Journal of Heterocyclic Chemistry

Article	Citations
Issue Information	89
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Novel ferrocene cyclopalladated compounds: Synthesis, and in‐vitro antitumor activity study	52
Synthesis and molecular modeling of some novel hydroxypyrone derivatives as antidermatophytic agents	48
Ultrasound‐promoted1,3‐dipolarcycloaddition of azomethine yields for synthesis of dispiropyrrolidineoxindole derivatives in hexyltriphenylphosphonium bromide as an ionic liquid,	34
Issue Information	32
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies	30
Synthesis and herbicidal activity of pyrimidyl‐1,2,4‐triazole derivatives containing aryl sulfonyl moiety	27
Synthesis of novel amide/amino acid functionalized pyrazolo[3,4‐b]pyridine derivatives; their anticancer activity and docking studies	27
Efficient synthesis of piperidine derivatives using dendrimer based catalytical pockets	26
A quick and easy access to a series of thiocyanated enaminones and 2‐iminothiazolones using PIDA under mild conditions	26
Novel angularly substituted [1,4]thiazino[3,4‐a]isoquinoline carboxylic acids prepared by cyclic imine‐cyclic anhydride reaction	24
NiO‐Nanoparticles as green catalyst for an efficient synthesis of 4‐iminopyrido[1,2‐a]pyrimidine fluorophores via one pot cyclization of α‐aminonicotinonitrile	24
Photoinduced 6π‐electrocyclization of 2,5‐dichlorothiophene containing benzofuranylacrylonitriles as efficient method for the generation of hydrogen chloride	24
Unprecedented, catalyst‐free, and rapid one‐pot, three‐component green synthesis of substituted 3‐hydroxy‐2‐oxindoles in water	23
Palladium‐Catalyzed Synthesis of Pyrrolo[1,2‐α]Pyrazines From N‐Phenacyl Pyrrole‐2‐Carbonitriles and Aryl Boronic Acids	23
A regiospecific fischer indole reaction with 3‐oxo‐24‐nor‐allobetulin	21
Synthesis and biological assessment of some fused Pyran derivatives	20
Synthesis of substituted 5‐aryl‐2,3‐dihydropyrazine 1,4‐dioxides based on condensation of N,N′‐(2,3‐dimethylbutane‐2,3‐diyl)bis(hydroxylamine) with various arylglyoxals	19
A synthetic strategy for the preparation of alkoxy‐functionalized bis‐1,2,4‐triazinyl‐2,6‐pyridines	18
Synthesis, antimicrobial activity, and molecular docking studies of new fused pyrimidinethiones	18
Synthesis, and reverse screening of 6‐(3,4,5‐trimethoxyphenyl)pyrimidine‐5‐carbonitrile derivatives as anticancer agents: Part‐II	18
Trifluorodiazoethane: A versatile building block to access trifluoromethylated heterocycles	17
[3+2] cycloaddition synthesis of new (nicotinonitrile‐chromene)‐based bis(pyrazole) hybrids as potential acetylcholinesterase inhibitors	17

Combination of N‐amino‐1,2,4‐triazole and 4‐hydroxy‐3,5‐dinitropyrazole for the synthesis of high performing explosives	17
Microwave‐Assisted One‐Pot Synthesis of 1,5‐Benzodiazepine Derivatives Using Novel ZnFe2O4.Cu(OH)2 Magnetic Nanocomposite as Heterogeneous Cataly	17
Facile access to 2‐amino‐4‐aryl‐5H‐chromeno[4,3‐b]pyridine‐3‐carbonitriles through a strategy of one‐pot Michael/cyclization reaction	17
Hybrid of the 1,2,3‐triazole nucleus and sesquiterpene skeleton as a potential antitumor agent: Hemisynthesis, molecular structure, Hirshfeld surface analysis, density functional theory, and in vitro	17
The applications of β‐keto amides for heterocycle synthesis	17
Synthetic Approaches Toward Imidazo‐Fused Heterocycles: A Comprehensive Review	16
Efficient preparation of (S)‐2‐(3,5‐dimethylphenyl)pyrrolidine via a recycle process of resolution	16
Solvent‐free Darzens condensation of 3‐chlorooxindoles with aryl aldehydes for diastereoselective construction of spiro‐epoxyoxindoles by grinding	16
