Journal of Labelled Compounds & Radiopharmaceuticals

Article	Citations
Use of radioiodine in nuclear medicine—A brief overview	23
Radiosynthesis and quality control testing of the tau imaging positron emission tomography tracer [18F]PM‐PBB3 for clinical applications	16
Radioiodination of balsalazide, bioevaluation, and characterization as a highly selective radiotracer for imaging of ulcerative colitis in mice	13
Production of [89Zr]Oxinate4 and cell radiolabeling for human use	12
Automated radiosynthesis of [68Ga]Ga‐PSMA‐11 and [177Lu]Lu‐PSMA‐617 on the iPHASE MultiSyn module for clinical applications	11
Fully automated production of the fibroblast activation protein radiotracer [18F]FAPI‐74	8
Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier	8
Copper‐mediated radioiodination reaction through aryl boronic acid or ester precursor and its application to direct radiolabeling of a cyclic peptide	7
Review: Self‐radiolysis of compounds containing tritium and carbon‐14	7
Polyethylene oxide–polyacrylic acid–folic acid (PEO‐PAAc) nanogel as a99mTc targeting receptor for cancer diagnostic imaging	7
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	6
Development of an automated production process of [64Cu][Cu (ATSM)] for positron emission tomography imaging and theranostic applications	6
Peptides for trans‐blood–brain barrier delivery	6
Evaluating N‐difluoromethyltriazolium triflate as a precursor for the synthesis of high molar activity [18F]fluoroform	5
Preclinical evaluation of anti‐VEGFR2 monoclonal antibody ramucirumab labelled with zirconium‐89 for tumour imaging	5
Synthesis of deuterium‐labeled cinnamic acids: Understanding the volatile benzenoid pathway in the flowers of the Japanese loquat Eriobotrya japonica	4
Preparation, Characterization, and Radiolabeling of Anti‐HER2 scFv With Technetium Tricarbonyl and Stability Studies	4
Detailed radiosynthesis of [18F]mG4P027 as a positron emission tomography radiotracer for mGluR4	4
The impact of radiochemistry in drug projects: The use of C‐14 label in the AZD8529, AZD7325, and AZD6280 projects	4
Carbon‐11 carboxylation of terminal alkynes with [11C]CO2	4
Synthesis and automated fluorine‐18 radiolabeling of new PSMA‐617 derivatives with a CuAAC radiosynthetic approach	4
Synthesis of [H‐3]‐ and [C‐14]‐labeled elagolix	4
Synthesis of [13C6]‐ibrutinib	3
An improved one‐pot preparation of [18F]FMISO based on solid phase extraction purification: Pitfalls on the analytical method reported in the Ph.Eur.'s monograph	3
Automated radiosynthesis of 1‐(2‐[18F]fluoroethyl)‐L‐tryptophan ([18F]FETrp) for positron emission tomography (PET) imaging of cancer in humans	3

Development of a novel [18F]fluorobenzyl derivative of the AT1 receptor antagonist Candesartan	3
Synthesis of 13C‐labelled cutin and suberin monomeric dicarboxylic acids of the general formula HO213C‐(CH2)n‐13CO2H (n<	3
Synthesis and analysis of isotopically stable labeled nitrosamines as mass spectrometry standards for drug impurity quality control	3
A practical and environmentally friendly protocol for synthesis of α‐deuterated carboxylic acids	3
Exploration of alcohol‐enhanced Cu‐mediated radiofluorination toward practical labeling	3
Carbon 14 synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	3
Comparison of three different methods in [68Ga]Ga‐PSMA11 radiolabeling	3
Isotopically labelled compounds in research projects of life sciences	3
