‐diarylurea molecules with activity against multidrug‐resistant Staphylococcus aureus	10
Tail‐approach based design, synthesis, and molecular modeling of benzenesulfonamides carrying thiadiazole and urea moieties as novel carbonic anhydrase inhibitors	10
Exploration of cytotoxicity of iodoquinazoline derivatives as inhibitors of both VEGFR‐2 and EGFRT790M: Molecular docking, ADMET, design, and syntheses	10
New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition	10
Pyrazole scaffold‐based derivatives: A glimpse of α‐glucosidase inhibitory activity, SAR, and route of synthesis	10
Quinoxaline‐based efflux pump inhibitors restore drug susceptibility in drug‐resistant nontuberculous mycobacteria	10
A decade's overview of 2‐aminothiophenes and their fused analogs as promising anticancer agents	10
Design, synthesis, in silico ADMET, docking, and antiproliferative evaluations of [1,2,4]triazolo[4,3‐c]quinazolines as classical DNA intercalators	10
Novel 2‐substituted thioquinazoline‐benzenesulfonamide derivatives as carbonic anhydrase inhibitors with potential anticancer activity	10
Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review	10
Novel substituted 5‐methyl‐4‐acylaminoisoxazoles as antimitotic agents: Evaluation of selectivity to LNCaP cancer cells	9
Triazolo‐linked benzimidazoles as tubulin polymerization inhibitors and DNA intercalators: Design, synthesis, cytotoxicity, and docking studies	9
	9
Development and in vitro antiviral activity of ivermectin liposomes as a potential drug carrier system	9
Pharmacophore‐linked pyrazolo[3,4‐d]pyrimidines as EGFR‐TK inhibitors: Synthesis, anticancer evaluation, pharmacokinetics, and in silico mechanistic studies	9
Synthesis of 2‐(N‐cyclicamino)quinoline combined with methyl (E)‐3‐(2/3/4‐aminophenyl)acrylates as potential antiparasitic agents	9
In vitro and in silico studies of fluorinated 2,3‐disubstituted thiazolidinone‐pyrazoles as potential α‐amylase inhibitors and antioxidant agents	9
Design, synthesis, and characterization of PROTACs targeting the androgen receptor in prostate and lung cancer models	9
In‐vitro and in‐silico investigations of SLC‐0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors	9
Synthesis of 1,2,3‐triazole‐1,3,4‐thiadiazole hybrids as novel α‐glucosidase inhibitors by in situ azidation/click assembly	9
New hydrazide derivatives of N‐amino‐11‐azaartemisinin as promising epidermal growth factor receptor inhibitors for therapeutic development in triple‐negative breast cancer	9
Anticancer activities, structure–activity relationship, and mechanism of action of 12‐, 14‐, and 16‐membered macrolactones	9
Indole clubbed 2,4‐thiazolidinedione linked 1,2,3‐triazole as a potent antimalarial and antibacterial agent against drug‐resistant strain and molecular modeling studies	9
Selective cytotoxicity of ent‐kaurene diterpenoids isolated from Baccharis lateralis and Baccharis retusa (Asteraceae)	9
Discovery of sulfadrug–pyrrole conjugates as carbonic anhydrase and acetylcholinesterase inhibitors	9
Synthesis and biological evaluation of salophen nickel(II) and cobalt(III) complexes as potential anticancer compounds	9
Sulfonamide‐incorporated bis(α‐aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X‐ray crystallographic studies	9
Pyrazole/pyrazoline as an excellent pharmacophore in the design of carbonic anhydrase inhibitors (2018–2022)	9
Discovery of novel potent PI3K/mTOR dual‐target inhibitors based on scaffold hopping: Design, synthesis, and antiproliferative activity	9
Novel isoxazoline‐linked 1,3,4‐thiadiazole hybrids as anticancer agents: Design, synthesis, biological evaluation, molecular docking, and molecular dynamics simulation	9
Design, synthesis, and evaluation of new benzimidazole‏ ‏‎thiourea ‎derivatives as antitumor agents	9
Novel RP‐HPLC method for estimation of a newly developed combination of tizanidine and etoricoxib in rat plasma: Eight criteria for greens evaluation	9
Isatin thiazoles as antidiabetic: Synthesis, in vitro enzyme inhibitory activities, kinetics, and in silico studies	9
Synthesis and in vitro antiproliferative activity of certain novel pyrazolo[3,4‐b]pyridines with potential p38α MAPK‐inhibitory activity	9