One‐pot three‐component synthesis of novel chromeno[3,2‐c]pyridine‐1,9(2H)‐diones by using SnCl2⋅2H2O as catalyst	16
Catalyst‐free one‐pot three‐component rapid synthesis of polysubstituted pyrroles by liquid‐assisted grinding	16
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Thiazolidinedione‐Pyrimidine Hybrid as Potential Antidiabetic Agents and Their Cardioprotective Effect	15
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies	15
Synthesis and characterizations of some new selenolo[2,3‐b]quinoxaline derivatives	15
Cycloaddition or Metathesis: Selectivity in a Series of Indole‐2,3‐Quinodimethane Derivatives	15
Discovery of Promising Sulfadiazine Derivatives With Anti‐Proliferative Activity Against Tumor Cell Lines	15
An approach for the diastereoselective synthesis of (R)‐(+)‐methyl pipecolate and (+)‐dextro‐erythrophacetoperane from (S)‐(−)‐methylbenzylamine	15
New metal free organic dyes incorporating heterocyclic Benzofuran core as conjugated spacer: Synthesis, Opto‐electrochemical, DFT and DSSC studies	15
Synthesis of 1,3‐oxazepine derivatives via tandem reaction of 5‐benzylidine Meldrum's acids with TosMIC in presence of potassium carbonate	14
Visible‐light photoredox catalyzed synthesis of tetrahydrobenzofuranone: Oxidative [3 + 2] cycloaddition of dicarbonyl and alkene	14
New edaravone analogs incorporated with N‐benzylthiazole moiety: Multistep chemical synthesis, in vitro cytotoxicity with pRIPK3 inhibitory activities, and molecular docking	14
Synthesis and evaluation of the biological activities of novel hybrid isoindol‐1,3‐dione containing an aziridine unit	14
Iron‐catalyzed construction of cyanomethylated thiohydantoins by cross‐dehydrogenative C(sp3)‐C(sp3) coupling	14
Synthesis of novel Schiff bases as stable enol‐imine‐containing diazene bonds and pyrimidines using trimethinium salts	13
Long alkoxy substituted N2S2 porphyrins for liquid crystalline property	13
Saccharin‐catalyzed multicomponent cascade reactions for the synthesis of 1,2,3,4,6‐pentasubstituted piperidines	13
Overview of Hydroxychloroquine and Remdesivir on severe acute respiratory syndrome coronavirus 2 (SARS‐CoV‐2)	13
Synthesis of Novel 6H‐Furo[3,2‐e]Indole Derivatives via One‐Pot Three Component Reactions	13
Design, synthesis, antimicrobial evaluation, and in‐silico studies of some 4‐thiazolidinone hybrids bearing coumarin and pyridine moieties	13
An efficient organopromotor L‐arginine facilitated synthesis of thiazolo[3,2‐a]pyrimidine derivatives in EtOH:H2O solvent	13
Synthesis and bioactivity evaluation of 5‐trifluoromethyl‐1H‐pyrazole‐4‐carboxamide derivatives as potential anticancer and antifungal agents	12
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Synthesis of arylidene‐based benzoxazine derivatives as promising antimicrobial materials	12
Synthesis and Application of Azide‐Incorporated Copper‐Chelating Peptides for Efficient Click Conjugation Reaction	12
Design, synthesis, and pesticidal activities of novel pyrimidin‐4‐amine derivatives containing trifluoroethyl sulfide moiety	12
Manipulating sensitivities of planar oxadiazole‐based high performing energetic materials	12
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Thermal [2+2] Cycloaddition of Dihydropyrroles and Dimethyl Acetylenedicarboxylate	11
Research progress of oxazole derivatives in the discovery of agricultural chemicals	11
Novel pyrazole‐biphenyl‐carboxamides for SARS‐CoV2 entry‐level restriction and microbial infections	11
Imidazo[1,2,4]triazolone and fused imidazo[1,2,4]triazolone derivatives: Synthesis, in vitro anticancer screening, CDK2 inhibitory activity, and molecular modeling studies	11