Highly selective catalytic transfer hydrodeuteration of cyclic alkenes	3
Luminescence enhancement by deuterium	3
The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier	3
Development of radiotracers for riboflavin transporter 3 imaging in diseases—A brief overview	2
Improved protocol for the radiosynthesis of [18F]FTC‐146: A potent and selective sigma‐1 receptor radioligand	2
Synthesis of [2H5]baricitinib via [2H5]ethanesulfonyl chloride	2
Preparation, quality control, and biodistribution assessment of [111In]In‐DOTA‐PR81 in BALB/c mice bearing breast tumors	2
An updated synthesis of N1′‐([11C]methyl)naltrindole for positron emission tomography imaging of the delta opioid receptor	2
Development and physicochemical characterization of a biodegradable microspheres formulation loaded with samarium‐153 and doxorubicin for chemo‐radioembolization of liver tumours	2
Fluorine‐18 labeled aldehydes as prosthetic groups for oxime coupling with a FVIIa protein	2
Copper‐mediated nucleophilic radiofluorination of [18F]β‐CFT for positron emission tomography imaging of dopamine transporter	2
Automated radiosynthesis of [11C]MTP38—a phosphodiesterase 7 imaging tracer—using [11C]hydrogen cyanide for clinical applications	2
Synthesis of a dual carbon‐14‐labeled calcitonin gene‐related peptide receptor antagonist for use in a human absorption–distribution–metabolism–elimination study	2
An optimized radiosynthesis of [18F]DK222, a PET radiotracer for imaging PD‐L1	2
Radiosynthesis of 3H‐ and 14C‐labeled Veliparib	2
Good manufacturing procedure production of [18F]SynVesT‐1, a radioligand for in vivo positron emission tomography imaging of synaptic vesicle glycoprotein 2A	2
Novel developed HPLC analyses of [68Ga]Ga/[177Lu]Lu‐EDTMP and [68Ga]Ga/[177Lu]Lu‐DOTA‐Zoledronate	2
An efficient and general method for the synthesis of stable isotope deuterium labeled phthalate esters	2
Process validation, current good manufacturing practice production, dosimetry, and toxicity studies of the carbonic anhydrase IX imaging agent [111In]In‐XYIMSR‐01 for phase I regulatory app	2
Development of a 68Ga‐labelled PET tracer for carbonic anhydrase IX‐overexpressed tumors using the artificial sweetener saccharin	2
Benzylic deuteration of alkylnitroaromatics via amine‐base catalysed exchange with deuterium oxide	2
Enzymatic synthesis of halogen derivatives of L‐phenylalanine and phenylpyruvic acid stereoselectively labeled with hydrogen isotopes in the side chain	2
High‐yield synthesis of a tau PET radioligand and its nonradioactive ligand using an alternative protection and deprotection strategy	2
Automated synthesis of (R)‐[18F]MH.MZ on the iPhase Flexlab reaction platform	2
Automated radiosynthesis of the adenosine A2A receptor‐targeting radiotracer [18F]FLUDA	2
Exploring the enzyme‐catalyzed synthesis of isotope labeled cyclopropanes	1
The impact of zirconium‐89 solution formulation on the efficiency of [89Zr]Zr‐deferoxamine synthesis	1
Synthesis and radiolabeling of a polar [125I]I‐1,2,4,5‐tetrazine	1
RO6807936 as a novel positron emission tomography (PET) radiotracer for in vitro and in vivo visualization and quantification of beta‐site amyloid precursor protein cleaving enzyme (BACE1) in the rode	1
The synthesis of deuteriated tri‐tert‐butyl phosphine	1
Low‐scale syringe‐made synthesis of 15N‐labeled oligonucleotides	1
Automated radiochemical synthesis of pharmaceutical grade [18F]FLT using 3‐N‐Boc‐5′‐O‐dimethoxytrityl‐3′‐O‐nosyl‐thymidine precursor and its Sep‐Pak® purification employing selective elutio	1
