Journal of Labelled Compounds & Radiopharmaceuticals

Papers
(The median citation count of Journal of Labelled Compounds & Radiopharmaceuticals is 0. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-06-01 to 2025-06-01.)
ArticleCitations
Meet our advisors: Crist N. Filer17
Issue Information16
Issue Information11
9
9
Issue Information8
Automated radiolabeling and handling of 177Lu‐ and 225Ac‐PSMA‐617 using a robotic pipettor7
A flow electrochemistry‐enabled synthesis of 2‐substituted N‐(methyl‐d)piperidines6
6
Issue Information6
5
5
Radiosynthesis and Evaluation of [18F]FEHSP990 as Novel PET Tracer for Hsp90 PET Imaging5
5
Radiosynthesis of 3H‐ and 14C‐labeled Veliparib4
4
Small‐scale two‐dimensional liquid chromatography for a preparative re‐purification of a highly labile tritium‐labeled compound4
Applications of radiolabeled antibodies in neuroscience and neuro‐oncology4
4
Luminescence enhancement by deuterium4
Synthesis of deuterium‐labeled cinnamic acids: Understanding the volatile benzenoid pathway in the flowers of the Japanese loquat Eriobotrya japonica4
4
Issue Information3
Issue Information3
Synthesis of Carbon 14 and Deuterium‐Labelled Nerandomilast (BI 1015550)3
Carbon‐14 Labeling Synthesis of RORγt Inhibitor JNJ‐618035343
Fully Automated Cassette‐Based Synthesis of 2‐Deoxy‐2‐[18F]Fluorocellobiose Using Trasis AllInOne Module3
Issue Information3
Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET3
Synthesis and Characterization of 3‐Hydroxybupivacaine and Deuterated 3‐Hydroxybupivacaine for Use in Equine Medication Regulation3
Issue Information3
3
An efficient and general method for the synthesis of stable isotope deuterium labeled phthalate esters3
68Ga Radiolabeling of NODASA‐Functionalized Phage Display–Derived Peptides for Prospective Assessment as Tuberculosis‐Specific PET Radiotracers3
2
A comparative study on Suzuki‐type 11C‐methylation of aromatic organoboranes performed in two reaction media2
Photocatalyzed radiosynthesis of 11C‐phenylacetic acids2
[18F]Fluoropyridine‐losartan: A new approach toward human Positron Emission Tomography imaging of Angiotensin II Type 1 receptors2
11C‐Carbonylation for PET Imaging and Drug Discovery2
Tritium and deuterium labelling of a kainate receptor antagonist and evaluation as a radioligand2
Meet our advisors: Neil Vasdev2
Novel developed HPLC analyses of [68Ga]Ga/[177Lu]Lu‐EDTMP and [68Ga]Ga/[177Lu]Lu‐DOTA‐Zoledronate2
Total synthesis of [13C2]‐labeled phytosiderophores of the mugineic and avenic acid families2
Low‐scale syringe‐made synthesis of 15N‐labeled oligonucleotides2
2
Carbon 14 and stable isotope synthesis of two potent and selective phosphodiesterase type 4 inhibitors2
Application of Microfluidic Devices for Automated Two‐Step Radiolabeling of Antibodies2
2
Issue Information2
RO6807936 as a novel positron emission tomography (PET) radiotracer for in vitro and in vivo visualization and quantification of beta‐site amyloid precursor protein cleaving enzyme (BACE1) in the rode2
Synthesis of BI 894416 and BI 1342561, two potent and selective spleen tyrosine kinase inhibitors, labeled with carbon 14 and with deuterium2
Preliminary Research of Radiolabeled Atezolizumab for the Noninvasive Evaluation of TNBC PD‐L1 Expression In Vivo2
Meet our Special Issue Editor: Jessica Bridoux2
Issue Information1
Obituary1
Issue Information1
Issue Information1