Utility of pyrrole‐2‐thioacetohydrazide in synthesis of new heterocyclic compounds with promising antimicrobial activities and molecular docking studies	11
A Simple, Economical, and Green Protocol for the Synthesis of Benzyl‐Quinoline Analogues by Grinding	11
Convenient synthesis and antibacterial evaluation of new bipyrazolyl and pyrazolopyridazine derivatives utilizing 4‐acetyl‐5‐methyl‐N‐phenyl‐1‐(p‐tolyl)‐1H‐p	10
Investigation of some new main group metal complexes of hydrazine and 2‐mercaptopyridine‐3‐carboxylic acid mixed–ligands	10
Arylhydrazine salt‐selenium: A novel and efficient reagent system for arylselenenylation of unprotected uracil and its derivatives	10
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Synthesis and biological evaluation of baloxavir marboxil analogs for the treatment of influenza A (H1N1) virus	10

Neat multicomponent assembly of highly functionalized Acenaphtho[1,2‐b]pyrroles, in vitro evaluation for antioxidant and cytotoxic activities	9
Synthesis, characterization and crystal structure of some novel partially hydrogenated isoquinolines and their fused heterocyclic systems	9
Synthetic strategies of phenazine derivatives: A review	9
Kilogram synthesis of pinoxaden	9
Design, synthesis, biological evaluation, and molecular docking studies of some novel N,N‐dimethylaminopropoxy‐substituted aurones	9
Toward understanding the regioselectivity of the one‐pot reaction of phenylene diamines with aldehydes and cyclopentadiene (Povarov reaction). Combined experimental and theoretical approaches	9
Reactivity of pyrimidinylphosphazenes with acetylenic esters: Competitive [4 + 2] and [2 + 2] tandem cycloaddition or retro‐cycloaddition approaches	9
CuI–Zn(OAc)2 Catalyzed Selective CC Bond Cleavage of 1,3‐Diketones/β‐Ketoester for the Formation of Quinazolin‐4(3H)‐Ones: A Fast, Solvent‐Free, Syn	9
Visible‐Light Induced Rose Bengal Photocatalyzed One‐Pot Environmentally Sustainable Multicomponent Synthesis of Substituted Pyrazolo[3,4‐b]Quinolin‐5‐Ones	8
Facile synthesis and antimicrobial activity of bis(fused 4H‐pyrans) incorporating piperazine as novel hybrid molecules: Michael's addition approach	8
Recyclization of 3‐substituted‐6,8‐dimethylchromones with some heterocyclic enamines: Spectroscopic, quantum calculations (HOMO–LUMO, MEP, NLO), biological evaluation, and ADME investigation	8
Multicomponent synthesis of spiro 1,3,4‐thiadiazolines with anticancer activity by using deep eutectic solvent under microwave irradiation	8
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Regio Selective Synthesis of Pyrazole Derivatives of 5‐Chloro‐2‐Methoxy Phenyl Hydrazide and Their Biological Evaluation	8
An operationally simple, one‐pot, convenient synthesis, and in vitro anti‐inflammatory activity of some new spirotriazolotriazine derivatives	8
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Synthesis and Characterization of Benzo[6,7]Cyclohepta[1,2‐b]Pyrazolo[4,3‐e]Pyridines	8
Design, Synthesis, In Vitro Evaluation of New Tetrahydrooxazolo [5′,4′:4,5]Pyrimido[1,2‐a]Azepinone Derivatives as Anticancer Agents	8
Synthesis, antimicrobial activity, and in silico studies of fluoroquinolones bearing 1,3,4‐oxadiazolyl‐triazole derivatives	8
Synthesis of Alpha‐Acyloxy‐(1,2,5‐Oxadiazole‐2‐Oxide) Carboxamides via Passerini Multicomponent Reaction. Evaluation of Nitric Oxide‐Releasing and Anti‐Proliferative Properties	8
Direct synthesis of β2,3‐amino acid from β‐hydroxycarbamides: Implication in the synthesis of azumamide analogs and conformational analysis	8