Anticancer perspectives of monocarbonyl analogs of curcumin: A decade (2014–2024) review	8
Synthesis and examination of 1,2,4‐triazine‐sulfonamide hybrids as potential inhibitory drugs: Inhibition effects on AChE and GST enzymes in silico and in vitro conditions	8
Synthesis and in vitro cytotoxicity of benzoxazole‐based PPARα/γ antagonists in colorectal cancer cell lines	8
	8
Multi‐functional tyrosinase inhibitors derived from kojic acid and hydroquinone‐like diphenols for treatment of hyperpigmentation: Synthesis and in vitro biological evaluation	8
Corrigendum: The medicinal perspective of 2,4‐thiazolidinediones based ligands as antimicrobial, antitumor and antidiabetic agents: A review	8
Review on the pharmacological effects and pharmacokinetics of scutellarein	8
Correction to: Ecofriendly synthesis of pyrano[2,3‐d]pyrimidine derivatives and related heterocycles with anti‐inflammatory activities	8
Functional combination of resveratrol and tamoxifen to overcome tamoxifen‐resistance in breast cancer cells	8
Silver–N‐heterocyclic carbene complexes‐catalyzed multicomponent reactions: Synthesis, spectroscopic characterization, density functional theory calculations, and antibacterial study	8
Symmetrical 2,7‐disubstituted 9H‐fluoren‐9‐one as a novel and promising scaffold for selective targeting of SIRT2	8
Current scenario of indole hybrids with antibacterial potential against Acinetobacter baumannii pathogens: A mini‐review	8
Coumarin‐modified ruthenium complexes: Synthesis, characterization, and antiproliferative activity against human cancer cells	8
Unveiling new thiazole‐clubbed piperazine derivatives as multitarget anti‐AD: Design, synthesis, and in silico studies	8
Synthesis, biological activities, and structure–activity relationships of Morita–Baylis–Hillman adducts: An update	8
Citrus wastewater as a source of value‐added products: Quali‐quantitative analysis and in vitro screening on breast cancer cell lines	8
The current landscape of coumarin hybrids with antibreast cancer therapeutic applications: An updated review	8
Discovery of xanthone‐based nitric oxide donors targeting biofilm clearance	7
	7
Unveiling tomorrow: Carbonic anhydrase activators and inhibitors pioneering new frontiers in Alzheimer's disease	7
Phthalimide derivatives as a new class of papain‐like protease inhibitors in SARS‐CoV‐2	7
	7
Synthesis of 5‐[(1H‐indol‐3‐yl)methyl]‐1,3,4‐oxadiazole‐2(3H)‐thiones and their protective activity against oxidative stress	7
Design, synthesis, and evaluation of dual‐target inhibitors for the treatment of Alzheimer's disease	7
	7
Design and synthesis of pyridazin‐4‐one derivatives as necroptosis inhibitors	7
Identification and study of new NF‐κB‐inducing kinase ligands derived from the imidazolone scaffold	7
Natural flavonoids as promising lactate dehydrogenase A inhibitors: Comprehensive in vitro and in silico analysis	7
FDA‐approved drugs featuring macrocycles or medium‐sized rings	7
Cover Picture: Arch Pharm (10/2023)	7
A comprehensive update on the structure and synthesis of potential drug targets for combating the coronavirus pandemic caused by SARS‐CoV‐2	7
	7

Flucytosine‐based prodrug activation by cold physical plasma	7
New benzimidazole–indole–amide derivatives as potent α‐glucosidase and acetylcholinesterase inhibitors	7
Synthesis and antitumor evaluation of glycyrrhetinic acid‐dithiocarbamate hybrids	7
Evaluation of betanin‐loaded liposomal nanocarriers in AlCl3‐induced Alzheimer's disease in rats: Impact on cognitive function, neurodegeneration, and TREM2/ADAM10 pathways	7
Synthesis of new dihydropyrimidine derivatives and investigation of their antimicrobial and DNA gyrase inhibitory activities	7
2‐Oxoquinoline‐based‐thiosemicarbazones as multitargeting neurotherapeutics against Alzheimer's disease: In vitro and in silico studies of MAO and ChE inhibitors	7
Antiprotozoal agents: How have they changed over a decade?	7
Optimization of 4‐amino‐pyridazin‐3(2H)‐one as a valid core scaffold for FABP4 inhibitors	7
Novel pyrazolo[3,4‐b]pyridine derivatives: Synthesis, structure–activity relationship studies, and regulation of the AMPK/70S6K pathway	7