Formulation of patient dose of [177Lu]Lu‐Trastuzumab using in‐house developed freeze‐dried kit: A path forward for clinical translation1
1
Practical approaches to labelling terminal alkynes with deuterium1
Automated synthesis of (R)‐[18F]MH.MZ on the iPhase Flexlab reaction platform1
Ultrasound‐Assisted Microcontinuous Process Facilitates the Selective Deuteration of Steroid Hormones1
Synthesis and Preclinical Evaluation of Peptide Dimer‐Based PET Tracers for Imaging VEGFR‐2 Expression in Tumors1
Issue Information1
Meet our advisors: Dieter Muri1
Automated radiosynthesis of [18F]CETO, a PET radiotracer for imaging adrenal glands, on Synthra RNplus1
Initial evaluation of 99mTc‐labeled anti‐carcinoembryonic antigen single‐chain fragment variable for micro‐single‐photon emission computed tomography imaging in mice with colorectal cancer1
Issue Information1
1
Issue Information1
Synthesis and preclinical evaluation of a selective MET kinase positron emission tomography tracer1
Synthesis of 14C‐Labeled Polyethylene Terephthalate and Generation of 14C‐Nanoparticles for Fate and Disposition Studies1
Issue Information1
Automated radiochemical synthesis of pharmaceutical grade [18F]FLT using 3‐N‐Boc‐5′‐O‐dimethoxytrityl‐3′‐O‐nosyl‐thymidine precursor and its Sep‐Pak® purification employing selective elutio1
Issue Information1
Automated radiosynthesis of mGluR5 PET tracer [18F]FPEB from aryl‐chloro precursor and validation for clinical application1
14C‐radiolabeling of a new steroidal antiandrogen with a C‐18 angular methyl extension1
1
Nitrilase mediated mild hydrolysis of a carbon‐14 nitrile for the radiosynthesis of 4‐(7‐hydroxycarbamoyl‐[1‐14C‐heptanoyl]‐oxy)‐benzoic acid methyl ester, [14C]‐SHP‐141: A novel1
Targeting VEGF With 99mTc‐Labeled Ranibizumab for Noninvasive Diagnosis of Non‐Small Cell Lung Cancer1
1
High‐yielding, automated radiosynthesis of [11C]martinostat using [11C]methyl triflate1
Determination of isotope abundance for deuterium‐labeled compounds by quantitative 1H NMR + 2H NMR1
1
Issue Information1
Meet our advisors: Bart Cornelissen1
Good manufacturing procedure production of [18F]SynVesT‐1, a radioligand for in vivo positron emission tomography imaging of synaptic vesicle glycoprotein 2A1
Improving Routine 89Zr‐Immuno‐PET Applications: Mild Iron Removal Can Favor the Use of Fe‐DFO‐N‐suc‐TFP Ester Over p‐NCS‐Bz‐DFO1
Lead‐212/Bismuth‐212 In Vivo Generator Based on Ultrasmall Silver Telluride Nanoparticles1
Synthesis and spectroscopic characterization of 13C4‐labeled 4‐cyano‐2‐oxobutyraldehyde semicarbazone: A metabolite of nitrofurazone1
1
Issue Information0
0
Issue Information0
Issue Information0
Issue Information0
Synthesis and Preclinical Evaluation of [18F]AlF‐NOTA‐Asp2‐PEG2‐Folate as a Novel Folate‐Receptor‐Targeted Tracer for PET Imaging0
Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier0
The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier0
Synthesis and Application of D‐ and 13C‐Labelled tert‐Butyl Hoechst Dye0
Preparation and evaluation of radiolabeled acetaminosalol microspheres: A new potential selective radiotracer for ulcerative colitis early diagnosis0
Issue Information0
Preparation of Macrobicyclic Cryptands for Radiometal Complexation0
[18F]‐labeled positron emission tomography ligand for the histamine H4 receptor0
0
Automated radiosynthesis of the adenosine A2A receptor‐targeting radiotracer [18F]FLUDA0