Radical synthesis of dihydropyrano[2,3‐c]pyrazoles using acridine yellow G as a photo‐induced electron transfer photocatalyst	8
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Green Construction of Novel 3‐(Benzo[d][1,3]dioxol‐5‐yl)‐1,8‐naphthyridin‐2‐yl)amino)quinazoline‐2,4(1H,3H)‐dione and Phenyl‐[1,2,4]triazolo[4,3‐a][1,8]naphthyridine and Their An	8
Synthesis of new thiazine and thiazole derivatives via cyclization reactions; investigating their electronic properties and determination of antioxidant properties	8
Dimethyl‐1,4‐Dithiines From 2‐Chloroprop‐2‐Enylisothiouronium Salt in KOH/Hydrazine Hydrate Medium: Experiment and Quantum Chemical Study	7
Formation of anti‐Bredt‐type azabicyclo[4.2.0]octene frameworks through photochemical intramolecular [2+2] cycloaddition between indole and a distal double bond of allene	7
Facile synthesis and anticancer activity of tetrazolyl‐benzothiazole derivatives	7
Polycyclic Dicationic Heteroaromatic Compounds From One‐Step Multiple Condensation Reactions: Synthesis and Reactivity	7
Synthesis, characterization, anti‐proliferative evaluation, and molecular docking study of some new N‐(1, 3‐dioxoisoindolin‐4‐yl)acetamide derivatives	7
Recent developments in synthetic strategies and pharmacological outcomes of synthetic xanthine oxidase inhibitors: A comprehensive review	7
A simple and efficient approach for the clickability of super‐bulky aryl azides	7
An efficient and green synthesis of multi‐heteroatom heterocycles via a three components reaction in acetic acid/aqueous condition	7
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Efficient synthesis and biological evaluation of some new series of pyridine derivatives: Promising and potent new class of anticancer agents	7
Oxidative cross dehydrogenative coupling directed carbamates synthesis using Cu(II) pincer complex as active catalyst under mild reaction condition	7
Synthesis of Terminal Alkenylindolines via Rhodium‐Catalyzed Direct CH Alkenylation With Alkenyl Borates	7
N‐Azidoethyl azoles through N‐alkylation under highly harmonized reaction conditions: Synthesis, characterization, and complexation as energetic coordination compounds	7
Synthesis and Cellular Evaluation of Some Oxepino‐ and Pyranoxanthone Derivatives as Antitumor Agents: A Comparative Study	7
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An efficient synthesis of new 3,5‐bis(2‐arylthiazol‐4‐yl)‐1,2,4‐oxadiazole derivatives and their antimicrobial evaluation	7
Ultrasound promoted three‐component synthesis of dihydroindeno[1,2‐b]pyrrole derivatives	7
An elegant and efficient synthesis of heterocycles integrated with bis‐N‐acyl pyrazoline and bis‐1, 2, 3‐triazole via a green synthetic methodology	7
Medicinal perspective of quinazolinone derivatives: Recent developments and structure–activity relationship studies	7
Ni‐Ferrite an efficient catalyst for synthesis of 3‐aryl substituted isoxazole‐5‐carboxylic acids via one‐pot multicomponent reaction	7
Synthesis of Benzofuran‐Based Hybrid Molecules: Molecular Docking and Antibacterial Activity Against Pseudomonas aeruginosa	7
Synthesis a group of 5(6)‐substituted benzimidazole Zn(II) and Co(II) complexes and investigation their cytotoxic and antimicrobial activities	7
Study on halogen promoted cyclization of 2‐alkynylthiobenzimidazoles	7
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Synthesis, Photophysical Properties and Cytotoxic Activities of Isoxazole‐Containing Difluoroboron Complexes	7
Synthesis of various functionalized 2H‐azirines: An updated library	7
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A Comprehensive Report on Environmentally Benign Synthesis of 1, 8‐Dioxo‐Octahydroxanthene Derivatives	7