Efficient synthesis of carbon‐14 labeled metabolites of the strobilurin fungicide mandestrobin using biomimetic iron‐porphyrin catalyzed oxidation	1
A comparative study on Suzuki‐type 11C‐methylation of aromatic organoboranes performed in two reaction media	1
Synthesis of [4S‐2H]NADH, [4R‐2H]NADH, [4‐2H2]NADH and [4‐2H]NAD+ cofactors through heterogeneous biocatalysis in heavy	1
Preliminary PET imaging of [11C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated 11C‐car	1
Ultra‐fast liquid chromatography method coupled with ultraviolet detection to quantify dimethylsulfoxide, dimethylformamide and dimethylacetamide in short half‐lives radiopharmaceuticals	1
Synthesis of tritium labeled 30‐KDa PEG and conjugation to form [3H]Pegbelfermin	1
Site‐specifically radiolabeled nanobodies for imaging blood‐brain barrier penetration and targeting in the brain	1
Small‐scale two‐dimensional liquid chromatography for a preparative re‐purification of a highly labile tritium‐labeled compound	1
[18F]Fluoropyridine‐losartan: A new approach toward human Positron Emission Tomography imaging of Angiotensin II Type 1 receptors	1
Issue Information	1

Research on preparation and in vitro evaluation of the dendrimer–peptide nuclear acid conjugate for amplification pretargeting	1
Mild and selective hydrogen–deuterium exchange for aromatic hydrogen of amines	1
Tritium hydrogen‐isotope exchange with electron‐poor tertiary benzenesulfonamide moiety; application in late‐stage labeling of T0901317	1
Determination of isotope abundance for deuterium‐labeled compounds by quantitative 1H NMR + 2H NMR	1
An Improved HPLC Separation Method for TSPO Radioligand [11C]ER176 Clinical Production	1
Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET	1
Fully Automated Cassette‐Based Synthesis of 2‐Deoxy‐2‐[18F]Fluorocellobiose Using Trasis AllInOne Module	1
In vivo and in vitro binding of [125I]I‐R‐(+)‐TISCH: A dopamine D1 receptor ligand for studying pancreatic β‐cell mass	1
A facile synthesis of isotope labeled acylcarnitines	1
An improved synthesis of [18F]VAT and its precursor	1
Preparation and biological evaluation of radioiodine‐labeled triphenylphosphine derivatives as mitochondrial targeting probes	1
Synthesis of 13C‐labeled parabens from isotopically enriched phenols using the Houben–Hoesch reaction	1
Total synthesis of [13C2]‐labeled phytosiderophores of the mugineic and avenic acid families	1
Highly effective liquid and solid phase extraction methods to concentrate radioiodine isotopes for radioiodination chemistry	1
Radiosynthesis and validation of [18F]fluoroestradiol in a Synthra plus research platform for use in routine clinical practice	1
Synthesis of beta‐site amyloid precursor protein‐cleaving enzyme 1 inhibitors BI 1147560 and BI 1181181 labeled with carbon‐14 and deuterium	1
Practical approaches to labelling terminal alkynes with deuterium	0
Synthesis of carbon‐14 and stable isotope labeled Censavudine	0
Issue Information	0
Issue Information	0
Issue Information	0
Synthesis of Radiolabeled [14C]Rimsulfuron and Stable Isotope Labeled Rimsulfuron‐[M + 3] to Support Crop Metabolism Studies for Reregistration	0
	0
Issue Information	0
Nitrilase mediated mild hydrolysis of a carbon‐14 nitrile for the radiosynthesis of 4‐(7‐hydroxycarbamoyl‐[1‐14C‐heptanoyl]‐oxy)‐benzoic acid methyl ester, [14C]‐SHP‐141: A novel	0
Featured Cover	0