0
Issue Information0
Evaluation and improvement of CuI‐mediated 11C‐cyanation0
Improved protocol for the radiosynthesis of [18F]FTC‐146: A potent and selective sigma‐1 receptor radioligand0
Detailed radiosynthesis of [18F]mG4P027 as a positron emission tomography radiotracer for mGluR40
Development of an automated production process of [64Cu][Cu (ATSM)] for positron emission tomography imaging and theranostic applications0
Synthesis of Deuterated Endochin‐Like Quinolones0
0
0
Meet our advisors: Bill Lockley0
Simplified Flow Photosynthesis of Deuterium‐Labeled Pyocyanin0
Comparison of three different methods in [68Ga]Ga‐PSMA11 radiolabeling0
Stable isotope synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites0
A Brief Review of Radiolabelling Nucleic Acid‐Based Molecules for Tracking and Monitoring0
Open‐source flow setup for rapid and efficient [18F]fluoride drying for automation of PET tracer syntheses0
Issue Information0
Synthesis of 13C‐labelled ω‐hydroxy carboxylic acids of the general formula HO213C‐(CH2)n‐CH2OH or HO2C‐(CH20
Issue Information0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system0
Synthesis of 13C‐labeled parabens from isotopically enriched phenols using the Houben–Hoesch reaction0
Issue Information0
Synthesis and automated fluorine‐18 radiolabeling of new PSMA‐617 derivatives with a CuAAC radiosynthetic approach0
Radiosynthesis and validation of [18F]fluoroestradiol in a Synthra plus research platform for use in routine clinical practice0
0
A practical protocol for large‐scale copper‐mediated radioiodination of organoboronic precursors: Radiosynthesis of [123I]KX‐1 for Auger radiotherapy0
Preparation of [1′‐13C]citric acid as a probe in a breath test to evaluate tricarboxylic acid cycle flux0
Featured Cover0
A Novel 68Ga‐Labeled 2‐Azabicyclo[3.1.0]Hexane‐3‐Carbonitrile‐Based Fibroblast Activation Protein‐Targeted Tracer for Cancer Imaging With Positron Emission Tomography0
0
Issue Information0
Issue Information0
Peptides for trans‐blood–brain barrier delivery0
0
0
Synthesis of [13C6]‐ibrutinib0
Improved Radiosynthesis and Automation of [11C]2‐(2,6‐Difluoro‐4‐((2‐(N‐methylphenylsulfonamido)ethyl)thio)phenoxy)acetamide ([11C]K2) for Positron Emission Tomography of 0
Issue Information0
Issue Information0
A simplified protocol for the automated production of 2‐[18F]fluoro‐3‐[2‐((S)‐3‐pyrrolinyl)methoxy]pyridine ([18F]nifene) on an IBA Synthera® module0
Meet the editors: Danielle Vugts0
0
Issue Information0
An improved synthesis of [18F]VAT and its precursor0
Radiolabeling and brain penetration of [11C]VU0071063, a ligand of type 1 sulfonylurea receptors for positron emission tomography imaging0
Design and Synthesis of a 18F‐Radiolabeled Pyrrolo[2,3‐d]pyrimidine Ligand as a CSF1R Receptor PET Imaging Agent0
Exploring the enzyme‐catalyzed synthesis of isotope labeled cyclopropanes0
Correction to Validation of a Good Manufacturing Practice Procedure for the Production of [11C]AZD4747, a CNS Penetrant KRASG12c Inhibitor0
Synthesis of trifold‐labeled versatile reagent [3,5‐13C2,4‐15 N]4‐phenyl‐1,2,4‐triazoline‐3,5‐dione0
0
Development of radiotracers for riboflavin transporter 3 imaging in diseases—A brief overview0
Issue Information0
Synthesis and Imaging of Novel CDK19‐Targeted Tracers Incorporating an Albumin‐Binding Moiety0