The synthesis of novel 2, 3‐disubstituted 1,6‐dihydropyrrolo[2,3‐g]indazole derivatives via one‐pot three component reactions	6
Design, Synthesis of Novel Pyrimidine Derivatives Containing Alkenyl Moieties With Herbicidal Activities	6
Synthesis and biological evaluation of 3‐hydroxypyrazoles as aquaporin 9 inhibitors	6
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Synthesis and anticancer activity of cinnoline sulphonamides and 4‐heteroyclic derivatives: Cross‐coupling approach	6
Hantzsch‐like reaction of isoquinoline‐1‐acetonitrile in synthesis of 4H‐pyrido[2,1‐a]isoquinolines with antibacterial evaluation	6
Synthesis of new 1,4‐ and 1,5‐disubstituted N‐ethyl acetate and N‐α‐butyro‐γ‐lactone alkylimidazole derivatives as N‐acylhomoserine lactone analogs	6
Catalyst‐free one‐pot synthesis of quinoline tethered α‐amino ketones by multicomponent reactions	6
Pyranoquinolone derivatives: A potent multi‐targeted pharmacological scaffold	6
Highly efficient microwave‐assisted solvent free sequential one‐pot multicomponent synthesis of novel 2‐hydroxy indenopyridin‐5‐ones and mechanismic computational study	6
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Design, synthesis, and biological evaluation of 1,4,7,8‐tetrahydro‐5H‐furo[3,4‐b]pyrazolo[4,3‐e]pyridin‐5‐one‐based azo dyes	6
Green multicomponent approach to novel 5‐[(2H‐Pyran‐3‐yl)(aryl)methyl]‐1,3‐dimethylpyrimidines	6
A selective chromone‐based colorimetric chemosensor for detecting Cu2+ in near‐perfect aqueous solution and test kit	6
Base promoted CuFe2O4 catalyzed one‐pot synthesis of 3,5‐diaryl‐1H‐pyrazoles	6
Retraction statement: Design and synthesis of a bismethylsulfanyl‐steroid‐azetyl butanol derivative from 2‐nitroestradiol	6
BimetallicCoCeO2oxide nanoparticles: An efficient and reusable heterogeneous catalyst for the preparation of2‐amino‐3‐cyano‐4H‐pyran derivatives	6
Synthesis and antiviral activity of novel imidazo[2,1‐b]thiazoles coupled with morpholine and thiomorpholines	6
A review on advances in synthetic methodology and biological profile of spirothiazolidin‐4‐ones	6
Study on antitumor activity of parthenolide C‐14 derivatives	6
Synthesis and anticancer activity of some thiophene, thienyl‐thiazole, and thienyl‐benzofuran analogues	6
Novel oxadiazole functionalized pyridopyrimidine derivatives; their anticancer activity and molecular docking studies	6
A search for antiinflammatory therapies: Synthesis, in silico investigation of the mode of action, and in vitro analyses of new quinazolin‐2,4‐dione derivatives targeting phosphodiesterase‐4 enzyme	6
Oriented synthesis and insecticidal activities of novel meta‐diamide scaffolds incorporating with 1,2,4‐triazole moiety	5
Regioselective synthesis of fused pyrimidines and quinazolines linked to Phenoxy‐N‐arylacetamide moieties as novel hybrid molecules via Biginelli‐like reaction	5
A high‐yielding protocol for the synthesis of 4,5‐diarylpyrimidin‐2‐amine derivatives from chalcones	5

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One‐Pot, Multicomponent Synthesis of 1,3‐Oxazin‐One and Evaluation of Their Potential Antioxidant Activities	5
Synthesis, antiinflammatory, and cytotoxic activity of novel pyrazolo[4,3‐c][2,1]benzothiazine 4,4‐dioxide derivatives	5
Design, synthesis, antifungal activity, and molecular docking of novel trifluoromethyl pyrimidine derivatives containing 1,3,4‐oxadiazole and thioether moieties as potential succinate dehyd	5
N‐Methoxy Pyrazole‐4‐Carboxamide Derivatives: Synthesis, Spectral Analyses, Antifungal Activity, In Silico Molecular Docking, ADMET, and DFT Studies	5
