Journal of Labelled Compounds & Radiopharmaceuticals

Article	Citations
Thorium chelators for targeted alpha therapy: Rapid chelation of thorium‐226	17
Use of radioiodine in nuclear medicine—A brief overview	17
Nanoparticulate formulations of radiopharmaceuticals: Strategy to improve targeting and biodistribution properties	16
Radiosynthesis of a Bruton's tyrosine kinase inhibitor, [11C]Tolebrutinib, via palladium‐NiXantphos‐mediated carbonylation	15
Radioiodination of balsalazide, bioevaluation, and characterization as a highly selective radiotracer for imaging of ulcerative colitis in mice	13
Radiosynthesis and quality control testing of the tau imaging positron emission tomography tracer [18F]PM‐PBB3 for clinical applications	13
A 64Cu‐porphyrin‐based dual‐modal molecular probe with integrin αvβ3 targeting function for tumour imaging	13
Production of [89Zr]Oxinate4 and cell radiolabeling for human use	11
Enantioselective synthesis of tri‐deuterated (–)‐geosmin to be used as internal standard in quantitation assays	9
Production of [68Ga]Ga‐PSMA: Comparing a manual kit‐based method with a module‐based automated synthesis approach	8
Automated synthesis of 68Ga/177Lu‐PSMA on the Trasis miniAllinOne	8
Automated radiosynthesis of [68Ga]Ga‐PSMA‐11 and [177Lu]Lu‐PSMA‐617 on the iPHASE MultiSyn module for clinical applications	8
Polyethylene oxide–polyacrylic acid–folic acid (PEO‐PAAc) nanogel as a 99mTc targeting receptor for cancer diagnostic imaging	7
Fully automated production of the fibroblast activation protein radiotracer [18F]FAPI‐74	7
New synthesis of 6″‐[18F]fluoromaltotriose for positron emission tomography imaging of bacterial infection	7
A novel 99mTc‐diester complex as tumor targeting agent: Synthesis, radiolabeling, and biological distribution study	7
Positron emission tomography imaging of a novel Anxa1‐targeted peptide 18F‐Al‐NODA‐Bn‐p‐SCN‐GGGRDN‐IF7 in A431 cancer mouse models	6
A one‐pot radiosynthesis of [18F]PARPi	6
Review: Self‐radiolysis of compounds containing tritium and carbon‐14	6
Automated GMP production and long‐term experience in radiosynthesis of CB1 tracer [18F]FMPEP‐d2	6
Copper‐mediated radioiodination reaction through aryl boronic acid or ester precursor and its application to direct radiolabeling of a cyclic peptide	6
Dual‐labeled prostate‐specific membrane antigen (PSMA)‐targeting agent for preoperative molecular imaging and fluorescence‐guided surgery for prostate cancer	6
Development of an automated production process of [64Cu][Cu (ATSM)] for positron emission tomography imaging and theranostic applications	5
Development of a fully automated low‐pressure [11C]CO carbonylation apparatus	5
Arabinofuranose‐derived positron‐emission tomography radiotracers for detection of pathogenic microorganisms	5

A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	5
Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier	5
Radiolabeled (R)‐(–)‐5‐iodo‐3′‐O‐[2‐(ε‐guanidinohexanoyl)‐2‐phenylacetyl]‐2′‐deoxyuridine: A new theranostic for neuroblastoma	4
Synthesis of a deuterated 6‐AmHap internal standard for the determination of hapten density in a heroin vaccine drug product	4
Preclinical evaluation of anti‐VEGFR2 monoclonal antibody ramucirumab labelled with zirconium‐89 for tumour imaging	4
Carbon‐11 carboxylation of terminal alkynes with [11C]CO2	4
Synthesis of deuterium‐labeled cinnamic acids: Understanding the volatile benzenoid pathway in the flowers of the Japanese loquat Eriobotrya japonica	4
Evaluating N‐difluoromethyltriazolium triflate as a precursor for the synthesis of high molar activity [18F]fluoroform	4
Facile synthesis of 2‐deoxy‐2‐[18F]fluorosorbitol using sodium borohydride on aluminum oxide	3
Synthesis and analysis of isotopically stable labeled nitrosamines as mass spectrometry standards for drug impurity quality control	3
Selective synthesis of L‐2‐[18F]fluoro‐alpha‐methylphenylalanine via copper‐mediated 18F‐fluorination of (mesityl)(aryl)iodonium salt	3
Radiosynthesis, in vitro and preliminary biological evaluation of [18F]2‐amino‐4‐((2‐((3‐fluorobenzyl)oxy)benzyl)(2‐((3‐(fluoromethyl)benzyl)oxy)benzyl)amino)butanoic acid, a novel alanine	3
Synthesis of 13C‐labelled cutin and suberin monomeric dicarboxylic acids of the general formula HO213C‐(CH2)n‐13CO2H (n<	3
Synthesis of [H‐3]‐ and [C‐14]‐labeled elagolix	3
Detailed radiosynthesis of [18F]mG4P027 as a positron emission tomography radiotracer for mGluR4	3
An improved one‐pot preparation of [18F]FMISO based on solid phase extraction purification: Pitfalls on the analytical method reported in the Ph.Eur.'s monograph	3
Exploration of alcohol‐enhanced Cu‐mediated radiofluorination toward practical labeling	3