An improved radiosynthesis of [18F]FAraG, a PET radiotracer for imaging T‐cell activation0
Synthesis and analysis of isotopically stable labeled nitrosamines as mass spectrometry standards for drug impurity quality control0
Ultra‐fast liquid chromatography method coupled with ultraviolet detection to quantify dimethylsulfoxide, dimethylformamide and dimethylacetamide in short half‐lives radiopharmaceuticals0
Automated radiosynthesis of [11C]MTP38—a phosphodiesterase 7 imaging tracer—using [11C]hydrogen cyanide for clinical applications0
Development of a high‐performance liquid chromatography method for rapid radiochemical purity measurement of [18F]PSMA‐1007, a PET radiopharmaceutical for detection of prostate cancer0
Synthesis of [2H5]baricitinib via [2H5]ethanesulfonyl chloride0
Evaluating N‐difluoromethyltriazolium triflate as a precursor for the synthesis of high molar activity [18F]fluoroform0
Issue Information0
Synthesis of Stable Isotope, Tritiated, and Carbon‐14 Labeled Balcinrenone0
0
Current Advances in PARP1‐Targeted Theranostics0
0
0
Towards Optimal Automated 68Ga‐Radiolabeling Conditions of the DOTA‐Bisphosphonate BPAMD Without Pre‐Purification of the Generator Eluate0
Tritium hydrogen‐isotope exchange with electron‐poor tertiary benzenesulfonamide moiety; application in late‐stage labeling of T09013170
The synthesis of deuteriated tri‐tert‐butyl phosphine0
0
Abstracts From the 29th International Isotope Society UK Meeting 17th November 20230
Meet our advisors: Jordi Llop0
Mild and selective hydrogen–deuterium exchange for aromatic hydrogen of amines0
Meet the editorial staff—Interview series0
Synthesis of tritium labeled 30‐KDa PEG and conjugation to form [3H]Pegbelfermin0
Development of an economical method to synthesize O‐(2‐[18F]fluoroethyl)‐L‐tyrosine (18FFET)0
Issue Information0
0
A practical and environmentally friendly protocol for synthesis of α‐deuterated carboxylic acids0
0
0
Enzymatic synthesis of halogen derivatives of L‐phenylalanine and phenylpyruvic acid stereoselectively labeled with hydrogen isotopes in the side chain0
Issue Information0
Issue Information0
Imidazolium‐methylene‐trifluoroborate: A novel radioprosthetic group validated with preclinical 18F‐Positron Emission Tomography imaging of Prostate Specific Membrane Antigen in mice0
An Improved HPLC Separation Method for TSPO Radioligand [11C]ER176 Clinical Production0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system0
Synthesis of deuterium‐labeled CCR2 antagonist JNJ‐26131300, [4‐(1H‐indol‐ 3‐yl)‐piperidin‐1‐yl]‐{1‐[3‐(3,4,5‐trifluoro‐phenyl)‐acryloyl]‐piperidin‐4‐yl}‐acetic acid0
[11C]CO2 BOP fixation with amines to access 11C‐labeled ureas for PET imaging0
Issue Information0
0
0
The impact of zirconium‐89 solution formulation on the efficiency of [89Zr]Zr‐deferoxamine synthesis0
Meet the advisors ‐ Suzy Lapi0
Issue Information0
Meet our advisors: An interview with John Katzenellenbogen0
Validation of a good manufacturing practice procedure for the production of [11C]AZD4747, a CNS penetrant KRASG12c inhibitor0
A synthesis of [14C]formamidine acetate0
Carbon 14 synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites0
Synthesis and evaluation of 111In‐labeled tetrapeptide‐based compounds as single‐photon emission computed tomography imaging probes targeting granzyme B0
Preliminary PET imaging of [11C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated 11C‐car0