Synthesis and Cancer Cell Cytotoxicity of 6‐, 7‐, or 8‐Substituted 2‐(Hetero)aryl‐4‐(4‐(Hetero)aryl‐2‐Oxobut‐3‐en‐1‐Ylidene)Benzothiazepanes	5
Preparation of chiral DMAP derivatives and investigation on their enantioselective catalytic activity in benzazetidine synthesis and kinetic resolutions of alcohols	5
Synthesis, physico‐chemical characterization and theoretical exploration of some 2,4,5‐triaryl imidazole derivatives	5
Chemoselective direct amidation of fatty acids with furfurylamine without coupling reagents in reversed micellar microenvironment	5
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Baylis–Hillmanadducts as an important synthon for the synthesis of α‐carbolinone and α‐carboline derivatives	5
Organocatalytic Enantioselective Synthesis of Oxindole‐4‐Aminopyrazolone Derivatives via Mannich Reaction of 3‐Substituted Oxindoles With Pyrazolinone Ketimines	5
Synthesis, characterization, and photophysical properties of some new thieno[2,3‐b]pyridines bearing phenylethenyl moiety	5
A convenient and efficient process for the synthesis of 9‐aryl‐6,9‐dihydro‐1H‐pyrazolo[3,4‐f] quinoline‐8‐carbonitrile and 1‐aryl‐1,4‐ dihydrobenzo[f]quinoline‐2‐carbon	5
Synthetic, spectroscopic, and computational investigations of readily accessible 2‐phenyl‐3‐alkylbenzoxazaboroles	5
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Synthesis, anticancer evaluation and in silico studies of novel N‐substituted arylidenethiazolidine‐2,4‐dione derivatives as adenosine monophosphate‐activated protein kinase activators	5
An efficient synthesis of 4,6‐diarylnicotinonitrile‐acetamide hybrids via 1,2,3‐triazole linker as multitarget microbial inhibitors	5
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Pyrazolo[3,4‐d]pyrimidine‐based scaffolds as antibacterial agents: Synthetic strategies, reactions, and in vitro biological evaluation	5
An eco‐efficient new path of mortar pestle grinding approach for the construction of methanol and ethylthio substituted pyridines with in silico studies	5
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β‐Nitrostyrenes as a valuable precursor for the synthesis of β‐aryl‐γ‐lactam and 2‐oxo‐1,2‐dihydroquinoline derivatives	5
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Substrate‐controlled chemoselective synthesis of 1‐sulfonylquinazoline‐2,4(1H,3H)‐diones and 2‐sulfonamidobenzonitriles	5
Design, enantioselective synthesis, and antiviral activities against potato virus Y of axially chiral thiazine derivatives	5
Green synthesis and biological activity investigation of new derivatives of spiroisatins	5
(±)‐cis‐4a‐alkyl‐1,3,4,4a,9,9a‐hexahydro‐2H‐carbazol‐2‐ones by domino nitro reduction‐aza‐Michael addition to enones	5
A Green Approach for the Synthesis of 5,6‐Dihydropyrimido[4,5‐d]Pyrimidines From N‐Uracil Amidines in Water	5
Regioselective synthesis and computational calculation studies of some new pyrazolyl‐pyridine and bipyridine derivatives	5
New thieno[2,3‐d]pyrimidine derivatives as EGFRWT and EGFRT790M inhibitors: Design, synthesis, antiproliferative activities, docking studi	5
Unusual impurity formation during the process development of Olsalazine sodium leads to a new efficient and economical synthesis of tricaine mesylate	5
Practical synthesis of (S)‐pyroglutamic acid	5
One‐pot three‐component reaction; synthesis of new symmetrically bridge 4,4′‐(1,4‐phenylene)di‐pyrimidines under solvent free conditions	5
Synthesis, crystal structure, and DFT study of 4‐(2‐Chlorobenzyl)‐1‐(furan‐2‐yl)‐[1,2,4]triazolo[4,3‐a]quinazolin‐5(4H)‐one	5
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