Production of the next‐generation positron nuclide zirconium‐89 (89Zr) guided by Monte Carlo simulation and its good quality for antibody labeling	3
Isotopically labelled compounds in research projects of life sciences	3
The impact of radiochemistry in drug projects: The use of C‐14 label in the AZD8529, AZD7325, and AZD6280 projects	3
Radiolabeled hormones in insulin research, a minireview	3
Iodination of CART(61‐102) peptide: Preserved binding and anorexigenic activity in mice	2
Development of an automated, GMP compliant FASTlab™ radiosynthesis of [18F]GE‐179 for the clinical study of activated NMDA receptors	2
Development of a 68Ga‐labelled PET tracer for carbonic anhydrase IX‐overexpressed tumors using the artificial sweetener saccharin	2
Carbon 14 synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	2
Radiosynthesis of 3H‐ and 14C‐labeled Veliparib	2
Synthesis of 18F‐radiolabeled organophosphine fluorides for thiol‐chemoselective peptide conjugation	2
Improved protocol for the radiosynthesis of [18F]FTC‐146: A potent and selective sigma‐1 receptor radioligand	2
S‐(4‐nitrobenzyl)‐6‐thioinosine: Tritium labelling at high specific activity	2
Automated radiosynthesis of 1‐(2‐[18F]fluoroethyl)‐L‐tryptophan ([18F]FETrp) for positron emission tomography (PET) imaging of cancer in humans	2
Enzymatic synthesis of halogen derivatives of L‐phenylalanine and phenylpyruvic acid stereoselectively labeled with hydrogen isotopes in the side chain	2
Peptides for trans‐blood–brain barrier delivery	2
High‐yield synthesis of a tau PET radioligand and its nonradioactive ligand using an alternative protection and deprotection strategy	2
Synthesis of [13C6]‐ibrutinib	2
Process validation, current good manufacturing practice production, dosimetry, and toxicity studies of the carbonic anhydrase IX imaging agent [111In]In‐XYIMSR‐01 for phase I regulatory app	2
Synthesis of isotopically labelled αCGRP8‐37 and its lipidated analogue	2
Synthesis and automated fluorine‐18 radiolabeling of new PSMA‐617 derivatives with a CuAAC radiosynthetic approach	2
Carbon‐13 synthesis and NMR spectroscopic geometric isomer evaluation to support the filing of teriflunomide	2
An updated synthesis of N1′‐([11C]methyl)naltrindole for positron emission tomography imaging of the delta opioid receptor	2
Comparison of three different methods in [68Ga]Ga‐PSMA11 radiolabeling	2
Novel developed HPLC analyses of [68Ga]Ga/[177Lu]Lu‐EDTMP and [68Ga]Ga/[177Lu]Lu‐DOTA‐Zoledronate	2
Study of the 99mTc‐labeling conditions of 6‐hydrazinonicotinamide‐conjugated peptides from a new perspective: Introduction to the term radio‐stoichiometry	2
Automated radiochemical synthesis of pharmaceutical grade [18F]FLT using 3‐N‐Boc‐5′‐O‐dimethoxytrityl‐3′‐O‐nosyl‐thymidine precursor and its Sep‐Pak® purification employing selective elutio	1
Synthesis and radiolabeling of a polar [125I]I‐1,2,4,5‐tetrazine	1
Automated radiosynthesis of the adenosine A2A receptor‐targeting radiotracer [18F]FLUDA	1
Synthesis of a dual carbon‐14‐labeled calcitonin gene‐related peptide receptor antagonist for use in a human absorption–distribution–metabolism–elimination study	1
Exploring the enzyme‐catalyzed synthesis of isotope labeled cyclopropanes	1
Development of a novel [18F]fluorobenzyl derivative of the AT1 receptor antagonist Candesartan	1
Copper‐mediated nucleophilic radiofluorination of [18F]β‐CFT for positron emission tomography imaging of dopamine transporter	1
Benzylic deuteration of alkylnitroaromatics via amine‐base catalysed exchange with deuterium oxide	1

Preparation, quality control, and biodistribution assessment of [111In]In‐DOTA‐PR81 in BALB/c mice bearing breast tumors	1
Synthesis of [4S‐2H]NADH, [4R‐2H]NADH, [4‐2H2]NADH and [4‐2H]NAD+ cofactors through heterogeneous biocatalysis in heavy	1
Determination of isotope abundance for deuterium‐labeled compounds by quantitative 1H NMR + 2H NMR	1
Ultra‐fast liquid chromatography method coupled with ultraviolet detection to quantify dimethylsulfoxide, dimethylformamide and dimethylacetamide in short half‐lives radiopharmaceuticals	1
Automated radiosynthesis of [11C]MTP38—a phosphodiesterase 7 imaging tracer—using [11C]hydrogen cyanide for clinical applications	1
Fluorine‐18 labeled aldehydes as prosthetic groups for oxime coupling with a FVIIa protein	1
The synthesis of one H‐2 labeled and two H‐3 labeled leukotriene C4 synthase inhibitors	1
Highly selective catalytic transfer hydrodeuteration of cyclic alkenes	1
An improved synthesis of [18F]VAT and its precursor	1
In vivo and in vitro binding of [125I]I‐R‐(+)‐TISCH: A dopamine D1 receptor ligand for studying pancreatic β‐cell mass	1
Low‐scale syringe‐made synthesis of 15N‐labeled oligonucleotides	1
Highly effective liquid and solid phase extraction methods to concentrate radioiodine isotopes for radioiodination chemistry	1