Fragment‐type 4‐azolylcoumarin derivatives with anticancer properties	6
Novel substituted 1,8‐naphthyridines: Design, synthesis, radiolabeling, and evaluation of apoptosis and topoisomerase II inhibition	6
Editorial Board: Arch Pharm (10/2023)	6
Editorial Board: Arch Pharm (5/2022)	6
Cover Picture: Arch Pharm (5/2024)	6
First‐in‐class pyrido[2,3‐d]pyrimidine‐2,4(1H,3H)‐diones against leishmaniasis and tuberculosis: Rationale, in vitro, ex vivo studies and mechanistic insights	6
Synthesis of new N‐(3‐oxo‐1‐thia‐4‐azaspiro[4.5]decan‐4‐yl)pyridine‐3‐carboxamide derivatives and evaluation of their anti‐influenza virus and antitubercular activities	6
Identification of active main metabolites of anti‐infective inhibitors of the macrophage infectivity potentiator protein by liquid chromatography using mass detection	6
Piperazine and piperidine‐substituted 7‐hydroxy coumarins for the development of anti‐inflammatory agents	6
Aromatic linker variations in novel dopamine D2 and D3 receptor ligands	6
	6
Thiophene‐containing compounds with antimicrobial activity	6
Bioevaluation of quinoline‐4‐carbonyl derivatives of piperazinyl‐benzothiazinones as promising antimycobacterial agents	6
Morpholinodiazenyl chalcone blocks influenza A virus capsid uncoating by perturbing the clathrin‐mediated vesicular trafficking pathway	6
Green synthesis of novel antifungal 1,2,4‐triazoles effective against γ‐irradiated Candida parapsilosis	6
	6
Synthesis of the chromone‐thiosemicarbazone scaffold as promising α‐glucosidase inhibitors: An in vitro and in silico approach toward antidiabetic drug design	6
A comparative untargeted metabolomic analysis and assessment of antiplasmodial potential of nine Albizia species	6
Spirooxadiazoline‐oxindoles derived from imatinib show antimyeloproliferative potential in K562 cells	6
Cover Picture: Arch Pharm (8/2023)	6
Discovery of 5‐alkyl‐2‐pyrazol‐oxazolidin‐4‐one derivatives as novel hepatitis B virus capsid assembly modulators	6
Replacing the oxidation‐sensitive triaminoaryl chemotype of problematic KV7 channel openers: Exploration of a nicotinamide scaffold	6
Design and synthesis of novel chalcone derivatives and evaluation of their inhibitory activities against acetylcholinesterase	6
Sulfonyl thioureas with a benzo[d]thiazole ring as dual acetylcholinesterase/butyrylcholinesterase and human monoamine oxidase A and B inhibitors: An in vitro and in silico study	6
Liposomal formulation of model pentathiepin improves solubility and stability toward glutathione while preserving anticancer activity	6
Chemical composition and biological activities of Cucurbita okeechobeensis extracts from its aerial parts, seeds, and fruit shells	6
Limonoids isolated from Chisocheton ceramicus Miq. and the antiadipogenic mechanism of action of ceramicine B	6
4‐{3‐[(Pyridin‐4‐ylmethyl)amino]‐[1,2,4]triazolo[4,3‐b][1,2,4]triazin‐6‐yl}phenol: An improved anticancer agent in hepatocellular carcinoma and a selective MDR1/MRP modulator	6
Editorial: Promising tools in targeted cancer therapy	6
Cover Picture: Arch Pharm (9/2021)	5
Design, synthesis, biological evaluation, and molecular modeling simulations of new phthalazine‐1,4‐dione derivatives as anti‐Alzheimer's agents	5
Development of fluorinated nicotinonitriles and fused candidates as antimicrobial, antibiofilm, and enzyme inhibitors	5
	5
Multitargeting in cardioprotection: An example of biaromatic compounds	5
Cover Picture: Arch Pharm (12/2022)	5
Identification of 9H‐purin‐6‐amine derivatives as novel aldose reductase inhibitors for the treatment of diabetic complications	5
	5
Editorial Board: Arch Pharm (7/2021)	5
Development of heterodimeric estrogen receptor alpha antagonists to target simultaneously the ligand and coactivator binding site	5
Synthesis of benzylated amine‐substituted xanthone derivatives and their antioxidant and anti‐inflammatory activities	5
Insights into modulating the monastrol scaffold: Development of new pyrimidinones as Eg5 inhibitors with anticancer activity	5
Cover Picture: Arch Pharm (7/2023)	5
Editorial Board: Arch Pharm (10/2022)	5