Synthesis of deuterium‐labeled CCR2 antagonist JNJ‐26131300, [4‐(1H‐indol‐ 3‐yl)‐piperidin‐1‐yl]‐{1‐[3‐(3,4,5‐trifluoro‐phenyl)‐acryloyl]‐piperidin‐4‐yl}‐acetic acid	0
	0
	0
Issue Information	0
Issue Information	0
Issue Information	0
Meet our Special Issue Editor: Jessica Bridoux	0
Next Generation of Solid Target Radionuclide Antibody Conjugates for Tumor Immuno‐Therapy	0
	0
	0
Issue Information	0
Issue Information	0
Issue Information	0
	0
Issue Information	0
Issue Information	0
Wiley Young Scientist Awards were handed over at the 14th International Symposium on the synthesis on the Synthesis and Applications of Isotopically Labelled Compounds in Raleigh, USA	0
	0
Efficient Reductive N‐11C‐Methylation Using Arylamines or Alkylamines and In Situ–Generated [11C]Formaldehyde From [11C]Methyl Iodide	0
Issue Information	0
	0
	0
	0
18F‐Fluorination of a supported 2‐(aryl‐di‐tert‐butylsilyl)‐N‐methyl‐imidazole for indirect 18F‐labeling of a VHH single‐variable domain	0
Issue Information	0
	0
Synthesis and preclinical evaluation of a selective MET kinase positron emission tomography tracer	0
Issue Information	0
	0
Meet our advisors: Crist N. Filer	0
Meet the advisors: An interview with Gunnar Antoni	0
Imidazolium‐methylene‐trifluoroborate: A novel radioprosthetic group validated with preclinical 18F‐Positron Emission Tomography imaging of Prostate Specific Membrane Antigen in mice	0
	0
Carbon 14 and stable isotope synthesis of two potent and selective phosphodiesterase type 4 inhibitors	0
	0
	0
Issue Information	0
	0
Development of 11C‐labeled CRANAD‐102 for positron emission tomography imaging of soluble Aβ‐species	0
Preparation of [1′‐13C]citric acid as a probe in a breath test to evaluate tricarboxylic acid cycle flux	0
	0
	0
Obituary	0
	0
Carbon‐14 Labeling Synthesis of RORγt Inhibitor JNJ‐61803534	0
Issue Information	0
High‐yielding, automated radiosynthesis of [11C]martinostat using [11C]methyl triflate	0
Issue Information	0
Issue Information	0
14C‐radiolabeling of a new steroidal antiandrogen with a C‐18 angular methyl extension	0
A simplified protocol for the automated production of 2‐[18F]fluoro‐3‐[2‐((S)‐3‐pyrrolinyl)methoxy]pyridine ([18F]nifene) on an IBA Synthera® module	0
	0
Issue Information	0
	0

Automated radiosynthesis of [18F]CETO, a PET radiotracer for imaging adrenal glands, on Synthra RNplus	0
Applications of radiolabeled antibodies in neuroscience and neuro‐oncology	0
Meet our advisors: Bill Lockley	0
	0
An improved radiosynthesis of [18F]FAraG, a PET radiotracer for imaging T‐cell activation	0
Synthesis of trifold‐labeled versatile reagent [3,5‐13C2,4‐15 N]4‐phenyl‐1,2,4‐triazoline‐3,5‐dione	0
	0
	0
Novel synthesis of 11C‐labeled imidazolines via Pd(0)‐mediated 11C‐carbomethoxylation using [11C]CO and arylborons	0
Meet our advisors: Jordi Llop	0
Issue Information	0
	0
Initial evaluation of 99mTc‐labeled anti‐carcinoembryonic antigen single‐chain fragment variable for micro‐single‐photon emission computed tomography imaging in mice with colorectal cancer	0
Issue Information	0
Direct Multi‐Deuterium Labelling of Pirtobrutinib	0
Issue Information	0
Issue Information	0
	0
Development of a high‐performance liquid chromatography method for rapid radiochemical purity measurement of [18F]PSMA‐1007, a PET radiopharmaceutical for detection of prostate cancer	0
Issue Information	0
Carbon 14 and Carbon 13 Syntheses of Velagliflozin	0
	0
Synthesis of N‐acetyl‐l‐aspartyl‐l‐glutamic acid; [3H]NAAG	0