A comparative study on Suzuki‐type 11C‐methylation of aromatic organoboranes performed in two reaction media	1
Hydrogen isotope exchange labelling: A brief update	1
Automated synthesis of (R)‐[18F]MH.MZ on the iPhase Flexlab reaction platform	1
Site‐specifically radiolabeled nanobodies for imaging blood‐brain barrier penetration and targeting in the brain	1
Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET	1
Synthesis of [2H5]baricitinib via [2H5]ethanesulfonyl chloride	1
An efficient and general method for the synthesis of stable isotope deuterium labeled phthalate esters	1
A facile synthesis of isotope labeled acylcarnitines	1
A practical and environmentally friendly protocol for synthesis of α‐deuterated carboxylic acids	1
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Research on preparation and in vitro evaluation of the dendrimer–peptide nuclear acid conjugate for amplification pretargeting	1
Studies of hydrogen isotope scrambling during the dehalogenation of aromatic chloro‐compounds with deuterium gas over palladium catalysts	1
Efficient synthesis of carbon‐14 labeled metabolites of the strobilurin fungicide mandestrobin using biomimetic iron‐porphyrin catalyzed oxidation	1
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Nitrilase mediated mild hydrolysis of a carbon‐14 nitrile for the radiosynthesis of 4‐(7‐hydroxycarbamoyl‐[1‐14C‐heptanoyl]‐oxy)‐benzoic acid methyl ester, [14C]‐SHP‐141: A novel	0
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Synthesis and preclinical evaluation of a selective MET kinase positron emission tomography tracer	0
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High‐yielding, automated radiosynthesis of [11C]martinostat using [11C]methyl triflate	0
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Meet our advisors: Neil Vasdev	0
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Development of a high‐performance liquid chromatography method for rapid radiochemical purity measurement of [18F]PSMA‐1007, a PET radiopharmaceutical for detection of prostate cancer	0
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Abstracts of the 27th International Isotope Society (UK group) symposium: Synthesis and applications of labelled compounds 2018	0
Synthesis of N‐acetyl‐l‐aspartyl‐l‐glutamic acid; [3H]NAAG	0
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The synthesis of deuteriated tri‐tert‐butyl phosphine	0
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A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
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Synthesis of 13C‐labelled ω‐hydroxy carboxylic acids of the general formula HO213C‐(CH2)n‐CH2OH or HO2C‐(CH2	0
A synthesis of [14C]formamidine acetate	0
Meet the advisors: An interview with Gunnar Antoni	0
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A flow electrochemistry‐enabled synthesis of 2‐substituted N‐(methyl‐d)piperidines	0
Synthesis and spectroscopic characterization of 13C4‐labeled 4‐cyano‐2‐oxobutyraldehyde semicarbazone: A metabolite of nitrofurazone	0
An optimized radiosynthesis of [18F]DK222, a PET radiotracer for imaging PD‐L1	0
Automated radiolabeling and handling of 177Lu‐ and 225Ac‐PSMA‐617 using a robotic pipettor	0
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Facile synthesis of 14C‐nitrofurazone from 14C‐urea	0
Novel synthesis of 11C‐labeled imidazolines via Pd(0)‐mediated 11C‐carbomethoxylation using [11C]CO and arylborons	0
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Luminescence enhancement by deuterium	0
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Obituary	0
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Practical approaches to labelling terminal alkynes with deuterium	0
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Small‐scale two‐dimensional liquid chromatography for a preparative re‐purification of a highly labile tritium‐labeled compound	0
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Tritium hydrogen‐isotope exchange with electron‐poor tertiary benzenesulfonamide moiety; application in late‐stage labeling of T0901317	0
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Stable isotope synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	0
Meet our advisors: Bart Cornelissen	0
Synthesis of stable‐isotope‐labeled N‐(3‐dimethylaminopropyl)‐N′‐ethylcarbodiimide and N‐(3‐dimethylaminopropyl)‐N′‐ethylurea	0
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Synthesis of BI 894416 and BI 1342561, two potent and selective spleen tyrosine kinase inhibitors, labeled with carbon 14 and with deuterium	0
Synthesis of C‐14 labeled Rac‐(3R,2S)‐glycopyrronium bromide	0
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Synthesis of stable isotope‐labelled firocoxib	0