Evaluation of in vitro SARS‐CoV‐2 inactivation by a new quaternary ammonium compound: Bromiphen bromide	5
Editorial Board: Arch Pharm (6/2022)	5
	5
Editorial Board: Arch Pharm (3/2021)	5
Combining chemical profiles and biological abilities of different extracts from Tanacetum nitens (Boiss. & Noë) Grierson using network pharmacology	5
Anticancer 5‐arylidene‐2‐(4‐hydroxyphenyl)aminothiazol‐4(5H)‐ones as tubulin inhibitors	5
Editorial Board: Arch Pharm (11/2022)	5
	5
	5
Editorial Board: Arch Pharm (2/2022)	5
Editorial Board: Arch Pharm (5/2023)	5
	5
Exploration of 3‐aryl pyrazole‐tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors	4
Some phenolic natural compounds as carbonic anhydrase inhibitors: An in vitro and in silico study	4
Synthesis and molecular docking simulation of new benzimidazole–thiazole hybrids as cholinesterase inhibitors	4
Issue Information: Arch Pharm (7/2024)	4
Uncovering chemical profiles, biological potentials, and protection effect against ECM destruction in H2O2‐treated HDF cells of the extracts of Stachys tundjeliensis	4
Inhibitory effect of galantamine and donepezil combination against cholinesterase: An in silico and in vitro study	4
Design, synthesis, and biological evaluation of naphthalene imidazo[1,2‐b]pyridazine hybrid derivatives as VEGFR selective inhibitors	4
Unlocking nitrogen compounds’ promise against malaria: A comprehensive review	4
Novel therapeutic strategies and drugs for idiopathic pulmonary fibrosis	4
Structure‐guided design of potent JAK1‐selective inhibitors based on 4‐amino‐7H‐pyrrolo[2,3‐d]pyrimidine with anti‐inflammatory efficacy	4
Development and evaluation of 2,4‐disubstituted‐5‐aryl pyrimidine derivatives as antibacterial agents	4
Synthesis of selenophene‐based chalcone analogs and assessment of their biological activity as anticancer agents	4
Benzimidazolone‐piperazine/triazole/thiadiazole/furan/thiophene conjugates: Synthesis, in vitro urease inhibition, and in silico molecular docking studies	4
Nanomolar potency of imidazo[2,1‐b]thiazole analogs as indoleamine 2,3‐dioxygenase inhibitors	4
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis	4
Identification and assessment of new PIM2 inhibitors for treating hematologic cancers: A combined approach of energy‐based virtual screening and machine learning evaluation	4
New labdane diterpenoids from Alpinia galanga: A new type of GLP‐1 secretagogues targeting the PKA‐CREB and PI3K‐Akt signaling axes	4
Quinolone bioisosteres of phenolic GluN2B‐selective NMDA receptor antagonists	4
Recent advances on quinoxalines as target‐oriented chemotherapeutic anticancer agents through apoptosis	4
1,2,3‐Triazole hybrids as anticancer agents: A review	4
Quality parameters for the medicinal plant Drosera rotundifolia L.: A new approach with established techniques	4
Benzothiazole‐based apoptosis inducers: A comprehensive overview and future prospective	4
Facile synthesis of C6‐substituted benz[4,5]imidazo[1,2‐a]quinoxaline derivatives and their anticancer evaluation	4
Phenol—Benzoxazolone bioisosteres: Synthesis and biological evaluation of tricyclic GluN2B‐selective N‐methyl‐d‐aspartate receptor antagonists	4
Discovery of novel triazolophthalazine derivatives as DNA intercalators and topoisomerase II inhibitors	4
Hybridization‐based design of novel anticholinesterase indanone–carbamates for Alzheimer's disease: Synthesis, biological evaluation, and docking studies	4
In silico characterization of ligand–receptor interactions for U‐47700, N,N‐didesmethyl‐U‐47700, U‐50488 at mu‐ and kappa‐opioid receptors	4
Soft drug inhibitors for the epigenetic targets lysine‐specific demethylase 1 and histone deacetylases	4
Pharmacophore‐based, rationale design, and efficient synthesis of novel tetrahydrobenzo[b]thiophene candidates as potential dual Topo I/II inhibitors and DNA intercalators	4
Novel hydrazide‐hydrazone containing 1,2,4‐triazole as potent inhibitors of antiapoptotic protein Bcl‐xL: Synthesis, biological evaluation, and docking studies	4
Exosomal miR‐122, miR‐128, miR‐200, miR‐298, and miR‐342 as novel diagnostic biomarkers in NAFL/NASH: Impact of LPS/TLR‐4/FoxO3 pathway	4