A flow electrochemistry‐enabled synthesis of 2‐substituted N‐(methyl‐d)piperidines	0
Synthesis of [3H]Org24598 using in‐house prepared [3H]MeI	0
	0
	0
Issue Information	0
	0
	0
Meet our advisors: Neil Vasdev	0
Meet the advisors ‐ Suzy Lapi	0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
	0
Meet our advisors—Matteo Zanda	0
Issue Information	0
	0
Improved Radiosynthesis and Automation of [11C]2‐(2,6‐Difluoro‐4‐((2‐(N‐methylphenylsulfonamido)ethyl)thio)phenoxy)acetamide ([11C]K2) for Positron Emission Tomography of	0
Issue Information	0
	0
68Ga Radiolabeling of NODASA‐Functionalized Phage Display–Derived Peptides for Prospective Assessment as Tuberculosis‐Specific PET Radiotracers	0
	0
Meet our advisors: Dieter Muri	0
	0
Issue Information	0
Issue Information	0
Open‐source flow setup for rapid and efficient [18F]fluoride drying for automation of PET tracer syntheses	0
	0
Improving Routine 89Zr‐Immuno‐PET Applications: Mild Iron Removal Can Favor the Use of Fe‐DFO‐N‐suc‐TFP Ester Over p‐NCS‐Bz‐DFO	0
Synthesis of Stable Isotope, Tritiated, and Carbon‐14 Labeled Balcinrenone	0
Facile synthesis of 14C‐nitrofurazone from 14C‐urea	0
Issue Information	0
Preparation and evaluation of radiolabeled acetaminosalol microspheres: A new potential selective radiotracer for ulcerative colitis early diagnosis	0
Synthesis of Deuterated Endochin‐Like Quinolones	0
A facile synthesis of precursor for the σ‐1 receptor PET radioligand [18F]FTC‐146 and its radiofluorination	0
Issue Information	0
	0
Meet our advisors: Mathew Thakur	0
Issue Information	0
Synthesis and Application of D‐ and 13C‐Labelled tert‐Butyl Hoechst Dye	0
Issue Information	0
Validation of a good manufacturing practice procedure for the production of [11C]AZD4747, a CNS penetrant KRASG12c inhibitor	0
Formulation of patient dose of [177Lu]Lu‐Trastuzumab using in‐house developed freeze‐dried kit: A path forward for clinical translation	0
Photocatalyzed radiosynthesis of 11C‐phenylacetic acids	0
Abstracts From the 29th International Isotope Society UK Meeting 17th November 2023	0
Issue Information	0
A synthesis of [14C]formamidine acetate	0
	0
Stable isotope synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	0
Issue Information	0
Preclinical evaluation of [11C]L‐235 as a radioligand for Positron Emission Tomography cathepsin K imaging in bone	0
Issue Information	0
Synthesis of BI 894416 and BI 1342561, two potent and selective spleen tyrosine kinase inhibitors, labeled with carbon 14 and with deuterium	0
	0
Issue Information	0
Issue Information	0
	0
Issue Information	0
	0
Synthesis and spectroscopic characterization of 13C4‐labeled 4‐cyano‐2‐oxobutyraldehyde semicarbazone: A metabolite of nitrofurazone	0
	0
	0
Issue Information	0
Carbon‐13 labeling of ibrutinib for human microdosing	0
Meet our advisors: Bart Cornelissen	0
Synthesis and Preclinical Evaluation of [18F]AlF‐NOTA‐Asp2‐PEG2‐Folate as a Novel Folate‐Receptor‐Targeted Tracer for PET Imaging	0
	0
Evaluation and improvement of CuI‐mediated 11C‐cyanation	0
Synthesis of 13C‐labelled ω‐hydroxy carboxylic acids of the general formula HO213C‐(CH2)n‐CH2OH or HO2C‐(CH2	0
Automated radiolabeling and handling of 177Lu‐ and 225Ac‐PSMA‐617 using a robotic pipettor	0
Issue Information	0
[11C]CO2 BOP fixation with amines to access 11C‐labeled ureas for PET imaging	0
[18F]‐labeled positron emission tomography ligand for the histamine H4 receptor	0
Issue Information	0
	0