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Radiosynthesis and validation of [18F]fluoroestradiol in a Synthra plus research platform for use in routine clinical practice	0
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Carbon‐13 labeling of ibrutinib for human microdosing	0
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Preparation and biological evaluation of radioiodine‐labeled triphenylphosphine derivatives as mitochondrial targeting probes	0
Meet our advisors: Mathew Thakur	0
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Development of 11C‐labeled CRANAD‐102 for positron emission tomography imaging of soluble Aβ‐species	0
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Meet the advisors ‐ Suzy Lapi	0
A facile synthesis of precursor for the σ‐1 receptor PET radioligand [18F]FTC‐146 and its radiofluorination	0
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Meet our advisors: Dieter Muri	0
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Applications of radiolabeled antibodies in neuroscience and neuro‐oncology	0
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Featured Cover	0
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RO6807936 as a novel positron emission tomography (PET) radiotracer for in vitro and in vivo visualization and quantification of beta‐site amyloid precursor protein cleaving enzyme (BACE1) in the rode	0
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Wiley Young Scientist Awards were handed over at the 14th International Symposium on the synthesis on the Synthesis and Applications of Isotopically Labelled Compounds in Raleigh, USA	0
[18F]‐labeled positron emission tomography ligand for the histamine H4 receptor	0
Synthesis of trifold‐labeled versatile reagent [3,5‐13C2,4‐15 N]4‐phenyl‐1,2,4‐triazoline‐3,5‐dione	0
Meet our advisors: Jordi Llop	0
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Synthesis of carbon‐14 and stable isotope labeled Censavudine	0
[11C]CO2 BOP fixation with amines to access 11C‐labeled ureas for PET imaging	0
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Obituary for Prof. Rudolf Münze	0
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Meet our advisors: Crist N. Filer	0
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Radiosynthesis of novel N‐18F‐labeled 18F‐FHex‐α‐l‐Glu and 18F‐FHex‐β‐Glu	0
[18F]Fluoropyridine‐losartan: A new approach toward human Positron Emission Tomography imaging of Angiotensin II Type 1 receptors	0
Total synthesis of [13C2]‐labeled phytosiderophores of the mugineic and avenic acid families	0
Validation of a good manufacturing practice procedure for the production of [11C]AZD4747, a CNS penetrant KRASG12c inhibitor	0
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An improved radiosynthesis of [18F]FAraG, a PET radiotracer for imaging T‐cell activation	0
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Preliminary PET imaging of [11C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated11C‐carb	0
Imidazolium‐methylene‐trifluoroborate: A novel radioprosthetic group validated with preclinical 18F‐Positron Emission Tomography imaging of Prostate Specific Membrane Antigen in mice	0
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Meet our advisors—Matteo Zanda	0
Meet our Special Issue Editor: Jessica Bridoux	0
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The impact of zirconium‐89 solution formulation on the efficiency of [89Zr]Zr‐deferoxamine synthesis	0
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Automated radiosynthesis of [18F]CETO, a PET radiotracer for imaging adrenal glands, on Synthra RNplus	0
Synthesis of deuterium‐labeled CCR2 antagonist JNJ‐26131300, [4‐(1H‐indol‐ 3‐yl)‐piperidin‐1‐yl]‐{1‐[3‐(3,4,5‐trifluoro‐phenyl)‐acryloyl]‐piperidin‐4‐yl}‐acetic acid	0
Preparation of [1′‐13C]citric acid as a probe in a breath test to evaluate tricarboxylic acid cycle flux	0
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Evaluation and improvement of CuI‐mediated 11C‐cyanation	0
Photocatalyzed radiosynthesis of 11C‐phenylacetic acids	0
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Development of radiotracers for riboflavin transporter 3 imaging in diseases—A brief overview	0
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The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier	0
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Initial evaluation of 99mTc‐labeled anti‐carcinoembryonic antigen single‐chain fragment variable for micro‐single‐photon emission computed tomography imaging in mice with colorectal cancer	0
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14C‐radiolabeling of a new steroidal antiandrogen with a C‐18 angular methyl extension	0