Carbon 14 and Carbon 13 Syntheses of Velagliflozin0
Automated Radiolabeling and Evaluation of [18F]FPMBBG: A Novel Cardiac Neuronal PET Imaging Agent0
Next Generation of Solid Target Radionuclide Antibody Conjugates for Tumor Immuno‐Therapy0
Synthesis of 18F‐Labeled FC‐119S and Its Tosyl Precursor0
18F‐Fluorination of a supported 2‐(aryl‐di‐tert‐butylsilyl)‐N‐methyl‐imidazole for indirect 18F‐labeling of a VHH single‐variable domain0
0
0
Automated radiosynthesis of 1‐(2‐[18F]fluoroethyl)‐L‐tryptophan ([18F]FETrp) for positron emission tomography (PET) imaging of cancer in humans0
Issue Information0
Synthesis of beta‐site amyloid precursor protein‐cleaving enzyme 1 inhibitors BI 1147560 and BI 1181181 labeled with carbon‐14 and deuterium0
Novel synthesis of 11C‐labeled imidazolines via Pd(0)‐mediated 11C‐carbomethoxylation using [11C]CO and arylborons0
0
Issue Information0
Development and Validation of an HPLC Method to Determine Chemical and Radiochemical Purity of [18F]Florbetazine Injection0
0
[68Ga]Ga‐PentixaFor: Development of a fully automated in hospital production on the Trasis miniAllinOne synthesizer0
Highly effective liquid and solid phase extraction methods to concentrate radioiodine isotopes for radioiodination chemistry0
0
Issue Information0
Issue Information0
Direct Multi‐Deuterium Labelling of Pirtobrutinib0
Development of 11C‐labeled CRANAD‐102 for positron emission tomography imaging of soluble Aβ‐species0
Synthesis of Radiolabeled [14C]Rimsulfuron and Stable Isotope Labeled Rimsulfuron‐[M + 3] to Support Crop Metabolism Studies for Reregistration0
Issue Information0
Meet our advisors: Mathew Thakur0
Issue Information0
Synthesis and Evaluation of a Cathepsin B–Recognizing Trifunctional Chelating Agent to Improve Tumor Retention of Radioimmunoconjugates0
Meet our advisors—Matteo Zanda0
Synthesis of [3H]Org24598 using in‐house prepared [3H]MeI0
Carbon‐13 labeling of ibrutinib for human microdosing0
Efficient Reductive N11C‐Methylation Using Arylamines or Alkylamines and In Situ–Generated [11C]Formaldehyde From [11C]Methyl Iodide0
Issue Information0
Synthesis of a Potent Bruton's Tyrosine Kinase Inhibitor Labelled With Carbon‐14 and Deuterium0
Radioiodination, purification, and evaluation of antihuman tumor‐derived immunoglobulin G light chain monoclonal antibody in tumor‐bearing nude mice0
Meet our advisors: Billy Kerr0
Efficient synthesis of carbon‐14 labeled metabolites of the strobilurin fungicide mandestrobin using biomimetic iron‐porphyrin catalyzed oxidation0
Issue Information0
0
Wiley Young Scientist Awards were handed over at the 14th International Symposium on the synthesis on the Synthesis and Applications of Isotopically Labelled Compounds in Raleigh, USA0
An improved one‐pot preparation of [18F]FMISO based on solid phase extraction purification: Pitfalls on the analytical method reported in the Ph.Eur.'s monograph0
Development and physicochemical characterization of a biodegradable microspheres formulation loaded with samarium‐153 and doxorubicin for chemo‐radioembolization of liver tumours0
Synthesis, Preclinical Characterizations and Imaging Studies of [18F]AlF‐Labeled NY104, a CAIX‐Targeting Diagnostic Agent0
Synthesis of a dual carbon‐14‐labeled calcitonin gene‐related peptide receptor antagonist for use in a human absorption–distribution–metabolism–elimination study0
0
0.10663795471191